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4-fluoro-2-({methyl[1-(pyridin-4-yl)ethyl]amino}methyl)phenol
7-ethyl-3-methyl-1-[3-(1H-pyrazol-5-yl)piperidine-1-carbonyl]-5H,6H,7H,8H-imidazo[1,5-a]pyrazin-8-one
4-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]pyridine-2-carboxylic acid
N-(1-methylpiperidin-3-yl)-5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-amine
2-(oxolan-2-ylmethyl)-5-(4H-1,2,4-triazol-4-yl)-2,3-dihydro-1H-isoindole-1,3-dione
methyl 3-(1H-indole-2-amido)azepane-1-carboxylate
N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-4,5,6,7-tetrahydro-2-benzothiophene-1-carboxamide
N,1-diethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-1H-pyrazole-4-carboxamide
2-(cyclopropylmethyl)-9-[(2S)-2-hydroxy-3-phenylpropanoyl]-2,9-diazaspiro[5.5]undecan-3-one
(1S,5R)-6-propyl-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(pyridin-3-ylmethyl)piperazine
N-{[1-(2-methoxyethyl)piperidin-3-yl]methyl}-3-azaspiro[5.5]undecan-9-amine
9-(6-oxo-1,6-dihydropyridine-3-carbonyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-methyl-N-{[4-(methylsulfanyl)phenyl]methyl}-N-propyl-1H-1,2,3-benzotriazole-5-carboxamide
4-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-2,6-dimethylpyrimidine
6-(3-hydroxyazetidin-1-yl)-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(naphthalen-2-yloxy)piperidine-4-carboxylic acid
(2S)-N-cyclopropyl-2-acetamido-4-(methylsulfanyl)-N-{[4-(methylsulfanyl)phenyl]methyl}butanamide
1-{2-oxo-2-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]ethyl}-1,2-dihydroquinoxalin-2-one
N-[(2-chlorophenyl)methyl]-3-[1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]propanamide
3,4-dimethoxy-N-[(5-{[(3-methylphenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]benzamide
1-{[1-(2-hydroxyethyl)-3-(1H-indol-3-yl)-1H-1,2,4-triazol-5-yl]methyl}-5,5-dimethylimidazolidine-2,4-dione
methyl (2S,4R)-4-[3-(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)propanamido]-1-methylpyrrolidine-2-carboxylate
N-methyl-2-oxo-N-[(1-phenylpyrrolidin-3-yl)methyl]-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
2-(2-butoxy-5-methylphenyl)-N,N-dimethylpyridine-3-carboxamide
1-ethyl-6-{[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]methyl}-1H-indole
(1R,7S)-N-cyclopropyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-4-oxo-3-(pyridin-3-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
3-[3-methyl-1-(3-methylphenyl)-1H-1,2,4-triazol-5-yl]-1,2-dihydroquinoxalin-2-one
[1-(furan-2-ylmethyl)-3-(prop-2-en-1-yl)piperidin-3-yl]methanol
[1-(5-{3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)piperidin-4-yl]methanol
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}[(2,4-dimethylphenyl)methyl]methylamine
(3S,4R)-1-{imidazo[1,2-a]pyridine-3-carbonyl}-4-methyl-3-(2-methylpropyl)piperidin-4-ol
5-(4-{[(1R,9aR)-1-hydroxy-octahydro-1H-quinolizin-1-yl]methyl}piperazin-1-yl)-2,3-dihydropyridazin-3-one
2-cyclopropyl-4-phenyl-9-(pyrrolidine-1-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
2-methyl-8-{[2-(2-phenylethoxy)phenyl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine
4-({2-[2-(dimethylamino)ethyl]piperidin-1-yl}methyl)-1-ethyl-1H-pyrrole-2-carbonitrile
N-[3-(dimethylamino)propyl]-1-(ethanesulfonyl)-N-methylpiperidin-3-amine
5-{[4-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-3-(propan-2-yl)-1,2-oxazole
(3S,4R)-N,N-dimethyl-1-[(4-methyl-1,3-thiazol-5-yl)methyl]-4-(4-methylphenyl)pyrrolidin-3-amine
N-{[1-(phenoxymethyl)cyclopropyl]methyl}-4-(piperidin-3-yl)benzamide
6-({3-[3-(2-methylpropyl)pyrrolidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)quinoline
1-[2-(3-chlorophenyl)ethyl]-4-{[(1-ethyl-1H-pyrazol-4-yl)methyl]amino}pyrrolidin-2-one
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[4-(oxolane-2-carbonyl)piperazin-1-yl]ethan-1-one
4-(4-fluoro-2-hydroxyphenyl)-3-methyl-1-propyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
3-[(3S)-3-(dimethylamino)azepane-1-carbonyl]-1-methyl-6-(propan-2-yl)-1,2-dihydropyridin-2-one
1-(3-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}pyrrolidin-1-yl)-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
4-[3-(2,6-dioxo-1,3-diazinan-1-yl)propoxy]benzamide
7-chloro-4-methyl-N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]quinolin-2-amine
{1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}(pyridin-2-yl)methanol
N-cyclopentyl-4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carboxamide