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[(3R,4R)-1-(3-chloro-4-methoxybenzoyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
5-{[3-(5-chloro-2-methoxybenzoyl)piperidin-1-yl]methyl}-2-(methylsulfanyl)pyrimidine
1-[1'-(4-methyl-1,3-thiazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]pyridin-2-amine
3-{[(2,3-dihydro-1-benzofuran-2-ylmethyl)(methyl)amino]methyl}-N-(1-methyl-1H-1,2,3-triazol-4-yl)benzamide
5-ethyl-N,2,3-trimethyl-N-(1H-pyrazol-3-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
3-methyl-1-[4-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]-3-[3-(oxolan-2-yl)propyl]urea
5-(1H-indol-3-ylmethyl)-N,N-dimethyl-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(methylsulfanyl)propan-1-one
N-[(2-chlorophenyl)methyl]-3-{1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidin-3-yl}propanamide
4-(2-fluoro-4-methylphenyl)-1-[2-(propan-2-ylsulfanyl)ethyl]-1H-1,2,3-triazole
N-[1-(4-fluorophenyl)propyl]-1-methyl-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]cyclopentanecarboxamide
N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-3-(2-oxopiperidin-1-yl)propanamide
8-[2-(methylamino)-1,3-thiazole-4-carbonyl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
1-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
(4-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}morpholin-3-yl)methanol
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)acetamide
2-(2-{[(2-fluorophenyl)methyl](methyl)amino}acetyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
(2S,4S)-1-[(2-chlorophenyl)methyl]-4-{[(2,5-difluorophenyl)methyl]amino}-N-methylpyrrolidine-2-carboxamide
1-[7-chloro-2-(1-ethyl-1H-pyrazol-4-yl)quinoline-4-carbonyl]piperidine-4-carbonitrile
N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-4-(pyridin-3-yl)pyrimidin-2-amine
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}oxane-4-carboxamide
(2S,4S)-4-amino-N-ethyl-1-methyl-N-[(5-methylfuran-2-yl)methyl]pyrrolidine-2-carboxamide
(2-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-oxoethyl)urea
1-(4-methylquinazolin-2-yl)-N-[(4-phenyloxan-4-yl)methyl]pyrrolidine-2-carboxamide
3-{[1-ethyl-3-(1-phenylcyclopropyl)-1H-1,2,4-triazol-5-yl]methyl}-3,4-dihydroquinazolin-4-one
3-{[(2-hydroxyethyl)(methyl)amino]methyl}-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
2-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
5-{[3-hydroxy-2-oxo-1-(2-phenylethyl)piperidin-3-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonitrile
N-[(1S,3S)-3-{[4-(pyridin-4-yl)pyrimidin-2-yl]amino}cyclopentyl]-2-(1H-1,2,4-triazol-1-yl)acetamide
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-sulfonamide
2-(1,2-benzoxazol-3-yl)-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}acetamide
8-(1H-indol-2-ylmethyl)-1-(3-methylbutyl)-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(dimethyl-1,3-thiazol-2-yl)methyl]acetamide
5-[(3R,4S)-3-(3-hydroxypropyl)-4-(morpholin-4-yl)piperidine-1-carbonyl]-2-methylphenol
2-[(3R,4S)-4-(dimethylamino)-3-(3-hydroxypropyl)piperidin-1-yl]-4,6-dimethylpyridine-3-carbonitrile
N-[4-({[(1-methyl-1H-imidazol-2-yl)methyl]carbamoyl}methyl)phenyl]cyclopropanecarboxamide
N-[1-(3-fluoro-4-methoxyphenyl)ethyl]-4-(1H-pyrazol-3-yl)benzamide
2-(dimethylamino)-N-{2-[(4-fluorophenyl)formamido]ethyl}-2-(3-methylphenyl)acetamide
4-[4-(2-hydroxyethyl)-1H-1,2,3-triazol-1-yl]-N-[(1S)-1-phenylethyl]piperidine-1-carboxamide
2-(2,4-dichlorophenoxy)-1-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}ethan-1-one
1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-1,2-dihydroquinoxalin-2-one
(2,1,3-benzoxadiazol-4-ylmethyl)(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
2-benzyl-9-(6-oxo-1,6-dihydropyrimidine-5-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
4-(4-butyl-1H-1,2,3-triazol-1-yl)-1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}piperidine
1-[(4-methoxypiperidin-1-yl)sulfonyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
3-(1,2-dihydroacenaphthylene-5-carbonyl)-1-(1-ethyl-1H-pyrazole-4-carbonyl)piperidine
4-{1-[4-(4-methyl-1H-pyrazol-3-yl)piperidin-1-yl]-1-oxopropan-2-yl}-1,2-dihydrophthalazin-1-one