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1-(cyclohexylmethyl)-N,N-dimethyl-5-[(3-methylbutyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(3S,5R)-1-[(2E)-3-phenylprop-2-en-1-yl]-5-[(pyridin-3-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
1-ethyl-N-[2-(5-methoxy-1H-indol-3-yl)ethyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-[(3R,4R)-4-amino-3-hydroxypiperidin-1-yl]-2-(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)ethan-1-one
1-cyclohexyl-3-methyl-5-(oxan-2-yl)-1H-1,2,4-triazole
5-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-ylmethyl]-N,N-dimethylpyrimidin-2-amine
4-[2-(naphthalen-1-yl)-3H-imidazo[4,5-b]pyridin-3-yl]-1-(1,3-thiazole-5-carbonyl)piperidine
(4S)-1-(2-ethyl-4-methyl-1,3-thiazole-5-carbonyl)-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
1-cyclopentyl-5-[4-(6-hydroxypyrimidin-4-yl)piperidine-1-carbonyl]piperidin-2-one
4-(2-methyl-1H-imidazol-1-yl)-1-(pyridin-4-yl)piperidine-4-carboxylic acid
2-(azocan-1-yl)-N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylacetamide
[2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl][(5-methylthiophen-2-yl)methyl]amine
N-[3-(1H-pyrazol-1-yl)phenyl]-1-[3-(1H-pyrazol-4-yl)propanoyl]pyrrolidine-2-carboxamide
1-(3-{4-[(3-methylphenyl)methyl]piperazin-1-yl}-3-oxopropyl)pyrrolidin-2-one
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methanesulfonamide
1-{4-[(2,3-dihydroxypropyl)amino]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
(3ar,6ar)-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
5-ethyl-N,2,3-trimethyl-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-4-phenoxybutanamide
N-[4-({3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.4]nonan-7-yl}methyl)phenyl]acetamide
5-(4-chloro-3,5-dimethylphenoxymethyl)-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,2-oxazole-3-carboxamide
9-[(4-methyl-1H-imidazol-2-yl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
4-[(3aS,6aS)-1-(1-benzofuran-2-ylmethyl)-octahydropyrrolo[2,3-c]pyrrol-5-yl]-2-methylpyridine
2-{1-[(4-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-(propan-2-yl)acetamide
6-ethyl-N-{3-[(1-methylpiperidin-4-yl)oxy]propyl}pyrimidin-4-amine
(2E)-1-[(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-3-hydroxypiperidin-1-yl]-3-(pyridin-3-yl)prop-2-en-1-one
2-(1H-imidazol-4-yl)-1-(2-methoxy-5-phenylphenyl)-1H-imidazole
(2R,3R,6R)-5-{[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
5-{2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]acetyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid
N-(2,1,3-benzoxadiazol-5-ylmethyl)-5-[(4-ethylpiperazin-1-yl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
2-methyl-5-(4-phenylazepane-1-carbonyl)pyrimidin-4-ol
5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]-N-(thiolan-3-yl)pyridin-2-amine
3-[2-(aminomethyl)-1H,2H-naphtho[2,1-b]furan-7-yl]-1,2-dihydropyridin-2-one
[(2S,4R,5R)-5-(4-chlorophenyl)-1-ethyl-2-methyl-4-{[(pyridin-3-ylmethyl)amino]methyl}pyrrolidin-2-yl]methanol
{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}(methyl)[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amine
5-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-2-amine
(1S,4S)-2-(2,3-dihydro-1H-inden-5-yl)-5-(pyridin-3-ylmethyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
dimethyl[2-(2-{[2-(morpholin-4-ylmethyl)piperidin-1-yl]methyl}phenoxy)ethyl]amine
5-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]quinoxaline
1-[(3,4-dimethylphenyl)methyl]-4-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)piperazin-2-one
2-[1-(4-chlorophenyl)-5-oxo-3-propyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(oxan-4-yl)acetamide
4-ethyl-6-[3-(piperidin-1-yl)pyrrolidin-1-yl]pyrimidine
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)benzamide
[(2S)-1-(2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-1,3-oxazole-4-carbonyl)pyrrolidin-2-yl]methanol
2-[benzyl(methyl)amino]-N-[1-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
2-[(3S,4R)-3-methanesulfonamido-4-(propan-2-yl)pyrrolidin-1-yl]pyridine-4-carboxylic acid
N-(2-methylbutyl)-1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carboxamide
N-[2-(3-methylphenyl)ethyl]-3-(1-methylpiperidin-2-yl)propanamide
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-3-methylpiperidine-3-carboxamide
1-cyclopentyl-4-[4-(5,6-dimethylpyrimidin-4-yl)piperazine-1-carbonyl]pyrrolidin-2-one