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1-[(1-benzyl-1H-pyrazol-4-yl)methyl]-3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]urea
N'-(2-fluoro-5-methylphenyl)-N-[3-oxo-3-(pyrrolidin-1-yl)propyl]butanediamide
(1R,2R,6S,7S)-N-[3-(pyridin-3-yl)phenyl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane-4-carboxamide
1-[2-methoxy-4-({[2-(4-methylphenyl)ethyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
4-[4-(dimethylamino)phenyl]-1-methyl-3-(pyridin-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-(3-chloro-4-fluorophenoxy)-1-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]ethan-1-one
N-[(2,6-difluoro-3-methoxyphenyl)methyl]-1,9-dioxaspiro[5.5]undecan-4-amine
3-[(3R,4S)-1-[(1-methyl-1H-indol-6-yl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
N-[(2,4-dimethoxyphenyl)methyl]-3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
1-{[3-(cyclopropylmethyl)-1-(2,3-dihydro-1H-inden-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{N-methyl-2-[4-methyl-6-(morpholine-4-carbonyl)-3,4-dihydro-2H-1,4-benzoxazin-3-yl]acetamido}acetic acid
N-cyclopropyl-2-[(3-fluorophenyl)methyl]-6-methyl-1-[3-(morpholin-4-yl)propyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
2-[4-(2,1,3-benzothiadiazol-5-ylmethyl)-1-[(4-fluorophenyl)methyl]piperazin-2-yl]ethan-1-ol
methyl 1-[2-(1H-indol-3-yl)ethyl]-5-{[1-(methylsulfanyl)propan-2-yl]amino}-3-(oxolane-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-[(2-methylpyridin-3-yl)oxy]-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}piperidine-4-carboxamide
5-(4-chloro-2-methoxyphenoxymethyl)-N-[(4-ethylphenyl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
3-{[1-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)propan-2-yl]oxy}pyridine
N-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-4-(hydroxymethyl)pyridine-2-carboxamide
N-(3-ethyl-4-methyl-1-phenyl-1H-pyrazol-5-yl)-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
N-cyclopropyl-N-({3-[(1-methylpiperidin-3-yl)methoxy]phenyl}methyl)furan-2-carboxamide
2-hydroxy-4-methyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]benzamide
4-[3-(4-{[2-(dimethylamino)ethyl](methyl)amino}piperidine-1-carbonyl)phenyl]-2-methylbutan-2-ol
1-(3-{4-chloro-2-[(3-methoxypyrrolidin-1-yl)methyl]phenoxy}propyl)-1H-imidazole
N-({1-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]piperidin-3-yl}methyl)-4-phenylbenzamide
5-methoxy-2-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}phenol
5-(4-cyclohexylpiperazine-1-carbonyl)-1-[(2-methoxyphenyl)methyl]piperidin-2-one
N-(1H-imidazol-2-ylmethyl)-5-{[(4-methoxynaphthalen-1-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
N,5-dimethyl-N-(propan-2-yl)-4-[(1,2,3,4-tetrahydronaphthalen-1-yl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
N-benzyl-2-[4-(2-methoxyphenyl)-3-oxopiperazin-1-yl]propanamide
2-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-6-(trifluoromethyl)pyridine
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-(2-oxoazepan-3-yl)acetamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-[N-(4-methylphenyl)methanesulfonamido]acetamide
4-(2-hydroxynaphthalene-1-carbonyl)-1-(4-methylphenyl)piperazin-2-one
2-(2-methyl-1H-1,3-benzodiazol-1-yl)-N-(1-methyl-1H-indazol-3-yl)acetamide
8-methyl-2-[2-oxo-2-(3-phenylpiperazin-1-yl)ethyl]-2,8-diazaspiro[4.5]decan-3-one
1-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-[4-(methylsulfanyl)phenyl]ethan-1-one
methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]{[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]methyl}amine
ethyl 4-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-3-yl}piperazine-1-carboxylate
2-(2-hydroxyethyl)-8-(3-phenoxypropanoyl)-2,8-diazaspiro[5.5]undecan-3-one
5-cyclopropyl-N-(1,4-dioxan-2-ylmethyl)-1-{8-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-N-methyl-1H-pyrazole-4-carboxamide
N-methyl-2-(4-propanoylphenoxy)-N-(quinolin-5-ylmethyl)acetamide
1-[2-(1-{3-[4-(dimethylamino)phenyl]propanoyl}piperidin-2-yl)ethyl]pyrrolidin-2-one
N-[2-(4-fluorobenzenesulfonyl)ethyl]-1,9-dioxaspiro[5.5]undecan-4-amine
(3S,4R)-4-(4-fluorophenyl)-1-(2-methyl-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)pyrrolidine-3-carboxylic acid
4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-methylpiperidine
5-methyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
methyl 4-oxo-1-(propan-2-yl)-5-[2-(trifluoromethyl)morpholine-4-carbonyl]-1,4-dihydropyridine-3-carboxylate
N,N-diethyl-3-(quinolin-5-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
methyl 4-oxo-1-(propan-2-yl)-5-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]-1,4-dihydropyridine-3-carboxylate
2-(3-chlorophenoxy)-1-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one