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5-methyl-2-{2-[(3-propylpyrrolidin-1-yl)methyl]phenyl}-6-(trifluoromethyl)-3,4-dihydropyrimidin-4-one
(5S)-5-({[(2,3-dimethyl-1H-indol-7-yl)methyl](pyridin-4-ylmethyl)amino}methyl)pyrrolidin-2-one
methyl 4-({3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)benzoate
7-(cyclobutylmethyl)-2-(4-methoxybenzoyl)-2,7-diazaspiro[4.5]decan-6-one
3-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-3-methyl-1-(3-oxo-1,3-dihydro-2-benzofuran-5-yl)urea
N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-3-(trifluoromethyl)pyridin-2-amine
2-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-1,3-thiazole-4-carboxamide
ethyl 4-[5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carbonyl]piperazine-1-carboxylate
dimethyl({2-[2-(1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidin-4-yl)-1H-imidazol-1-yl]ethyl})amine
(1S,5R)-3-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(4-ethylphenyl)methyl]-N,2,5-trimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(1,3-thiazol-2-ylmethyl)piperidine
1-(furan-3-ylmethyl)-4-[5-(oxan-2-yl)thiophen-2-yl]-1H-1,2,3-triazole
3-(4-{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}piperazin-1-yl)propanamide
N-(1-{10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}pyrrolidin-3-yl)acetamide
2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-5-methylpyridine
8-(1,8-naphthyridine-2-carbonyl)-1-oxa-8-azaspiro[4.5]decane
1-methyl-N-(2-methylpropyl)-5-oxo-N-(3-phenylprop-2-yn-1-yl)pyrrolidine-3-carboxamide
N-[4-(2-fluorophenoxy)phenyl]-1-(3-hydroxypropanoyl)piperidine-4-carboxamide
1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-4-(4-methoxyphenoxy)piperidine
2-{1-cyclohexyl-4-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
(3aS,6aS)-2-cyclopentyl-5-(5-methylthiophene-2-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[5-(methoxymethyl)thiophene-2-carbonyl]-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[(benzyloxy)methyl]-1H-1,2,3-triazole
2-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-5-methoxypyrimidine
(1S,5R)-3-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-({3-methyl-7-[2-(piperidin-1-yl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1-phenylmethanesulfonamide
1-(cyclohexylmethyl)-3-(2-fluoropyridin-3-yl)urea
1-[2-(1-benzylpiperidin-4-yl)ethyl]-3-{2-methyl-2H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}urea
N-[3-(cyclohexylsulfanyl)propyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
5-{[3-(3-methylphenoxy)azetidin-1-yl]methyl}-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
2-[4-(2H-1,3-benzodioxol-4-ylmethyl)-1-[(4-ethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
(2S)-2-(methoxymethyl)-N-[3-(1H-pyrazol-5-yl)phenyl]pyrrolidine-1-carboxamide
3-methyl-5-{6-[(piperidin-4-yl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridin-2-amine
1-(2-chlorophenyl)-3-(1-{1-[3-(1-methylcyclopropyl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
4-(7-butoxy-2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)benzoic acid
2-{4-[2-(2,4-difluorophenyl)acetyl]piperazin-1-yl}-1-(piperidin-1-yl)ethan-1-one
N-(1-benzothiophen-5-ylmethyl)-3-(4-methyl-1,3-thiazol-5-yl)propanamide
2,6-dimethyl-N-(2-oxopiperidin-3-yl)quinoline-4-carboxamide
1-(oxan-2-ylmethyl)-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
(1R,5R)-6-(2-methoxyethyl)-3-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-3,6-diazabicyclo[3.2.2]nonane
1-{[1-(4-butylphenyl)-1H-pyrazol-4-yl]methyl}azetidin-3-ol
1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(1H-indol-1-yl)ethan-1-one
2-(2,6-dioxo-1,3-diazinan-1-yl)-N-(oxolan-2-ylmethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]acetamide
4-methyl-1-{2-[4-phenyl-5-(1,3-thiazol-2-yl)-1H-imidazol-1-yl]ethyl}-1H-1,2,3-triazole
4-(2-methoxyphenoxy)-1-(2-methyl-1,3-thiazole-5-carbonyl)piperidine
N-[(3R,4S)-1-(2-amino-2-methylpropyl)-4-propylpyrrolidin-3-yl]-2,2-dimethylpropanamide
methyl({[2-(propylsulfanyl)pyrimidin-5-yl]methyl})(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amine
N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1,3-benzothiazole-6-carboxamide
8-(5,6-dimethylpyrimidin-4-yl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one