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(4aS,7aR)-1-[6-(2-hydroxyethyl)pyrazolo[1,5-a]pyrimidine-3-carbonyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(2-aminoacetyl)-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
3-({ethyl[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]carbamoyl}amino)-4-methoxy-N-methylbenzamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-7-(2-methoxyacetamido)-1-methyl-2-phenyl-1H-1,3-benzodiazole-5-carboxamide
7-chloro-3-(2-methoxyethyl)-3,4-dihydroquinazolin-4-one
2-[4-(2-phenylphenyl)-1H-pyrazol-1-yl]acetic acid
2-methyl-N-{[7-(4-phenylbenzoyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}butanamide
4-(3-fluorophenoxy)-1-(5-methyl-1,3-oxazole-4-carbonyl)piperidine-4-carboxylic acid
3-(2-hydroxyethyl)-1-[3-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]-3-[(5-methylthiophen-2-yl)methyl]urea
2-{5-[4-(dimethylamino)phenyl]-1H-indazol-1-yl}-N-(2-ethyl-2H-1,2,3-triazol-4-yl)acetamide
4,4,4-trifluoro-1-{3-[(4-fluorophenyl)amino]piperidin-1-yl}butan-1-one
(3S,4R)-1-[2-methyl-2-(piperidin-1-yl)propyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
2-methyl-4-phenyl-9-(9H-purin-6-yl)-2,9-diazaspiro[5.5]undecan-3-one
3-(3-methoxyphenyl)-5-(thiophene-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
2,6-dimethyl-5-(2-oxo-2-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}ethyl)-3,4-dihydropyrimidin-4-one
4-fluoro-3-methyl-N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]benzamide
2-{1-[(1-methyl-4-phenylpiperidin-4-yl)methyl]-1H-imidazol-2-yl}benzoic acid
3-[(5-chlorothiophen-2-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-(2-methyl-1H-imidazol-4-yl)-1,2,3,4-tetrahydroisoquinoline
N-(2-ethoxyethyl)-3-{[(3R)-piperidin-3-yl]sulfamoyl}benzamide
N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
N-(2-methanesulfonylethyl)-3-(4-methylphenyl)-1H-pyrazole-5-carboxamide
2-methyl-3-[(4-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}piperidin-4-yl)oxy]pyridine
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperazine
methyl (2S)-3-methyl-2-({1-[1-(3-phenylpropyl)piperidin-4-yl]piperidin-4-yl}formamido)butanoate
4-(2,6-dimethylpyridin-3-yl)-N-[1-(pyridin-4-yl)propan-2-yl]pyrimidin-2-amine
1-(cyclohexylmethyl)-N-[3-(1H-pyrazol-1-yl)propyl]piperidin-3-amine
N4-[1-(4-cyclopentyl-4H-1,2,4-triazol-3-yl)ethyl]-6-(propan-2-yloxy)pyrimidine-2,4-diamine
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-2-(pyridin-4-yl)pyrimidine-5-carboxamide
2-{4-[4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)quinolin-2-yl]-1H-pyrazol-1-yl}ethan-1-ol
3-[(benzylamino)methyl]-1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxypiperidin-2-one
5-[3-(methylcarbamoyl)benzenesulfonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
2-(2H-1,3-benzodioxol-5-yl)-1-[9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
5-[4-(2-methoxyphenyl)piperazine-1-carbonyl]-2-(pyridin-4-yl)pyrimidine
2-(2-cyclopentylacetyl)-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
N-(1,4-dioxan-2-ylmethyl)-2-[(5-methyl-1H-1,3-benzodiazol-2-yl)sulfanyl]acetamide
4-tert-butyl-N-{3-[4-(4-methylpiperazine-1-carbonyl)-1H-1,2,3-triazol-1-yl]propyl}benzamide
N,N-diethyl-1-{1-[3-(trifluoromethyl)benzoyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
9-methoxy-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-3-(5-phenylpentanoyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-2,3-dihydro-1,2-benzothiazol-3-one
N-({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}methyl)-2,2-dimethyloxane-4-carboxamide
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl][2-(1H-imidazol-4-yl)ethyl]amine
5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-(piperidin-4-yl)pyridin-2-amine
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-(1H-indazol-3-yl)acetamide
2-({4-[3-(2-aminoethyl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)ethan-1-ol
(2S)-4-methyl-2-{[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]formamido}pentanoic acid
4-({4-amino-6-[(3-methylphenyl)amino]-1,3,5-triazin-2-yl}methyl)-1,4-oxazepan-6-ol
1-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-[1-(2-methylphenyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridine
3-{5-[(3-methylquinoxalin-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
3-(5-{3-[(4-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)phenol