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N-[2-(dimethylamino)ethyl]-4-(quinolin-2-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
1-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-3-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]urea
5-acetamido-N-[(4-fluorophenyl)methyl]-1-(2-methoxyethyl)-N-methyl-2-(pyridin-2-yl)-1H-1,3-benzodiazole-7-carboxamide
(3S,7S,8aS)-7-({[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)-3-[(4-hydroxyphenyl)methyl]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
(4aR,7aS)-1-(2-methoxyethyl)-4-[5-(methoxymethyl)furan-2-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-(propan-2-yl)-3-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
3-({[2-(2-methylphenoxy)pyridin-3-yl]methyl}carbamoyl)pyridin-1-ium-1-olate
1-{5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]benzoyl}-N,N-dimethylpyrrolidin-3-amine
2-[2-(4-methoxyphenoxy)ethyl]-2-azaspiro[4.4]nonan-3-one
5-[2-(ethylsulfanyl)ethyl]-1-[(4-fluorophenyl)methyl]-3-methyl-1H-1,2,4-triazole
5-{1-[(2-hydroxy-5-methylphenyl)methyl]piperidin-4-yl}-5-(pyridin-2-yl)imidazolidine-2,4-dione
N-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
5-(naphthalen-2-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
7-(2-methylphenyl)-4-[2-(pyridin-2-yl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[2-({2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazol-4-yl}formamido)ethyl]acetamide
1-(2-methoxyethyl)-2-[3-methyl-1-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1H-imidazole
2-(azepan-1-yl)-N-(2-ethoxypropyl)-N-methyl-2-oxoacetamide
1-cyclopentanecarbonyl-N-(1H-indol-4-ylmethyl)piperidine-4-carboxamide
3-{[methyl(pyrazin-2-ylmethyl)carbamoyl]methyl}-N-(thiophen-2-ylmethyl)morpholine-4-carboxamide
4-(2-{1-[3-(1H-pyrazol-1-yl)benzoyl]piperidin-2-yl}ethyl)morpholine
(3aS,6aR)-3-[(2-methoxyphenyl)methyl]-5-(quinolin-2-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-benzyl{[1-(pyrimidin-2-yl)piperidin-3-yl]amino}sulfonamide
N-({1-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-3-yl}methyl)pyridine-3-carboxamide
N-methyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-4-(1H-pyrazol-3-yl)benzamide
4-[1-(1-tert-butyl-1H-pyrrole-3-carbonyl)piperidin-3-yl]benzoic acid
N-(2-methoxyethyl)-N-methyl-5-(4-phenylazepane-1-carbonyl)pyridin-2-amine
(4aR,7aS)-1-(furan-2-carbonyl)-4-(oxane-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[1-(dimethyl-1,2-oxazole-4-carbonyl)piperidin-3-yl]methyl}-4-methoxybenzene-1-sulfonamide
4-methoxy-N-methyl-3-(pyrimidin-5-yl)benzamide
6-(3-hydroxyphenyl)-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide
ethyl 3-benzyl-1-(ethylcarbamoyl)piperidine-3-carboxylate
N-(2-methoxyethyl)-5-oxo-N-(thiophen-3-ylmethyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
methyl 4-{[3-ethyl-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-8-yl]methyl}benzoate
N-[2-(dimethylamino)ethyl]-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)acetamide
N,N-dimethyl-2-{[(5-phenyl-1,2,4-oxadiazol-3-yl)amino]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[(2-methoxyphenyl)methyl]piperidine-3-carboxamide
(2S)-1-[(5-chloro-2,4-dimethoxyphenyl)methyl]-4-methyl-2-phenylpiperazine
10-methoxy-5-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
3-(2-fluorophenyl)-N-[2-(pyridin-3-yl)ethyl]-1H-pyrazole-5-carboxamide
1-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)-4-(3-methylpyridin-2-yl)piperazine
2-(1-{[1-(pyridine-4-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-2-ol
4-(4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)thiomorpholine
N-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-5-[1-(4-methoxyphenyl)-1H-pyrazol-3-yl]-4-methyl-1,3-thiazol-2-amine
1'-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
4-[(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidin-1-yl)methyl]-1H-pyrazole-3-carboxylic acid
6-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]-4-methyl-1,3-benzothiazol-2-amine
(3R,4R)-4-hydroxy-1-methyl-N-(3-phenylprop-2-yn-1-yl)-N-propylpiperidine-3-carboxamide
6-(6-{[2-(dimethylamino)ethyl]amino}-1H-pyrrolo[2,3-b]pyridin-4-yl)quinazolin-4-amine
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]pyrazine-2-carboxamide
4-(4-chlorophenyl)-1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-ol