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(2S,4R)-4-amino-N-methyl-1-[(3R)-3-phenylbutanoyl]pyrrolidine-2-carboxamide
{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}({[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl})amine
9-[2-(2,3-dihydro-1H-inden-1-yl)acetyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-3-(1-methyl-1H-pyrazol-5-yl)-N-(piperidin-4-yl)propanamide
2-{1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]pyrrolidin-2-yl}pyridine
2-(4-acetyl-1,4-diazepan-1-yl)-2-(dimethyl-1,2-oxazol-4-yl)acetic acid
2-[4-(9H-fluoren-2-ylmethyl)-1-(propan-2-yl)piperazin-2-yl]ethan-1-ol
4-(2-methoxyphenyl)-1-{1H-pyrrolo[2,3-b]pyridin-6-yl}piperidine
2-[(3-hydroxy-2,2-dimethylpropyl)amino]-N-(1,3-thiazol-2-yl)propanamide
5-cyclopropyl-4-(3,4,5-trimethoxyphenyl)-1H-pyrazole
N'-(1-fluoro-3-phenylpropan-2-yl)-N-(2-fluoro-5-methylphenyl)butanediamide
3,3-dimethyl-1-[(5-{[4-(methylsulfanyl)phenyl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]urea
(3R,4R)-4-cyclopropyl-N-[(3-fluorophenyl)methyl]-4-hydroxy-3-methylpiperidine-1-carboxamide
1-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}-4-(1H-pyrazol-4-yl)butan-1-one
3-[4-(4-methoxybenzoyl)piperazine-1-carbonyl]-2,6-dimethyl-1,4-dihydropyridin-4-one
2-[({5-[1-(2-methoxy-3-methylbenzoyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)(methyl)amino]ethan-1-ol
3-(3-methylphenyl)-N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-pyrazole-4-carboxamide
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-(1,4-oxazepane-4-sulfonyl)benzamide
[(5-chlorofuran-2-yl)methyl](oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
N,3,5-trimethyl-N-[1-(1,2-oxazol-3-yl)ethyl]-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
(3R,4S)-4-phenyl-1-[2-(1H-1,2,3,4-tetrazol-1-yl)pyridine-4-carbonyl]pyrrolidin-3-amine
1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-6-yl}urea
1-(pyridin-3-ylmethyl)-4-[6-(thiomorpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]-1,4-diazepane
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]acetamide
6-(2-methylpropyl)-4-[4-(pyridin-2-ylmethyl)-1,4-diazepane-1-carbonyl]-1,2-dihydropyrimidin-2-one
1-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2-methyl-4-(2-methylphenyl)piperazine
1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-2-(2-methyl-1H-imidazol-1-yl)propan-1-one
1-{5-[(cycloheptylamino)methyl]-2-methoxyphenoxy}-3-(pyrrolidin-1-yl)propan-2-ol
5-{4-hydroxy-1-[(4-methylphenyl)methyl]piperidin-4-yl}-N-methyl-N-[2-(pyridin-2-yl)ethyl]-1-benzofuran-2-carboxamide
7-[(3,4-difluorophenyl)methyl]-2-[(1-methyl-1H-imidazol-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-{[1-(ethoxymethyl)cyclobutyl]methyl}-4-hydroxy-2-phenylpyrimidine-5-carboxamide
1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-4-(1,3-thiazol-2-yl)piperazine
(1R,2R,6S,7S)-4-(2-methyl-4-phenylpyrimidine-5-carbonyl)-10-oxa-4-azatricyclo[5.2.1.02,6]decane
1-[4-(benzyloxy)piperidin-1-yl]-2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethan-1-one
[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl](oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
N-[(2S,4R,6R)-2-(2,1,3-benzothiadiazol-4-yl)-6-(4-fluoro-3-methoxyphenyl)oxan-4-yl]acetamide
3-benzyl-1-methyl-8-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl (2S,4R)-1-[(5-chloro-2-hydroxyphenyl)methyl]-4-{2-[3-(trifluoromethyl)phenyl]acetamido}pyrrolidine-2-carboxylate
N-[4-(furan-2-yl)butan-2-yl]-5-(1H-indol-1-ylmethyl)-1H-pyrazole-3-carboxamide
4-[4-(1-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]piperidine
3-[1-(2H-1,3-benzodioxol-4-ylmethyl)piperidin-3-yl]-N-[(2-chlorophenyl)methyl]propanamide
N-[3-(2,6-dimethylphenoxy)propyl]-2-ethyl-N-methylpyrimidine-5-carboxamide
1-ethyl-3-(4-phenyl-1H-imidazol-5-yl)piperidine
(3S,4R)-N,N-dimethyl-4-(4-methylphenyl)-1-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}pyrrolidin-3-amine
N-(4-{5-[(2-methoxypyridin-3-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}phenyl)acetamide
1-[2-(dimethylamino)ethyl]-N-{[2-fluoro-3-(trifluoromethyl)phenyl]methyl}-5-oxopyrrolidine-3-carboxamide
1-(2-fluoro-4-methoxyphenyl)-2-{[5-(methoxymethyl)furan-2-yl]methyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
2-[1-cyclopentyl-3-(2-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
2-(2-{[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
2-[3-(dimethylamino)propyl]-9-(6-oxo-1,6-dihydropyridine-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one