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3-[1-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1H-1,2,3-triazol-4-yl]piperidine
2-cyclopropyl-9-(2-oxoimidazolidine-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
5-[({[1-(2-methoxyethyl)piperidin-4-yl]methyl}(pyridin-4-ylmethyl)amino)methyl]pyrimidin-2-amine
3-[2-chloro-5-(morpholine-4-carbonyl)phenyl]-1-[(3R)-piperidin-3-yl]urea
2-(3-{1-[(3-methoxyphenyl)methyl]-1H-pyrazol-3-yl}phenyl)pyrimidine
N-[(3S,4R)-4-(4-methylphenyl)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-3-yl]acetamide
N-[(5-chloro-1H-indol-2-yl)methyl]-2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]acetamide
5-(2-methoxyphenoxymethyl)-N-[(2S)-pyrrolidin-2-ylmethyl]-1H-pyrazole-3-carboxamide
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-(2-oxopyrrolidin-3-yl)benzamide
4-[4-(4-methylpyridin-2-yl)piperazin-1-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[2-(dimethylamino)ethyl]-N-ethyl-1,3-oxazole-4-carboxamide
(7-chloro-5-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-2,3-dihydro-1-benzofuran-2-yl)methanamine
2-(1-{[2-(ethylamino)pyrimidin-5-yl]methyl}piperidin-2-yl)acetic acid
2-methyl-N-(1-methylpiperidin-4-yl)-5-(propan-2-yl)-N-(pyridin-3-ylmethyl)furan-3-carboxamide
2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-(pyridin-2-ylmethyl)-1,3-oxazole-4-carboxamide
1-(2-methylpyridin-4-yl)-4-(thiophene-3-carbonyl)-1,4-diazepane
3-(2-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-2-oxoethyl)-4-ethylpiperazin-2-one
1-{2-[3-(2-ethylphenoxy)azetidin-1-yl]-2-oxoethyl}-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
N-[(1S,2R)-2-carbamoylcyclopentyl]-3-(3-fluorophenyl)-1H-pyrazole-4-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(1,3-thiazole-4-carbonyl)piperidin-3-ol
1-{3-[4-(3-methoxyphenyl)-3-oxopiperazin-1-yl]-3-oxopropyl}azepan-2-one
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2,6-dimethoxypyridine-3-carboxamide
2-(cyclopentylmethyl)-N-[3-(1H-imidazol-1-yl)propyl]-1-(2-methoxyethyl)-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N,5-dimethyl-2-phenyl-1H-imidazole-4-carboxamide
4-(4-fluorobutyl)-9-(2-methoxyethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]acetamide
(3S,4S)-1-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
2-{[(1,3-benzothiazol-2-yl)amino]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
4-phenyl-3-(piperidin-3-yl)-1-[3-(pyridin-3-yl)propyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-cyclohexyl-4-{4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carbonyl}piperazin-2-one
N-[2-(pyrrolidine-1-sulfonyl)ethyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
1-[(1-benzyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-3-(2,5-difluorobenzoyl)piperidine
(1S,5R)-6-benzyl-3-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-chloro-N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-1H-pyrazole-3-carboxamide
2-{[(1-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)oxy]methyl}pyridine
4-[8-(trifluoromethyl)quinolin-4-yl]benzamide
2-{[1-(2,5-dihydro-1H-pyrrole-2-carbonyl)piperidin-4-yl]oxy}-4-methoxy-N-(2-methoxyethyl)benzamide
1-(2-hydroxyethyl)-3-{4-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}-1-(1,3-thiazol-2-ylmethyl)urea
1-[(2,6-dichloro-3-hydroxyphenyl)methyl]piperidine-4-carbonitrile
N-ethyl-6-{6-[(2-hydroxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-N-methylpyridine-3-carboxamide
2-[(2-methoxyethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
4-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-N-(2-methoxyethyl)-N-(pyridin-4-ylmethyl)benzamide
1-[5-fluoro-4-(pyrrolidin-1-yl)pyrimidin-2-yl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[(3S,7S,8aS)-3-[(1R)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]benzamide
1,5-dimethyl-2-phenyl-4-(1-{1-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-imidazol-2-yl)-2,3-dihydro-1H-pyrazol-3-one
6-ethyl-N-(1H-imidazol-2-ylmethyl)-N-methyl-2-(morpholin-4-yl)pyrimidin-4-amine
(4aS,8aS)-2-(4-aminopyrimidin-2-yl)-7-cyclohexanecarbonyl-decahydro-2,7-naphthyridin-4a-ol
3-{3-[2-(pyridin-4-yl)-1H-imidazol-1-yl]phenyl}-1,3-oxazolidin-2-one
1-[5-(1,5-dimethyl-1H-pyrazol-4-yl)-1,2-oxazole-3-carbonyl]-3-(1H-imidazol-2-yl)piperidine
(3S,9aR)-3-benzyl-8-[(3-fluorophenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione