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2-methanesulfonyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(2-methylpropyl)acetamide
N-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-N-methyl-2-(1-oxo-1,2-dihydroisoquinolin-2-yl)acetamide
2-amino-3-ethyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-[(3S,4R)-3-methanesulfonamido-4-propylpyrrolidin-1-yl]-N,N-dimethylpyridine-3-carboxamide
3-(3-hydroxy-1,2-oxazol-5-yl)-1-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}propan-1-one
3-(1H-imidazol-2-yl)-1-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]piperidine
2-(dimethylamino)-2-(3-methylphenyl)-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}(cyclopropylmethyl)amine
1-[2-methoxy-4-({[2-(2-methylphenyl)ethyl]amino}methyl)phenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-3-(2-methoxyphenyl)propanamide
1-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-4-methoxy-3-methylbenzamide
N-ethyl-4-({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)piperidine-1-carboxamide
methyl (2S,4R)-4-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzamido}-1-(1-ethylpiperidin-4-yl)pyrrolidine-2-carboxylate
8-(2-methylpyrimidin-4-yl)-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one
5-[5-(2-chlorophenyl)furan-2-yl]-2-ethyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
2-[2-({4-chloro-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)ethyl]-3,4-dihydroquinazolin-4-one
1-(2,2-dimethylpropyl)-4-({[4-(pyrimidin-2-yloxy)phenyl]methyl}amino)pyrrolidin-2-one
1-(2-methyl-1,3-thiazole-4-carbonyl)-3-{[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[4-(1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
(4aS,8aR)-1-(3-methoxypropyl)-6-(4-methylpiperazine-1-carbonyl)-decahydro-1,6-naphthyridin-2-one
3-[({1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-3-yl}oxy)methyl]pyridine
1-[(2-fluorophenyl)methyl]-N-[3-(1H-imidazol-1-yl)-1-phenylpropyl]-1H-1,2,3-triazole-4-carboxamide
1'-(quinoxalin-2-yl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
2-chloro-N-(1-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
3-{[8-(6-methylpyridin-2-yl)-1,8-diazaspiro[4.5]decan-1-yl]methyl}phenol
1-[1-(4-phenylpiperidin-1-yl)propan-2-yl]-1H-1,3-benzodiazole
2-(4-{1-[(3-methylpyridin-2-yl)methyl]-1H-1,2,3-triazol-4-yl}phenoxy)pyrimidine
phenyl (7S,9aR)-7-[(benzyloxy)methyl]-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
N-(2-hydroxyethyl)-4-{[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl](methyl)amino}pyridine-2-carboxamide
6-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-N,N-dimethylpyrazin-2-amine
1-[(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octan-8-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
9-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
3,5-dimethyl-N-[2-methyl-1-(morpholin-4-yl)propan-2-yl]-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
4-[3-(furan-2-yl)-1H-pyrazol-1-yl]-1-(1,2-oxazole-3-carbonyl)piperidine-4-carboxylic acid
1-cycloheptyl-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-(methoxymethyl)-N-(1,2-oxazol-3-ylmethyl)-1H-pyrazole-4-carboxamide
2-[4-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetyl)-5-methyl-2-oxopiperazin-1-yl]benzonitrile
7-[(2-phenoxyethyl)sulfamoyl]-N-(propan-2-yl)-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)amine
2-{1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]pyrrolidin-2-yl}ethan-1-ol
2-(2-fluoro-5-methoxyphenyl)-4-(1H-imidazol-1-ylmethyl)-5-methyl-1,3-oxazole
8-methyl-N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]imidazo[1,2-a]pyridine-2-carboxamide
4-{[(3R,4S)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]methyl}-1-methyl-1H-pyrrole-2-carbonitrile
N3-tert-butyl-4-oxo-1-(propan-2-yl)-N5-(thiophen-3-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
7-(5-phenylpentanoyl)-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(1S,5R)-6-(2,3-difluoro-6-methoxybenzoyl)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
4-ethyl-3-{[1-(2-methoxy-6-methylbenzoyl)piperidin-4-yl]methyl}-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(1R,3R)-3-aminocyclopentyl]-1,2,3,4-tetrahydroquinoline-8-carboxamide
2-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}(2-hydroxyethyl)amino)ethan-1-ol