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1-[1-(2-butoxybenzoyl)piperidin-4-yl]pyrrolidin-2-one
3-[1-(dimethylsulfamoyl)piperidin-3-yl]-N-(4-methoxy-2-methylphenyl)propanamide
5-(2H-1,3-benzodioxol-4-ylmethyl)-3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
(1S,5R)-3-({7-chloro-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[2-(5-methylfuran-2-yl)ethyl]-1-(propan-2-yl)piperidine-4-carboxamide
6-ethyl-3-{4-[(3-fluorophenyl)methyl]-1,4-diazepane-1-carbonyl}-1,5-dimethyl-1,2-dihydropyridin-2-one
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methoxybutan-1-one
2-methoxy-6-{[methyl({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)amino]methyl}phenol
2-(1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}piperidin-4-yl)-4-methyl-1H-1,3-benzodiazole
3-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
(1S,5R)-6-(cyclobutylmethyl)-3-[(1-methyl-1H-indol-6-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-benzyl-1H-pyrazole-3-carboxamide
N-{1-[1-(1-benzylpiperidin-4-yl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide
N-[1-(furan-2-carbonyl)piperidin-4-yl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
1-methyl-2-{1-[2-methyl-2-(morpholin-4-yl)propyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
7-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]-N,N,2-trimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(3S)-1-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]pyrrolidin-3-ol
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-(1,2-oxazinan-2-yl)pyridine-3-carboxamide
3-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-1-[2-methyl-5-(4H-1,2,4-triazol-4-yl)phenyl]urea
2-(2-hydroxyethyl)-N-[2-(4-methoxyphenyl)phenyl]-3-oxopiperazine-1-carboxamide
4-(2,6-difluoro-3-methoxybenzoyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
2,6,8-trimethyl-4-({4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}methyl)quinoline
6-(4-fluorophenyl)-N-methyl-N-[1-(pyridin-3-yl)propyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-{9-[(4-cyanophenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}propanoic acid
3-[4-(pyridin-2-ylmethoxy)piperidine-1-carbonyl]piperidine-1-carboxamide
5-[4-(1-benzyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2-methyl-3,4-dihydropyrimidin-4-one
N,N-dimethyl-5-{[methyl({[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl})amino]methyl}-1,3-thiazol-2-amine
N-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}-1-(pyrimidin-2-yl)piperidin-3-amine
ethyl 2-[4-({[(1-ethyl-1H-imidazol-5-yl)methyl]carbamoyl}amino)phenyl]acetate
2-(4-{[(1S,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}phenoxy)ethan-1-ol
1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-3-({[(3-methylphenyl)methyl]amino}methyl)piperidin-2-one
4-(4-fluorophenyl)-1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}butan-1-one
2-(2-methoxy-4-{[3-(2-methylphenoxy)azetidin-1-yl]methyl}phenoxy)acetamide
8-fluoro-2-[({[1-(2-methoxyethyl)piperidin-3-yl]methyl}(methyl)amino)methyl]quinolin-4-ol
9-(2-methylquinoline-4-carbonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
2-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]-1,2-oxazolidin-4-ol
4-{3H-imidazo[4,5-b]pyridin-5-yl}-1-methyl-1H-pyrrolo[2,3-b]pyridine
1-[2-(2-methoxyethyl)piperidin-1-yl]-3-[4-(3-methylphenyl)piperazin-1-yl]propan-1-one
N-[(2S,4R,6R)-2-[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]-6-(propan-2-yl)oxan-4-yl]acetamide
N-(3,3-diphenylpropyl)-6-(2-oxo-2-phenylacetyl)-6-azaspiro[2.5]octane-1-carboxamide
6-methyl-4-oxo-1-(oxolan-2-ylmethyl)-2-(2-phenylethyl)-N-(pyridin-3-ylmethyl)-1,4-dihydropyridine-3-carboxamide
8-[(6,8-dimethyl-4-oxo-1,4-dihydroquinolin-2-yl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-2-(pyridin-4-ylsulfanyl)ethan-1-one
3-[(3S,7S,8aS)-3-[(benzyloxy)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3,5-dimethylphenyl)urea
4-ethyl-3-{1-[2-(1H-pyrrol-1-yl)pentanoyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
5-(2-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-oxoethyl)-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(3aR,6aR)-2-methanesulfonyl-5-[(4-methyl-1,3-thiazol-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-chloro-2-({4-[(2-chlorophenyl)methyl]-4-(hydroxymethyl)piperidin-1-yl}methyl)phenol
2,5,6-trimethyl-N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}pyrimidin-4-amine