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4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-[3-(methylsulfanyl)propyl]benzamide
2-[(1,2-dimethyl-1H-imidazol-4-yl)sulfonyl]-8-methyl-2,8-diazaspiro[4.5]decane
N-methyl-3-(2-oxoazepan-1-yl)-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]propanamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(1,3,6-trimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)pyrrolidine-1-carboxamide
7-methyl-4-{[3-(propan-2-yl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-2H-chromen-2-one
4-[2-(3,3-diphenylpiperidin-1-yl)-2-oxoethyl]-1,2,3,6-tetrahydropyridazine-3,6-dione
3-{5-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
(3R,4R)-4-ethyl-1-(5-methoxyfuran-2-carbonyl)piperidine-3,4-diol
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-N-methyl-2-oxo-1,2-dihydroquinoline-4-carboxamide
5-[4-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-1-(2-methoxyethyl)piperidin-2-one
2-{[1-(4-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1-ethyl-1H-imidazole
5,6-dimethyl-3-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
1-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-2-[(cyclopropylmethyl)sulfanyl]ethan-1-one
4-{[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
3-ethoxy-1-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]propan-1-one
methyl 5-{[1-(methylsulfanyl)propan-2-yl]amino}-3-(oxolane-3-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-benzoyl-2-(cyclohexylmethyl)morpholine
3-{[1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}-4-(propan-2-yl)piperazin-2-one
1-(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-1H-pyrazole-4-carbonyl)-N,N-diethylpyrrolidin-3-amine
2-methyl-N-[3-(4-methylpiperazin-1-yl)propyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
N-(2,2-diphenylethyl)-2-(1-methyl-3-oxopiperazin-2-yl)acetamide
N-methyl-N-(2-phenylethyl)-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-(diphenylmethyl)-4-[(2-methyl-1,3-oxazol-4-yl)methyl]piperazine
{4-[2-(2-aminoethyl)phenyl]phenyl}methanol
2-(3-hydroxypiperidin-1-yl)-1-[4-(2-methylphenyl)-1,4-diazepan-1-yl]ethan-1-one
1-ethyl-4-(2-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}-2,3-dihydro-1H-inden-2-yl)piperazine
2-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-7-(cyclobutylmethyl)-2,7-diazaspiro[4.5]decan-6-one
ethyl 2-{[7-(1-phenylcyclopropaneamido)-1,2,3,4-tetrahydroisoquinoline-2-carbonyl]amino}acetate
2-({5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-5-methoxy-4H-pyran-4-one
1-{1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]pyrrolidin-3-yl}-4-methylpiperazine
N-{[5,8-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-3-(4-methylphenyl)propanamide
2-[2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)acetyl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
(3R,4R)-1-{[2-(5-methylfuran-2-yl)phenyl]methyl}-4-(4-methylpiperazin-1-yl)piperidin-3-ol
N-(5-chloro-2-methoxyphenyl)-2-{2-[(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]-4-(pyrimidin-2-yl)phenoxy}acetamide
6-methyl-N-(1,2-oxazol-3-ylmethyl)-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
N-[(3R,4S)-1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-propylpyrrolidin-3-yl]-2-(propan-2-yloxy)acetamide
N-({1-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]piperidin-4-yl}methyl)acetamide
(1S,5R)-6-[(3,5-difluoro-4-methoxyphenyl)methyl]-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-2-(4,6,7-trimethyl-1-benzofuran-3-yl)acetamide
2-(4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperazin-1-yl)pyridine-3-carboxamide
N,1,3-trimethyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
3-tert-butyl-5-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-1,2,4-oxadiazole
2-(dimethyl-1,2-oxazol-4-yl)-N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}acetamide
N-methyl-3-(2-oxoazepan-1-yl)-N-[1-(thiophen-2-yl)ethyl]propanamide
1-{2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
1-{3-cyclopropyl-5-[2-(1,2-oxazolidin-2-yl)ethyl]-1H-1,2,4-triazol-1-yl}isoquinoline
N,1-dimethyl-2-oxo-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2-dihydroquinoline-4-carboxamide
4-{1-[(5-ethylfuran-2-yl)methyl]azetidin-3-yl}morpholine
ethyl 2-{1-[2-(2-amino-4,6-dimethylpyrimidin-5-yl)acetyl]piperidin-2-yl}acetate
(3R,5R)-N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}-5-(morpholine-4-carbonyl)piperidine-3-carboxamide