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N-ethyl-5-(morpholin-4-ylmethyl)-N-propyl-1,2-oxazole-3-carboxamide
4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidine
1-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-1-methyl-3-[5-(4-methylphenyl)-1,3,4-thiadiazol-2-yl]urea
(3S,5R)-1-(1H-imidazol-2-ylmethyl)-5-[(pyridin-3-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
1-(propan-2-yl)-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}piperidine-4-carboxamide
2-(2-hydroxyethyl)-9-[4-(2-methylpropyl)benzoyl]-2,9-diazaspiro[5.5]undecan-3-one
2-methanesulfonyl-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
4-(3,5-dimethyl-1H-pyrazol-1-yl)-1-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}butan-1-one
2-(pyridin-2-yl)-N-[1-(thiophen-2-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-[(3-phenoxyphenyl)methyl]piperazine
[(3R,4R)-1-[2-(benzyloxy)benzoyl]-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl){[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}amine
1-{2-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydropyrimidin-2-one
(3S)-3-{[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]amino}azepan-2-one
2-{[1-(pyrimidin-4-yl)ethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-[(3S,4R)-1-[(2,4-diethoxy-3-methylphenyl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
N-[1-(3,5-difluorophenyl)ethyl]-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-[2-(3-methoxyphenyl)ethyl]-1-(thian-4-yl)piperidine
2-(3-{[3-(piperidin-1-yl)azetidin-1-yl]methyl}phenoxy)ethan-1-ol
2-[3-(2-chloro-4-fluorophenyl)-1H-indazol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
3-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-6-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
1-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(2-fluorophenoxy)piperidine
[7-(3,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
[(1R,2S)-2-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)cyclopentyl]methanol
N-(2-methoxyethyl)-4-{[2-(3-methoxyphenyl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
5-[(1R,2S)-2-propylcyclopropanecarbonyl]-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-[(3S,4R)-3-acetamido-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]-1,3-thiazole-4-carboxamide
2-[2-({4-[(dimethylamino)methyl]-4-hydroxyazepan-1-yl}methyl)phenoxy]acetic acid
1-[1-(5,6-dimethylpyrimidin-4-yl)piperidin-4-yl]-1,4-diazepan-5-one
N-[(2-phenyl-1,3-oxazol-4-yl)methyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
N-[(2-phenoxypyridin-3-yl)methyl]quinoxaline-5-carboxamide
1-[(2,6-dichlorophenyl)methyl]-3-(1-methyl-1H-1,2,4-triazol-5-yl)-1,2-dihydropyridin-2-one
N-cyclopropyl-1-(6-fluoro-2-oxo-1,2-dihydroquinoline-4-carbonyl)piperazine-2-carboxamide
(1R,9aR)-1-[({2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}amino)methyl]-octahydro-1H-quinolizin-1-ol
3-methoxy-1-(6-{[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl}-1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
1'-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-{4-[5-methyl-4-(1-methyl-1H-pyrazol-5-yl)pyrimidin-2-yl]piperazin-1-yl}-1,3-benzoxazole
2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methyl-N-[2-(2-oxopiperidin-1-yl)ethyl]acetamide
(3aS,6aS)-1-oxo-5-(5-phenyl-1,2,4-oxadiazol-3-yl)-2-propyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(4-ethoxyphenyl)methyl]-N,1-bis(2-methoxyethyl)piperidine-4-carboxamide
8-[(4-methoxyphenyl)methyl]-1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-cyclohexyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1,3-benzoxazole-6-carboxamide
7-(cyclopropylmethyl)-2-[6-(methoxymethyl)pyridine-2-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}pyrrolidine-3-carboxamide
2-cyclobutaneamido-N-(2-methylpropyl)-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
1-{2-[5-(3,4-difluorophenyl)-4-phenyl-1H-imidazol-1-yl]ethyl}imidazolidin-2-one
2-[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]-1H-1,3-benzodiazole
5-(dimethylamino)-2-(2-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-2-oxoethyl)-2,3-dihydropyridazin-3-one
4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-[(4-methyl-1H-imidazol-2-yl)methyl]benzamide
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-(pyridin-2-yl)propanamide