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1-(3,4-dichlorophenyl)-4-{5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}piperazine
7-[(2-fluorophenyl)methyl]-2-(4,4,4-trifluorobutyl)-2,7-diazaspiro[4.5]decan-6-one
[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl][3-(1H-imidazol-1-yl)propyl](pyridin-3-ylmethyl)amine
N,N-dimethyl-1-[3-(1H-pyrazol-1-yl)benzoyl]azepan-4-amine
1-(7-chloro-3-{[(thiophen-2-ylmethyl)amino]methyl}quinolin-2-yl)piperidin-3-ol
1-(2,3-dihydro-1H-indol-1-yl)-2-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]ethan-1-one
2-[4-(3-chloropyridin-2-yl)-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl]ethan-1-ol
(2S)-2-hydroxy-1-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}-3-phenylpropan-1-one
3-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-1-(2-methyl-1H-1,3-benzodiazol-6-yl)urea
7-(cyclobutylmethyl)-2-{2-methylthieno[2,3-d]pyrimidin-4-yl}-2,7-diazaspiro[4.5]decan-6-one
(1S,5R)-6-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-[1-(hydroxymethyl)cyclohexyl]-3,4,7-trimethyl-1H-indole-2-carboxamide
methyl 6-[2-oxo-7-(2-oxoimidazolidin-1-yl)-1,2,3,4-tetrahydroquinolin-4-yl]pyridine-2-carboxylate
5-{methyl[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]carbamoyl}-2,1,3-benzoxadiazol-1-ium-1-olate
1-ethyl-4-({4-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-1-yl}methyl)-1H-pyrrole-2-carbonitrile
5-{[2-(cyclohex-1-en-1-yl)ethyl]amino}-1-methyl-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
5-[4-(3-methoxybenzoyl)piperazine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(2,4-dichlorophenoxy)-N-[(3S,4R)-4-ethoxyoxolan-3-yl]acetamide
N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
1-phenyl-4-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]butane-1,4-dione
N-(2-hydroxy-2-phenylethyl)-N-methyl-2-(3-phenylpropyl)-1,3-benzoxazole-5-carboxamide
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-2-(dimethylamino)-4-methylpyrimidine-5-carboxamide
3-({[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}amino)-N-(2,4,6-trimethylphenyl)propanamide
N-tert-butyl-2-(4-{1,3-dimethyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}phenoxy)acetamide
2-[1-(propan-2-yl)piperidin-4-yl]-N-[2-(1H-pyrrol-1-yl)ethyl]acetamide
4-{[(2-methylphenyl)methyl]amino}-N-[2-(morpholin-4-yl)ethyl]pyridine-2-carboxamide
2-ethyl-N-[3-(1H-imidazol-1-yl)-1-phenylpropyl]-4-methyl-1,3-oxazole-5-carboxamide
2-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
[1-(1-cyclobutanecarbonylpiperidin-4-yl)-3-(cyclopropylmethyl)piperidin-3-yl]methanol
N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
9-[(3,4-dimethylphenyl)methyl]-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-1,4-diazepane-6-carboxylic acid
1-(2-ethoxyethyl)-2-oxo-N-[2-(2-oxopyrrolidin-1-yl)ethyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
4-(methylsulfanyl)-2-[2-(4-phenylpiperidin-1-yl)acetamido]butanoic acid
5-(2-{[(4-methoxyphenyl)methyl]amino}ethyl)-1-[2-(thiophen-2-yl)ethyl]pyrrolidin-2-one
4-[4-(4-fluorophenyl)-1H-1,2,3-triazol-1-yl]-1-(thian-4-yl)piperidine
1-[(4-fluoro-2-methylphenyl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-[2-oxo-2-(2-phenylmorpholin-4-yl)ethyl]-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
1-[4-(3-aminopyrrolidin-1-yl)-2-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
3-{[(hexahydro-1H-pyrrolizin-7a-ylmethyl)amino]methyl}-3-hydroxy-1-(3-phenylpropyl)piperidin-2-one
4-(2-phenylmorpholine-4-carbonyl)-2-(1H-pyrazol-4-yl)quinoline
(3S,7S,8aS)-3-(4-aminobutyl)-7-{[(4-phenyl-1,3-thiazol-2-yl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
2-[2-(1H-imidazol-1-yl)ethyl]-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidine
(1R,5R)-6-[5-(hydroxymethyl)furan-2-carbonyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
N-cyclopentyl-3-[(1H-imidazol-2-ylmethyl)sulfamoyl]benzamide
2-(1H-1,3-benzodiazol-1-yl)-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]acetamide
1-(furan-2-ylmethyl)-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]piperidine-3-carboxamide
5-{1-[3-(2-methyl-1H-imidazol-1-yl)propyl]-4-phenyl-1H-imidazol-5-yl}isoquinoline
6-cyclopentyl-2-[4-({methyl[2-(1H-pyrazol-4-yl)ethyl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
N-methyl-2-[1-(3-phenylbutyl)piperidin-4-yl]acetamide