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2-(cyclopentylmethyl)-6-methyl-4-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]-N-(pyridin-3-ylmethyl)-1,4-dihydropyridine-3-carboxamide
{[5-(1-{imidazo[1,2-b]pyridazine-3-carbonyl}piperidin-3-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}dimethylamine
2-(4-fluorophenyl)-4-(4-phenyl-1H-imidazole-5-carbonyl)morpholine
6-[(1-methylpiperidin-4-yl)methyl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}benzamide
4-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]butanamide
(3S,7S,8aS)-7-{[(3-chlorophenyl)methyl]amino}-3-[(4-methoxyphenyl)methyl]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
1-(3-methylfuran-2-carbonyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
(3S,4S)-4-cyclopropyl-1-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]pyrrolidine-3-carboxylic acid
5-acetyl-N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}thiophene-2-carboxamide
1-(2-oxo-6-phenyl-1,2-dihydropyridine-3-carbonyl)-3-propylpiperidine-3-carboxylic acid
4-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-N,6-dimethylpyrimidin-2-amine
1-[5-({[3-(dimethylamino)-2,2-dimethylpropyl]amino}methyl)-2-methoxyphenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
2-ethyl-9-(3-hydroxy-2-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-1,2,4-triazole
(1R,5S)-3-(2,2-diphenylethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-ethyl-5-[(1E)-pent-1-en-1-yl]thiophene-2-carboxamide
1-({1-[6-(3-fluorophenyl)pyridine-3-carbonyl]piperidin-4-yl}methyl)pyrrolidin-2-one
N'-[1-(furan-2-carbonyl)piperidin-3-yl]-N-(2-methylphenyl)ethanediamide
6-[(dimethylamino)methyl]-N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-2-(3-methoxyphenyl)-1,3-benzoxazole-6-carboxamide
2-(2-chloro-4-fluorophenoxymethyl)-N-(pyridin-3-ylmethyl)-1,3-oxazole-4-carboxamide
3-({[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}(prop-2-en-1-yl)amino)-1λ6-thiolane-1,1-dione
N-[(6-chloro-1H-1,3-benzodiazol-2-yl)methyl]-2,3-dimethylquinoxaline-6-carboxamide
N-[(3-cyclopropyl-1H-1,2,4-triazol-5-yl)methyl]-4-ethylcyclohexane-1-carboxamide
3-{1-[5-(hydroxymethyl)furan-2-carbonyl]piperidin-4-yl}-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{[4-(propan-2-yl)piperidin-1-yl]sulfonyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
3-(2-chloro-4-fluoro-5-methylphenyl)-1-[1-(oxolan-2-ylmethyl)piperidin-4-yl]urea
2-{[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]methyl}pyridine
5-{2-[2-(4-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{2-[3-(1-methoxyethyl)phenyl]phenyl}ethan-1-amine
1-{[2-(3-chlorophenyl)-6,7-dimethoxyquinolin-3-yl]methyl}-N,N-dimethylpyrrolidin-3-amine
methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}amine
1-(3-{[(2-methylprop-2-en-1-yl)amino]methyl}phenoxy)-3-(morpholin-4-yl)propan-2-ol
N-[3-(1H-indazol-1-yl)propyl]-4-(pyridin-3-yl)pyrimidin-2-amine
ethyl 3-benzyl-1-(3-fluorobenzenesulfonyl)piperidine-3-carboxylate
1-[5-(methoxymethyl)-1,3,4-oxadiazole-2-carbonyl]piperidin-3-ol
4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
8-(2-amino-2-methylpropyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
1-[1-(2-hydroxyethyl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-3-carboxamide
4-[2-(3-methoxyphenyl)azetidine-1-carbonyl]-1-(propan-2-yl)pyrrolidin-2-one
2-(1-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)ethan-1-ol
2-({5-[1-(1H-imidazol-1-yl)ethyl]-4-phenyl-4H-1,2,4-triazol-3-yl}sulfanyl)acetic acid
N-(1-methylpiperidin-4-yl)-3-(1,2-oxazinan-2-yl)-N-(2-phenylethyl)propanamide
N-[4-(4-hydroxyphenyl)-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]-2-methoxybenzamide
2-[1-(2,3-dihydro-1H-inden-2-yl)-5-[(1S)-1-(methylamino)ethyl]-1H-1,2,4-triazol-3-yl]acetamide
5-({4-[(3-methylphenyl)methyl]piperazin-1-yl}methyl)-2-phenylpyrimidine
4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)-N-{2-[(3-methylpyridin-2-yl)amino]ethyl}pyrimidine-5-carboxamide
3-fluoro-4-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-4-(1H-pyrazol-3-yl)benzamide