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6-(2-fluoro-4-methoxyphenyl)-7-methyl-8-oxo-N-[2-(1H-pyrazol-1-yl)ethyl]-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl][(1-ethyl-1H-imidazol-2-yl)methyl]methylamine
2-(2,5-dioxoimidazolidin-1-yl)-N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]acetamide
3-[1-(6-aminopyridine-3-carbonyl)piperidin-3-yl]-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-{4-[3-(1H-pyrazol-1-yl)azetidin-1-yl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl}benzamide
1-methyl-1'-(5-methyl-1H-indole-2-carbonyl)-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
N,N-dimethyl-7-(4-methyl-1H-pyrrole-2-carbonyl)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1'-[(1-phenyl-1H-pyrazol-5-yl)methyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
N2-{[4-(dimethylamino)oxan-4-yl]methyl}-N4-ethylpyrimidine-2,4-diamine
[(3R,4R)-4-[(dimethylamino)methyl]-1-(5-phenyl-1,3,4-thiadiazol-2-yl)pyrrolidin-3-yl]methanol
1-(4-chlorophenyl)-N-{[1-(1,2,4-oxadiazol-3-ylmethyl)piperidin-3-yl]methyl}cyclopropane-1-carboxamide
3-[5-(1-cyclopropanecarbonylpiperidin-2-yl)-1,2,4-oxadiazol-3-yl]pyridazine
8-[2-(methylamino)acetyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
1-[2-(1-cyclohexanecarbonylpiperidin-2-yl)ethyl]-N-cyclopropyl-1H-1,2,3-triazole-4-carboxamide
methyl 2-[({1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)amino]-2-methylpropanoate
methyl[3-(1-methyl-1H-imidazol-2-yl)propyl]{[3-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}amine
1-[(2-chloro-5-ethoxy-4-methoxyphenyl)methyl]azepan-4-ol
N,1-dimethyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-[(3-hydroxypiperidin-1-yl)methyl]-N-(1-propyl-1H-1,2,4-triazol-3-yl)benzamide
(3S,4S)-1-(benzenesulfonyl)-4-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]pyrrolidin-3-ol
4-({4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-2,1,3-benzoxadiazole
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-5-methyl-1,3,4-oxadiazol-2-amine
5-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)-3-methyl-1,2,4-oxadiazole
N-(2,1,3-benzoxadiazol-5-ylmethyl)-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
ethyl[(1-methyl-1H-pyrazol-4-yl)methyl]{[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}amine
1-(2,1,3-benzoxadiazol-4-ylmethyl)-4-(1H-imidazol-1-ylmethyl)piperidin-4-ol
N-(2-methoxyethyl)-N-[(3-methylthiophen-2-yl)methyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-5-(1H-pyrazol-1-ylmethyl)furan-2-carboxamide
(2S,4S)-4-amino-N-methyl-1-[4-(2-methyl-1H-imidazol-1-yl)butanoyl]pyrrolidine-2-carboxamide
N-(3-methoxypropyl)-3-{[(1-methyl-1H-pyrazol-4-yl)methyl]sulfamoyl}benzamide
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methyl-3-(1H-pyrazol-1-ylmethyl)benzamide
{3-benzyl-1-[(6-methoxy-2H-chromen-3-yl)methyl]piperidin-3-yl}methanol
2-[cyclopropyl({4-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-1,2,3-triazol-1-yl})methyl]-4-methylpyridine
N-{2-[3-(2-methylpropyl)-1-(quinolin-8-yl)-1H-1,2,4-triazol-5-yl]ethyl}acetamide
2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]acetic acid
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-6-methylimidazo[1,2-a]pyridine-2-carboxamide
5-(dimethyl-1,2-oxazole-4-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
(1S,5R)-6-(1,3-thiazol-4-ylmethyl)-3-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[4-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]-3-[1-(pyrimidin-2-yl)piperidin-3-yl]urea
N-{2-[(3,5-dimethyladamantan-1-yl)oxy]ethyl}-3-(1-methyl-1H-pyrazol-4-yl)propanamide
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-(5-methyl-1,3-oxazole-4-carbonyl)piperidine
1-(azepan-1-yl)-2-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethan-1-one
1-{4-[(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)amino]piperidin-1-yl}ethan-1-one
N-ethyl-2-(4-{[3-(furan-2-yl)phenyl]methyl}piperazin-1-yl)acetamide
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-8-fluoroquinoline-2-carboxamide
N-methyl-N-[(5-methylfuran-2-yl)methyl]-4-(propan-2-yl)pyrimidin-2-amine
(2S,4R)-N-[2-(4-fluorophenyl)ethyl]-1-[(4-phenylphenyl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-1-ethyl-7-methyl-4-oxo-1,4-dihydro-1,8-naphthyridine-3-carboxamide
1-{2-[4-fluoro-3-(hydroxymethyl)phenyl]phenoxy}-3-(piperidin-1-yl)propan-2-ol
3-(morpholine-4-carbonyl)-1-propyl-N-{[4-(trifluoromethoxy)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-5-amine