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2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-1-{5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethan-1-one
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]pyrimidin-2-amine
8-[2-(trifluoromethyl)-1H-1,3-benzodiazole-5-carbonyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
1-(propan-2-yl)-N-[1-(pyrazin-2-yl)propan-2-yl]piperidine-4-carboxamide
(4aR,7aS)-1-acetyl-4-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1-ethyl-1,2-dihydropyridin-2-one
7-(2-ethoxypyridine-3-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]oxane-4-carboxamide
3-[(3R,4S)-1-{[2-(difluoromethoxy)phenyl]methyl}-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
3-(1H-imidazol-2-yl)-1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}piperidine
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[3-(pyridine-2-carbonyl)piperidin-1-yl]ethan-1-one
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-(5-chloropyridine-3-carbonyl)piperidine-4-carboxylic acid
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-6-(pyrrolidine-1-carbonyl)pyrazin-2-amine
N-(3-methylphenyl)-3-[1-(thian-4-yl)piperidin-4-yl]propanamide
2-[3-(2-ethylphenoxy)azetidin-1-yl]quinoline
N-cyclopropyl-5-(1-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}pyrrolidin-2-yl)thiophene-2-carboxamide
N-[1-benzyl-6-(propan-2-yloxy)-1H-indazol-3-yl]-2,5-dimethyl-1,3-oxazole-4-carboxamide
4-{2-[(2-methyl-1H-imidazol-1-yl)methyl]phenyl}-4H-1,2,4-triazole
N-[2-(3-fluorophenyl)ethyl]-2-[4-(4-{[3-(pyridin-4-yl)propyl]amino}piperidin-1-yl)phenyl]acetamide
4-{2-propyl-3H-imidazo[4,5-b]pyridin-3-yl}-1-(2,3,4-trimethoxybenzoyl)piperidine
1-ethyl-3-(naphthalen-1-ylmethyl)-8-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[3-(4-{[2-(hydroxymethyl)phenyl]methyl}piperazin-1-yl)-3-oxopropyl]acetamide
1-{2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}-2-(pyridin-4-ylsulfanyl)ethan-1-one
4-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-2-(trifluoromethyl)morpholine
1-methyl-4-{4-[2-(5-methylfuran-2-yl)-1H-imidazol-1-yl]phenoxy}piperidine
3-[(1-methyl-1H-1,2,3-benzotriazol-5-yl)formamido]-N-(3-methylphenyl)propanamide
N-[2-(3,5-difluorophenyl)ethyl]-2-methylpyrimidine-5-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[1-(1H-1,2,4-triazole-5-carbonyl)piperidin-4-yl]propanamide
N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]-2-(pyridin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-(6-methoxynaphthalene-2-carbonyl)-1-(1-methyl-1H-pyrazole-5-carbonyl)piperidine
11-[(benzyloxy)methyl]-4,6,10,12-tetraazatricyclo[7.3.0.03,7]dodeca-1,3(7),8,10-tetraen-5-one
N-[3-(diethylamino)propyl]-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
2-methyl-7-(5-phenoxyfuran-2-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-2,4,7-trimethyl-1H-indole
2-[(3,5-difluorophenyl)methyl]-8-[(1-ethyl-1H-imidazol-5-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
(1R,5R)-6-[(2-ethoxyphenyl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
N-[(2R)-1-{2-[2-(1H-imidazol-4-yl)ethyl]-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}-1-oxopropan-2-yl]acetamide
5-{[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-2-(pyrrolidin-1-yl)-1,3-thiazole
N-[1-(1,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-(3-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)thiophene-2-carboxamide
1-(carbamoylmethyl)-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}piperidine-4-carboxamide
3-(2-fluorophenyl)-1-methyl-3-{2-oxo-2-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]ethyl}pyrrolidine-2,5-dione
1-{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidine-3-carboxamide
4-[(1S,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]-6-ethyl-2-(1-methyl-1H-pyrazol-4-yl)quinoline
(2S)-N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrrolidine-2-carboxamide
5-(2-methylpropyl)-1'-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-[1-(2-methylphenyl)-1H-pyrazol-4-yl]-N-[1-(pyridin-4-yl)propan-2-yl]pyrimidin-2-amine
2-(3-fluorophenoxymethyl)-N-[1-(2-methoxyphenyl)ethyl]-N-methyl-1,3-oxazole-4-carboxamide
N-(4-methylpyridin-3-yl)-2-{4-[4-(1H-1,2,4-triazol-1-yl)butanoyl]morpholin-3-yl}acetamide
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[2-(morpholin-4-yl)butyl]acetamide