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3-chloro-4-fluoro-N-(2-hydroxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-benzothiophene-2-carboxamide
11-{[2-(4-fluorophenyl)ethyl]amino}-4-[(2-methoxyphenyl)methyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-[(1-benzoylpiperidin-4-yl)amino]-N-(2,5-dimethylphenyl)propanamide
8-fluoro-N-[1-(pyrazin-2-yl)propan-2-yl]quinoline-2-carboxamide
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-{[4-(methoxymethyl)piperidin-1-yl]methyl}piperidin-2-one
4-[(6-methylpyridin-3-yl)oxy]-1-(5-oxo-2,5-dihydro-1H-pyrazole-3-carbonyl)piperidine-4-carboxylic acid
4-(2,6-dimethylpyridin-3-yl)-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}pyrimidin-2-amine
3-methoxy-1-(2-oxo-2-{4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}ethyl)-1,2-dihydropyridin-2-one
7-acetamido-1-ethyl-2-(2-fluorophenyl)-N-[3-(1H-imidazol-1-yl)propyl]-1H-1,3-benzodiazole-5-carboxamide
N3-ethyl-N5-[(4-methoxyphenyl)methyl]-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
9-(2-hydroxypyridine-3-carbonyl)-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}({5-[1-(1,3-thiazol-4-ylmethyl)-1H-pyrazol-3-yl]furan-2-yl}methyl)amine
2-[(5-{[4-(1-hydroxy-2-methylpropyl)piperidin-1-yl]methyl}pyrimidin-2-yl)(methyl)amino]acetic acid
2-{1-[2-(2-chlorophenyl)-2-(dimethylamino)ethyl]-1H-imidazol-2-yl}benzoic acid
N-tert-butyl-3-({[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]carbamoyl}amino)-2-methylbenzamide
N-[(4-hydroxyazepan-4-yl)methyl]-5-[(4-methylpiperazin-1-yl)methyl]furan-2-carboxamide
1-[2-(morpholin-4-yl)ethyl]-6-oxo-N-[3-(pyridin-2-yl)propyl]piperidine-3-carboxamide
1-[4-(4-{[(1-benzothiophen-2-ylmethyl)(methyl)amino]methyl}phenoxy)piperidin-1-yl]-2-ethylbutan-1-one
2-amino-4-[3-(prop-2-en-1-yloxy)phenyl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
6-[(dimethylamino)methyl]-2-oxo-N-[(4-sulfamoylphenyl)methyl]-1,2-dihydropyridine-3-carboxamide
2-{1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline
2-[3-(dimethylamino)pyrrolidin-1-yl]-1-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]ethan-1-one
N-(2,5-dimethoxyphenyl)-3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carboxamide
9-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]-3-oxa-9-azaspiro[5.5]undecane
3-cyclopropyl-5-[2-(4-methylphenoxymethyl)furan-3-yl]-1H-1,2,4-triazole
2-{4-[3-(3-hydroxy-1,2-oxazol-5-yl)propanoyl]-5-methyl-2-oxopiperazin-1-yl}benzonitrile
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-propylbenzamide
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-2,6-dimethylpyridine-4-carboxamide
methyl[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amine
2-[benzyl(methyl)amino]-N-(2-hydroxy-2-phenylethyl)-N-methyl-6-phenylpyridine-3-carboxamide
4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-1-{[2-(trifluoromethyl)phenyl]methyl}piperidine
3-methyl-5-(3-phenyl-1H-pyrazol-5-yl)-1-propyl-1H-1,2,4-triazole
(4-methyl-5-{1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methanol
2-(pyridin-2-yl)-5-[4-(pyrrolidine-1-carbonyl)piperidine-1-carbonyl]pyrimidine
3-{[cyclohexyl(methyl)amino]methyl}-1-[(4-fluorophenyl)methyl]-3-hydroxypiperidin-2-one
N-[(1R,2R,4S)-bicyclo[2.2.1]heptan-2-yl]-6-(2,5-dimethylfuran-3-yl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
(3-{[1-(2,5-dimethylbenzoyl)pyrrolidin-3-yl]methyl}phenyl)methanol
5-[2-chloro-4-(4H-1,2,4-triazol-4-yl)phenyl]-3-cyclopropyl-1H-1,2,4-triazole
2-(5-{imidazo[1,2-a]pyridin-2-yl}-1,2,4-oxadiazol-3-yl)pyridine
2-cyclohexyl-5-{[3-ethyl-4-(propan-2-yl)piperazin-1-yl]methyl}pyrimidine
1-(cyclohexylmethyl)-N5-ethyl-N3-(2-hydroxy-2-phenylethyl)-N3-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-(pyrrolidin-1-yl)benzamide
2-methyl-5-{[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-1,3-benzodiazole
ethyl 4-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperazine-1-carboxylate
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-5-oxo-2,5-dihydro-1H-pyrazole-3-carboxamide
4-(5-tert-butyl-1H-pyrazol-3-yl)-N-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
8-(6-aminopyridine-3-carbonyl)-2-benzyl-2,8-diazaspiro[4.5]decan-3-one
({4-[5,6-dimethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-1,4-oxazepan-6-yl}methyl)dimethylamine
N-{[2-(diethylamino)pyridin-3-yl]methyl}oxolane-2-carboxamide
N-[(3-chlorophenyl)methyl]-3-(1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}piperidin-4-yl)propanamide