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2-cyclohexyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}acetamide
4-{[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}-2-methoxyphenol
13-[4-(1H-imidazol-1-yl)phenyl]-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
1-(2,3-dimethylphenyl)-N-[(3S,4R)-4-ethoxyoxolan-3-yl]piperidin-4-amine
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
5,6-dimethyl-3-[3-(morpholin-4-ylmethyl)phenyl]-1,2-dihydropyridin-2-one
methyl 3-cyclohexaneamido-6-({methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)thieno[2,3-b]pyridine-2-carboxylate
N,N-dimethyl-3-{[4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]sulfonyl}benzamide
1-(2-{4-[(dimethylamino)methyl]phenyl}piperidin-1-yl)-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
4-(4-methoxyphenyl)-N-methyl-N-(quinolin-5-ylmethyl)butanamide
ethyl 1-(1-ethyl-5-methyl-1H-pyrazole-4-amido)cyclobutane-1-carboxylate
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-[4-(3-methylphenyl)phenyl]piperidine-4-carboxamide
2-methoxy-4-{1-[3-(pyrrolidin-1-ylmethyl)phenyl]-1H-imidazol-2-yl}phenol
4-ethyl-1-methyl-3-[1-(5-methylpyrazine-2-carbonyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
(3aS,6aS)-2-cyclohexyl-5-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-{[(1S,5R)-6-benzyl-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}benzonitrile
N-(1,3-benzothiazol-2-ylmethyl)-N-methyl-3-[5-(5-methyl-1,2-oxazol-3-yl)-1,3,4-oxadiazol-2-yl]propanamide
3-(6-methoxy-1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-1-[2-(6-methylpyridin-2-yl)ethyl]urea
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-1-(furan-2-ylmethyl)piperidine-3-carboxamide
1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-2-phenylbutan-1-one
methyl 2-[methyl({[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl})carbamoyl]piperidine-1-carboxylate
2-(5-fluoro-2-methyl-1H-indol-3-yl)-1-[2-(propan-2-yl)-2,5-dihydro-1H-pyrrol-1-yl]ethan-1-one
1-(1-{1-[3-methyl-4-(1H-pyrrol-1-yl)benzoyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
8-(butan-2-yl)-1-(2-methoxyethyl)-3-(naphthalen-1-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[3,5-difluoro-4-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-3-carboxamide
2-({[(1-methyl-1H-imidazol-2-yl)methyl](propan-2-yl)amino}methyl)pyridin-3-ol
3-{4-[(3-methylphenyl)sulfanyl]piperidine-1-carbonyl}-1H,2H,5H,6H,7H-cyclopenta[b]pyridin-2-one
N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-{[(3-methylthiophen-2-yl)methyl]amino}benzamide
1-(isoquinolin-5-ylmethyl)-N-(6-phenoxypyridin-3-yl)piperidine-4-carboxamide
(2S,4S)-N-ethyl-1-(2-methoxyethyl)-4-(7-methyl-1-benzofuran-2-amido)pyrrolidine-2-carboxamide
7-[4-(trifluoromethoxy)benzenesulfonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-cyclopentyl-4-({[1-(3,5-dimethylphenyl)piperidin-4-yl]amino}methyl)pyrrolidin-2-one
3-ethyl-N-(1H-indol-5-ylmethyl)-1H-pyrazole-5-carboxamide
N-[2-(2,5-dimethylphenyl)ethyl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
1-[4-(morpholin-4-ylmethyl)piperidin-1-yl]-3-(pyridin-3-yl)propan-1-one
N-[3-(4-methylpiperazine-1-carbonyl)phenyl]-3-propylmorpholine-4-carboxamide
N-{3-[3,5-dimethyl-4-(2-oxopropyl)-1H-pyrazol-1-yl]phenyl}-2-methylpropanamide
1-(2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carbonyl)-4-phenoxypiperidine-4-carboxylic acid
4-[2-(3-chloro-4-hydroxyphenyl)acetyl]-1-(3-methoxyphenyl)piperazin-2-one
4-(4-acetyl-1,4-diazepane-1-carbonyl)-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
3-(4-methoxypiperidine-1-carbonyl)-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine
3-[(3R,4S)-1-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
N-{3-[4-(3-cyanopyridin-2-yl)piperazin-1-yl]-3-oxopropyl}-4-fluorobenzamide
N-(2-ethylphenyl)-2-oxo-2-[3-(2-oxopyrrolidin-1-yl)piperidin-1-yl]acetamide
dimethyl({2-[(thiophen-3-ylmethyl)({[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl})amino]ethyl})amine
1-[1-(oxan-4-yl)piperidine-4-carbonyl]-3-phenylpiperazine
N-ethyl-N-(2-methoxyethyl)-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
N-[(3,4-dichlorophenyl)methyl]-6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-[4-(benzyloxy)-3-methylphenyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
2-{4-[2-(2,3-dihydro-1H-inden-1-yl)acetyl]piperazin-1-yl}-N-ethylacetamide