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N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-(5-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)acetamide
(1-methyl-1H-imidazol-2-yl)({1-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-4-yl})methanol
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2-[4-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)morpholin-3-yl]acetamide
4-sulfamoyl-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}butanamide
6-(1H-indol-5-yl)pyridine-3-carboxamide
(4aS,7aR)-1-[(2-aminopyridin-3-yl)methyl]-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[1-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-4-yl]-N-cyclopropylpiperidine-3-carboxamide
ethyl[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl](thiophen-3-ylmethyl)amine
1-ethyl-3-[(2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}phenyl)sulfanyl]pyrrolidine-2,5-dione
5-({2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}methyl)-N-propylpyrimidin-2-amine
N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
2-{1-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-1H-imidazol-2-yl}-1H-1,3-benzodiazole
1-[2-(3,5-dimethyl-1H-pyrazol-4-yl)acetyl]-3-(2-methoxyethyl)piperidine-3-carboxylic acid
(2R)-2-acetamido-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)butanamide
1-[(3-methoxyphenyl)methyl]-4-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]piperazin-2-one
N-{[5-(benzylsulfanyl)-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl]methyl}cyclopropanecarboxamide
3-(1H-imidazol-2-ylmethyl)-9-methyl-3,9-diazaspiro[5.6]dodecan-10-one
5-methyl-N-[(3R,5S)-1-methyl-5-[(propan-2-yl)carbamoyl]pyrrolidin-3-yl]-2-phenyl-1H-imidazole-4-carboxamide
{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}[(1,2-dimethyl-1H-imidazol-5-yl)methyl]amine
1-(6-fluoropyridin-3-yl)-3-methyl-3-(1-methylpyrrolidin-3-yl)urea
2-[cyclopentyl(prop-2-en-1-yl)amino]-2-(4-fluoro-3-methylphenyl)acetic acid
3-methyl-5-{4-[2-(4-methyl-1,3-thiazol-2-yl)-1H-imidazol-1-yl]phenyl}-4H-1,2,4-triazole
3-{2-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]-2-oxoethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[(3-methyl-1H-pyrazol-5-yl)methyl]-4-{[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
N-cyclopentyl-4-(1-phenyl-1H-pyrazol-4-yl)pyrimidin-2-amine
1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}-4-{[1,2,4]triazolo[4,3-a]pyrimidin-5-yl}piperazine
(4aS,8aR)-6-(2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carbonyl)-1-propyl-decahydro-1,6-naphthyridin-2-one
1-cyclopentyl-5-oxo-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]pyrrolidine-3-carboxamide
1-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}azetidin-3-ol
N-{1-[1-(1-phenoxypropan-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-phenylbutanamide
6-cyclopentyl-2-(2-{[4-(propan-2-yl)piperazin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
2-[4-(2-ethylpyrimidine-5-carbonyl)piperazin-1-yl]-1,3-benzothiazole
3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-N-phenylpiperidine-1-carboxamide
2-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-6-methylpyridine-3-carbonitrile
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-2-[(propan-2-yl)amino]pyrimidine-5-carboxamide
2-{3-oxo-9-[2-(pyrrolidin-1-yl)acetyl]-2,9-diazaspiro[5.5]undecan-2-yl}propanoic acid
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-(4-methyl-1H-pyrrole-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-methoxy-5-{5-methyl-[1,2,4]triazolo[4,3-a]pyridin-3-yl}pyrimidine
2-[3-(dimethylamino)pyrrolidin-1-yl]-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
8-[(3-hydroxyphenyl)methyl]-1-[2-(4-methoxyphenyl)ethyl]-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{3-[6-(morpholin-4-yl)pyrimidin-4-yl]piperidine-1-carbonyl}phenol
8-chloro-3-[2-(1-cyclopentylpiperidin-2-yl)ethyl]-3,4-dihydroquinazolin-4-one
3-[(4aR,7aS)-6,6-dioxo-4-[3-(1H-pyrrol-1-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methoxypyridine-3-carboxamide
N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-2-[4-(pyridin-4-ylmethyl)morpholin-3-yl]acetamide
ethyl({[(3R,4S)-1-(5-fluoropyridin-2-yl)-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl})methylamine
1-(2,3-dihydro-1-benzofuran-5-ylmethyl)-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-2-carboxamide
1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-[3-(trifluoromethyl)phenyl]ethan-1-one
N-[(2-fluorophenyl)methyl]-2-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]acetamide
N-(furan-3-ylmethyl)-N-methyl-4-(piperidin-3-yl)benzamide