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(1S,3R)-3-amino-N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]cyclopentane-1-carboxamide
1-{2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)amino]ethyl}imidazolidin-2-one
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidin-3-ol
5-acetyl-6-methyl-3-[4-(3-methylpyridin-2-yl)piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
(1S,3R)-1-ethoxy-3-hydroxy-N-[(4-methoxyphenyl)methyl]-7-azaspiro[3.5]nonane-7-carboxamide
5-{4-[(2-fluorophenyl)methyl]-1,4-diazepane-1-carbonyl}-2-methylpyrimidin-4-ol
6-[(E)-2-phenylethenyl]-1,2,3,4-tetrahydroquinazoline-2,4-dione
1-(4-methanesulfonyl-1,4-diazepan-1-yl)-2-(1,3-thiazol-4-yl)ethan-1-one
1-(2-aminoethyl)-N-[(3S,4R)-4-ethoxyoxolan-3-yl]-1H-1,2,3-triazole-4-carboxamide
2-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridine-6-carbonyl]imidazo[1,2-a]pyrimidine
4-{1-[(3,5-dichloro-2-methoxyphenyl)methyl]piperidin-4-yl}-5-methylpyrimidine
methyl 6-[(4-chlorophenyl)methyl]-2-[(1-methoxypropan-2-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-4-methoxybenzene-1-sulfonamide
N-(1-methoxypropan-2-yl)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N,1,3-trimethyl-N-[3-(3-methylphenoxy)propyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
{4-methyl-5-[1-(quinolin-4-ylmethyl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methanol
4-[(4-{2-[1-(pyridine-4-carbonyl)piperidin-2-yl]ethoxy}phenyl)methyl]piperazine-1-carbaldehyde
N-(2-methylpropyl)-5-oxo-N-(thiophen-3-ylmethyl)hexanamide
1-methyl-5-{[(5-methylfuran-2-yl)methyl]amino}-N-[2-(morpholin-4-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
{5-[1-(1-benzothiophen-2-ylmethyl)-1H-imidazol-2-yl]furan-2-yl}methanol
2,6-dimethoxy-N-propyl-N-(pyridin-3-ylmethyl)pyridine-3-carboxamide
3-(4-{2-[2-(oxolan-3-yl)-1H-imidazol-1-yl]ethyl}-1,3-thiazol-2-yl)pyridine
3-(azepane-1-sulfonyl)-5-(1H-pyrazol-1-yl)benzoic acid
N-methyl-N-[(5-phenyl-1H-pyrazol-4-yl)methyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
3-methyl-6-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)pyridazine
(3E)-N-cyclopropyl-N-{[4-(methylsulfanyl)phenyl]methyl}hex-3-enamide
3-(pentan-2-yl)-8-[4-(pyrrolidin-1-yl)butanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(dimethylamino)-3-[4-(1,2-oxazinan-2-ylmethyl)phenoxy]propan-2-ol
(2R)-2-amino-1-{7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}propan-1-one
3-(3-chlorophenyl)-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-3-phenylpropanamide
2-{2-ethoxy-4-[(4-fluoropiperidin-1-yl)methyl]phenoxy}propanoic acid
8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(3-methylbutyl)-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(2-{2-[5-(2-chlorophenyl)furan-2-yl]-1H-imidazol-1-yl}ethyl)imidazolidin-2-one
N-(6-phenoxypyridin-3-yl)-1-(pyrimidin-2-yl)piperidine-4-carboxamide
1-[(4aS,7aR)-4-[(4-methyl-1H-imidazol-5-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carbonyl]cyclopropane-1-carboxamide
4-[2-(dimethylamino)benzoyl]-1-[(3,4-dimethylphenyl)methyl]piperazin-2-one
6-methyl-N-[2-methyl-1-(pyridin-3-yl)propyl]-2-(morpholin-4-yl)pyrimidin-4-amine
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]pyridine-4-carboxamide
methyl 1-{[4-methyl-5-(piperidin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl}piperidine-2-carboxylate
5-[2-(pyrrolidin-1-yl)benzoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
{1-[2-(3-ethoxyphenoxy)ethyl]piperidin-4-yl}methanol
N-(furan-2-ylmethyl)-3-{[(1H-indol-5-yl)carbamoyl]methyl}morpholine-4-carboxamide
ethyl 5-({[1-cyclohexyl-4-oxo-5-(pyrrolidine-1-carbonyl)-1,4-dihydropyridin-3-yl]formamido}methyl)furan-2-carboxylate
3-{[methyl(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)carbamoyl]amino}-N-(2-methylpropyl)benzamide
2-({[(3R,4R)-4-(hydroxymethyl)-1-(4-phenylbenzoyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
1-methyl-6-(propan-2-yl)-N-[3-(pyridin-3-yloxy)propyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(dimethyl-1,3-thiazol-5-yl)-N-[2-(pyridin-2-ylsulfanyl)ethyl]acetamide
2-{[3-(3-methoxybenzoyl)piperidin-1-yl]methyl}pyridine
2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-(oxolan-3-ylmethyl)-1,3-oxazole-4-carboxamide
8-[(1-cyclopentyl-1H-imidazol-5-yl)methyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one