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3-(1H-1,3-benzodiazol-2-yl)-1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]propan-1-one
(2R)-N-[(7S,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-hydroxy-2-(naphthalen-2-yl)acetamide
2-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}-N-(propan-2-yl)acetamide
methyl 4-{4-[3-(6-oxo-1,6-dihydropyridazin-3-yl)propanoyl]piperazin-1-yl}benzoate
1-[(4-methyl-5-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]azepane
3-{[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}benzonitrile
2-[4-(5-ethylpyrimidin-2-yl)-1-(2-methylpropyl)piperazin-2-yl]ethan-1-ol
2-[1-(3-methylbut-2-en-1-yl)-4-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl]ethan-1-ol
4-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]-3-(3-fluorophenyl)-1H-pyrazole
N-(2-{[(4-{3-[benzyl(methyl)amino]-2-hydroxypropoxy}phenyl)methyl]amino}ethyl)acetamide
7-(2-cyclohexylethyl)-2-(2-cyclopentylacetyl)-2,7-diazaspiro[4.5]decan-6-one
2-methyl-5-(4-{4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}phenyl)-1,3,4-oxadiazole
1-(1-ethyl-1H-1,2,4-triazol-3-yl)-3-methyl-3-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]urea
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-N-methyl-2-oxo-1,2-dihydroquinoline-4-carboxamide
3-[(3R,4S)-4-(dimethylamino)-1-{2-[methyl(pyridin-3-ylmethyl)amino]acetyl}piperidin-3-yl]propanoic acid
4-(2-methoxyphenoxy)-1-(4-methyl-1H-imidazole-2-carbonyl)piperidine-4-carboxylic acid
4-(3,4-diethoxyphenyl)-2-(4-methyl-1H-imidazol-5-yl)-1H-imidazole
9-(3,6-dimethylpyrazin-2-yl)-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(3-{[2-(3-methoxyphenyl)azetidin-1-yl]methyl}-1H-indol-1-yl)propanamide
4-(5-methyl-4-phenyl-1H-imidazol-2-yl)-1-(2-methylpropyl)pyrrolidin-2-one
(4aS,8aR)-1-(3-aminopropyl)-6-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
methyl 2-hydroxy-5-({2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-1-yl}methyl)benzoate
4-fluorophenyl (7R,9aR)-6,9-dioxo-7-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
5-benzyl-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
8-[1-(2-methyl-1H-imidazol-1-yl)propan-2-yl]-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[1-(4-chloro-1-methyl-1H-pyrazole-5-carbonyl)piperidine-4-carbonyl]-1,2,3,4-tetrahydroisoquinoline
3-cyclopropyl-5-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
2-{5-[(8-methoxyquinolin-2-yl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
4-[1-(5-chloro-2-methoxyphenyl)-3-cyclopropyl-1H-1,2,4-triazol-5-yl]-1-(prop-2-en-1-yl)pyrrolidin-2-one
N-[(3S,5S,9S)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]-2,3-difluorobenzamide
1-[(2-methyl-1,3-oxazol-4-yl)methyl]-4-[(3-methylpyridin-2-yl)methyl]piperazine
N-[1-(1H-imidazol-1-yl)butan-2-yl]-3-(piperidin-4-ylmethyl)benzamide
2-(5-methyl-1H-pyrazol-1-yl)-1-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethan-1-one
1-ethyl-5-{[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)quinoline-3-carboxamide
4-benzyl-3-{1-[2-(pyrrolidin-1-yl)acetyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
6-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-2-methyl-2,3-dihydropyridazin-3-one
N-methyl-5-[(2-methyl-4-oxo-1,4-dihydroquinolin-1-yl)methyl]furan-2-carboxamide
1-[4-(2-methylphenyl)-1,4-diazepan-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-1-methyl-1H-pyrazole-3-carboxamide
4-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepane-1-carbonyl]-N-methylpyridin-2-amine
2-(1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}pyrrolidin-2-yl)-1,3-benzothiazole
methyl (1R,3S,3aR,6aS)-3-(6-methoxy-2H-chromen-3-yl)-1,5-dimethyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
(1S,9S)-11-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
5-[1-(3-methylbutyl)-3-(morpholine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]quinoxaline
N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
(5-{1-[2-(hydroxymethyl)-1H-1,3-benzodiazol-5-yl]-1H-imidazol-2-yl}furan-2-yl)methanol
5-{[2-(3-methoxypropyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]methyl}-N-methyl-1,2,4-oxadiazole-3-carboxamide
4-{4-[(2-fluoro-4-methoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazine-1-carbonyl}phenol
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-(2-oxo-1,2-dihydropyridin-1-yl)acetamide