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N-(4-phenylbutan-2-yl)-1H-1,2,3-triazole-5-carboxamide
methyl (2S,4S)-4-cyclohexaneamido-1-(1-ethylpiperidin-4-yl)pyrrolidine-2-carboxylate
1-[2-(ethoxymethyl)-4-{[(5-methyl-1,2-oxazol-3-yl)methyl]amino}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]ethan-1-one
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carboxamide
dimethyl({4-methyl-5-[1-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
2-(2-ethoxypyridin-3-yl)-2-[4-(piperidin-1-yl)piperidin-1-yl]acetic acid
6-[2-(4-fluorophenoxy)ethyl]-1,2-dihydroisoquinolin-1-one
(3aS,6aR)-5-[(4-methyl-1H-imidazol-5-yl)methyl]-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
3-[1-(hydroxymethyl)cyclopentyl]-1-(4-methoxy-3,5-dimethylphenyl)urea
4-(6-methylpyridin-2-yl)-N-[3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]piperazine-1-carboxamide
3-ethyl-1-[4-(3-hydroxy-3-methylbut-1-yn-1-yl)benzoyl]piperidine-3-carboxylic acid
ethyl({3-[3-(1H-pyrazol-3-yl)phenyl]phenyl}methyl)amine
4,6-dimethyl-2-oxo-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-1,2,3,4-tetrahydropyrimidine-5-carboxamide
N-[(4-chlorophenyl)methyl]-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(cyclopropylmethyl)-N-[(2-fluorophenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-methyl-2-(2-oxo-1,2-dihydroquinolin-1-yl)-N-(oxolan-3-ylmethyl)acetamide
[1-(2-{[6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]amino}ethyl)piperidin-2-yl]methanol
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-1H-indole-2-carboxamide
(4aS,8aR)-1-(4-hydroxybutyl)-6-(pyrrolidine-1-carbonyl)-decahydro-1,6-naphthyridin-2-one
5-oxo-1-(4-phenylbutyl)pyrrolidine-3-carboxylic acid
2-(3-methylphenyl)-5-({4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}methyl)pyrimidine
6-(4-butylpiperazin-1-yl)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(15),3(8),6,11,13-pentaen-4-one
7,8-dimethyl-N-[1-(1-methyl-1H-1,2,4-triazol-5-yl)propyl]-2-(pyrimidin-5-yl)quinoline-4-carboxamide
4-[(3R)-3-hydroxypyrrolidine-1-carbonyl]-N-(oxan-4-ylmethyl)benzene-1-sulfonamide
N-(hexan-3-yl)-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
N-[3-hydroxy-1-(4-methylphenyl)propyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
(3S,4S)-4-cyclopropyl-1-(1-methyl-2-oxo-1,2-dihydroquinoline-4-carbonyl)pyrrolidine-3-carboxylic acid
6-{7-cyclopentyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}pyridine-2-carbonitrile
4-(1H-1,3-benzodiazol-2-ylmethyl)-3-ethyl-3-methylpiperazin-2-one
1-{2-[methyl(3-phenylpropyl)amino]ethyl}-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-[(4-fluorophenyl)methyl]-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
1-(3-{[3-(2-hydroxyethyl)-4-[(5-methylfuran-2-yl)methyl]piperazin-1-yl]methyl}phenyl)ethan-1-one
1-[4-(1H-imidazol-1-yl)benzoyl]-3-(3-methylphenyl)piperidine
4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)-1-[5-(thiophen-2-yl)-1H-pyrazole-4-carbonyl]piperidine
(2S)-2-{[2-(dimethylamino)-4-methylpyrimidin-5-yl]formamido}-3-(1H-indol-3-yl)propanoic acid
{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(oxan-4-ylmethyl)amine
1-{5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-yl}piperidin-4-ol
1-[4-(morpholine-4-carbonyl)piperazin-1-yl]-2-(naphthalen-2-yloxy)propan-1-one
7-methyl-3-(5-phenylpentanoyl)-3,7,11-triazaspiro[5.6]dodecan-12-one
3-[2-(4-fluorophenyl)ethyl]-3,4-dihydropteridin-4-one
2-acetyl-8-[(3-methyl-1,2-oxazol-5-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-[methyl({4-methyl-5-[1-(1,3-thiazole-4-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amino]ethan-1-ol
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-{[(2,6-difluorophenyl)methyl]amino}-1-(propan-2-yl)pyrrolidine-2-carboxamide
(3S,4R)-4-(3-methoxyphenyl)-1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]pyrrolidine-3-carboxylic acid
3-({cyclopropyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)-6-methoxy-1,2-dihydroquinolin-2-one
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-ethyl-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
N'-cyclopentyl-N'-propyl-N-(1,3,4-thiadiazol-2-yl)ethanediamide
N,N-dimethyl-5-({2-[2-(pyridin-2-yl)ethyl]piperidin-1-yl}methyl)pyridin-2-amine