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1-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2,3-dimethylphenyl)piperazine
[3-(2-methoxyethyl)-1-(trimethyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]methanol
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-(4-fluoro-2-methylphenyl)acetamide
5-fluoro-2-[1-(1-methyl-1H-indole-3-carbonyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
4-(pyridin-4-yl)-N-[1-(thiophen-3-yl)propan-2-yl]pyrimidin-2-amine
methyl[(2-methyl-1,3-thiazol-5-yl)methyl][(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]amine
(3S)-1-({1-[1-(2-methylquinolin-4-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)pyrrolidin-3-ol
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]piperidine
N-[(3,4-dimethoxyphenyl)methyl]-N,1-dimethyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[(5-{[2-(3-methoxyphenyl)azetidin-1-yl]methyl}thiophen-2-yl)methyl]piperidine
N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]quinoline-3-carboxamide
(1R,7S)-6-(4,4-difluoropiperidine-1-carbonyl)-3-(pyridin-3-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
2-(dimethylamino)-N,4-dimethyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}pyrimidine-5-carboxamide
4-{3-[4-(1-methylpiperidin-4-yl)piperidine-1-carbonyl]phenyl}phenol
1-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(phenylsulfanyl)ethan-1-one
3-{[2-(1,3-benzothiazol-2-yl)pyrrolidin-1-yl]methyl}pyridin-2-amine
2-methyl-6-(1-{2-[(2-methylphenyl)sulfanyl]acetyl}piperidin-3-yl)-3,4-dihydropyrimidin-4-one
(3S,4S)-1-(1-benzothiophene-2-carbonyl)-4-(morpholin-4-yl)pyrrolidin-3-ol
4-{4-[1-(3-phenoxypropyl)-1H-imidazol-2-yl]-1H-1,2,3-triazol-1-yl}piperidine
5-{1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidin-4-yl}-5-(pyridin-3-yl)imidazolidine-2,4-dione
N-(2-methoxyethyl)-3-[(1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidin-4-yl)oxy]benzamide
N-[(3R,4S)-1-(2-ethoxyethyl)-4-(propan-2-yl)pyrrolidin-3-yl]-2-methoxy-2-methylpropanamide
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}furan-2-carboxamide
N-(2,2-diphenylethyl)-3-{2-[(4-methylphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
1-cyclopentyl-4-{4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine-1-carbonyl}pyrrolidin-2-one
9-(6-aminopyrimidin-4-yl)-2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carboxamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
2-methyl-4-{3-[3-(2-methylpiperidin-1-yl)azetidine-1-carbonyl]phenyl}butan-2-ol
N-methyl-4-(1H-pyrazol-1-yl)-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
2-(4-chlorophenyl)-4-[2-methyl-2-(morpholin-4-yl)propyl]morpholine
2-(2,5-dioxoimidazolidin-1-yl)-N-[3-(4-methylbenzenesulfonamido)propyl]acetamide
(1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-3-propylpiperidin-3-yl)methanol
(3R,4R)-1-[4-(difluoromethoxy)benzoyl]-4-ethylpiperidine-3,4-diol
6-[(3-methoxyphenyl)methoxy]-4-(1-methylpiperidin-4-yl)-1-(2-phenylethyl)-1,4-diazepan-2-one
N,3,5,7-tetramethyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-1H-indole-2-carboxamide
N-cyclopropyl-4-{2-methyl-4-[(3-methylphenyl)methyl]-3-oxopiperazin-1-yl}pyridine-2-carboxamide
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-chloro-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
N4-[2-(4-ethoxyphenoxy)ethyl]-N2,4-dimethylpyrimidine-4,6-diamine
(5-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}furan-2-yl)methanol
(2S)-N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-(1H-1,2,4-triazole-5-carbonyl)pyrrolidine-2-carboxamide
2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-[2-(methylsulfanyl)benzoyl]piperidine
(3S)-4-{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,3-dimethylpiperazin-2-one
N-[(1-benzylpiperidin-4-yl)methyl]-N-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
11-(2,4-dimethoxy-3-methylphenyl)-4,6,10,12-tetraazatricyclo[7.3.0.03,7]dodeca-1,3(7),8,10-tetraen-5-one
1-methyl-N-[2-(quinolin-8-yloxy)ethyl]-1H-indole-6-carboxamide
4-(4-fluorophenyl)-1-[2-(pyrrolidin-3-yl)benzoyl]-1,2,3,6-tetrahydropyridine
N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)ethane-1-sulfonamide
5-[2-(phenylsulfanyl)ethyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid