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N-(4-{[1-methyl-2,4-dioxo-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decan-8-yl]methyl}phenyl)acetamide
N-[1-(1-methyl-1H-pyrazol-4-yl)propyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
2-{4-cyclopentyl-1-[(3,5-dimethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
2-fluoro-N-(2-hydroxyethyl)-4-methyl-N-[(2-methylphenyl)methyl]benzamide
{1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-[(3-methoxyphenyl)methyl]piperidin-4-yl}methanol
N-methyl-6-(4-methylphthalazin-1-yl)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
3-(1,3-benzothiazol-2-ylmethyl)-1,3-diazinane-2,4-dione
N-[3-({[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]carbamoyl}amino)phenyl]cyclopentanecarboxamide
1-(4-{[3-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl}phenyl)imidazolidin-2-one
1-methyl-4-{3-methyl-5-[(2,3,6-trifluorophenyl)methyl]-1H-1,2,4-triazol-1-yl}piperidine
2-{4-[3-(dimethylamino)benzoyl]-2-oxopiperazin-1-yl}benzonitrile
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-(1H-pyrazol-1-yl)butanamide
4-{1-[1-(pyrimidin-2-ylmethyl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-[(3-fluorophenyl)methyl]benzamide
8-chloro-2-{[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methyl}quinoline
(4-methoxy-4-methylpentan-2-yl)({[3-(1H-pyrazol-1-yl)phenyl]methyl})amine
3-(2H-1,3-benzodioxol-5-yl)-1-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}propan-1-one
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(5,6-dimethylpyrimidin-4-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-2-(2-methyl-1,3-thiazol-4-yl)-N-[3-(2-oxopyrrolidin-1-yl)propyl]acetamide
3-{1-[(5-chloro-1-benzothiophen-3-yl)methyl]-1H-imidazol-2-yl}pyridine
N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)naphthalene-1-carboxamide
2-[3-(hydroxymethyl)-3-(3-methylbut-2-en-1-yl)piperidin-1-yl]pyridine-4-carbonitrile
1-[(dimethyl-1,2-oxazol-4-yl)methyl]-1-methyl-3-(2-methyl-1,3-benzothiazol-6-yl)urea
1-{imidazo[1,2-b]pyridazin-6-yl}-4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperazine
2-{3-[1-(4,4,4-trifluorobutyl)-1H-pyrazol-3-yl]phenyl}pyridine
1-[(4-methanesulfonylphenyl)methyl]-4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
3-[4-(1H-imidazole-2-carbonyl)phenyl]-1H-pyrazole
dimethyl({[1-(5-propyl-1,3,4-oxadiazol-2-yl)piperidin-4-yl]methyl})amine
4-(1H-indol-3-ylmethyl)-7-{[4-(pyridin-2-ylmethyl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
5,7-dimethyl-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
2-(dimethylamino)-2-(2-methylphenyl)-N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}acetamide
4-(4-chloro-1-methyl-1H-indole-2-carbonyl)-1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane
3-(2-oxo-2-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethyl)-1,3-oxazolidin-2-one
1-[4-(1H-pyrazol-1-yl)phenyl]-4-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-yl}piperidine
2-(dimethylamino)-2-(4-fluorophenyl)-N-[(2-fluorophenyl)methyl]-N-(2-hydroxyethyl)acetamide
(2-{2-[1-(2-chloro-4-fluorobenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
1-(furan-3-carbonyl)-4-(2-methylpyridin-4-yl)-1,4-diazepane-6-carboxylic acid
1-ethyl-3-methyl-N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]piperidine-3-carboxamide
3-{2-[2-(dimethylamino)ethyl]piperidine-1-carbonyl}-6-(trifluoromethyl)pyridin-2-ol
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-1,3-oxazole-4-carboxamide
1-{4-[3-(2-phenylethyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
N-(3-cyano-4-methoxyphenyl)-4-sulfamoylpiperazine-1-carboxamide
2-{4-[(2,5-difluorophenyl)methyl]morpholin-3-yl}-N-(1,3-dihydro-2-benzofuran-5-yl)acetamide
1-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one
6-{1-[(4-methanesulfonylphenyl)methyl]piperidin-4-yl}-2-methylpyrimidin-4-ol
9-{2-[(cyclopropylmethyl)sulfanyl]acetyl}-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
dimethyl[(4-{10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}-1,4-oxazepan-6-yl)methyl]amine
N-(1,3-benzothiazol-2-ylmethyl)-1-propyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[2-(3-benzyl-1,2,4-oxadiazol-5-yl)ethyl]-4-(pyridin-3-yl)pyrimidin-2-amine
2-[1-(2-methoxyphenyl)-5-{[(4-methyl-1,3-thiazol-2-yl)sulfanyl]methyl}-1H-1,2,4-triazol-3-yl]acetamide