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5-methyl-1-[(1-methyl-1H-pyrazol-4-yl)methyl]-5-phenylpiperidin-2-one
N-(pyridin-2-ylmethyl)-1-{1-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]piperidin-4-yl}piperidine-3-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-5-hydroxypyrazine-2-carboxamide
5-(6-methoxypyridin-3-yl)-1H-indazol-3-amine
1-cyclohexyl-3-hydroxy-4-(3-phenyl-1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
(4aS,7aR)-1-benzoyl-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-cyclopropyl-4-methoxy-3-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]oxy}benzamide
2-cyclohexyl-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]acetamide
N-cyclopentyl-6-(thiomorpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
3-(1-benzyl-1H-imidazol-2-yl)-1-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}piperidine
N-(3-acetylphenyl)-4-[(2-methylpyrrolidin-1-yl)methyl]benzamide
2-{2-[(4-chlorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}pyridine-3-carbonitrile
(4-{5-methyl-6-[(2-methylpyridin-3-yl)oxy]pyrimidin-4-yl}-1,4-oxazepan-6-yl)methanol
2-{4-[2-(2-hydroxyethyl)-4-methyl-1H-1,3-benzodiazol-1-yl]phenoxy}ethan-1-ol
N-({1-[(4-methylpiperazin-1-yl)methyl]cyclopropyl}methyl)-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-(2,4-dimethoxyphenyl)-3-(4-hydroxy-4-phenylpiperidin-1-yl)propanamide
2-(methylsulfanyl)-N-(piperidin-4-yl)-1,3-thiazole-4-carboxamide
2-ethyl-N-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}pyrimidine-5-carboxamide
4-[(4-methoxyphenyl)methyl]-1-[2-(2-methylphenyl)acetyl]-1,4-diazepan-5-one
4-[5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-3-carbonyl]thiomorpholine
1-(2,3-dihydro-1H-inden-2-yl)-4-[(2-methyl-6-propylpyrimidin-4-yl)amino]pyrrolidin-2-one
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(3-phenylpropyl)pyrrolidin-3-yl]methanol
6-{3-[(4-fluorophenyl)amino]piperidine-1-carbonyl}-2,3,4,5-tetrahydropyridazin-3-one
(3S,4R)-4-(3-fluorophenyl)-1-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}pyrrolidine-3-carboxylic acid
2-methyl-1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazine
(3R,5R)-N-{[3-(methylsulfanyl)phenyl]methyl}-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
N-(3-acetamidophenyl)-3-[4-(1-methyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]propanamide
8-(2,3-dihydro-1H-indene-5-carbonyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
methyl 5-(butane-2-sulfonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
1-[5-(4-methoxyphenyl)furan-2-carbonyl]-4-[2-(2-phenylethyl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidine
N-(3-{[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}-2,5-dimethyl-1H-pyrrol-1-yl)acetamide
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-2,4-dimethoxybenzamide
(3S,4S)-4-cyclopropyl-1-{[(3-fluorophenyl)methyl]carbamoyl}pyrrolidine-3-carboxylic acid
N-cyclopropyl-2-[4-(pyrimidin-2-yl)piperazin-1-yl]-N-(thiophen-3-ylmethyl)acetamide
7-methyl-3-[2-(1H-pyrazol-4-yl)ethyl]-3H,4H-thieno[3,2-d]pyrimidin-4-one
7-methyl-2-[2-(3-methylphenyl)benzoyl]-2,7-diazaspiro[4.5]decan-6-one
5-{[3-(1,3-benzoxazol-2-yl)piperidin-1-yl]methyl}-N-ethylpyrimidin-2-amine
5-({2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidin-1-yl}methyl)-N-propylpyrimidin-2-amine
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1-methyl-1H-pyrazole-5-carboxamide
5-(2,5-dichlorophenyl)pyridin-3-amine
5-chloro-2-{4-[(6-phenoxypyridin-3-yl)methyl]piperazin-1-yl}pyrimidine
1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
(2E)-N-{[2-(dimethylamino)-7-methoxyquinolin-3-yl]methyl}-3-(3-fluorophenyl)-N-(2-methoxyethyl)prop-2-enamide
1-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-3-{5-[(4-chlorophenyl)methyl]-1,3,4-thiadiazol-2-yl}urea
3-cyclopropyl-5-{4H-thieno[3,2-b]pyrrol-5-yl}-1H-1,2,4-triazole
3-(2-ethyl-1H-imidazol-1-yl)-1-[4-(naphthalen-2-yl)piperazin-1-yl]propan-1-one
[1-(2-methoxypyridine-3-carbonyl)-3-(2-phenoxyethyl)piperidin-3-yl]methanol
1-(1,3-benzothiazol-2-yl)-N-[1-(1H-imidazol-1-yl)butan-2-yl]piperidin-4-amine
3-({[7-methyl-2-oxo-1-(2-phenoxyethyl)-1,2-dihydroquinolin-3-yl]methyl}amino)-1λ6-thiolane-1,1-dione
4,6-dimethyl-2-[({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)amino]pyridine-3-carbonitrile