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3-{[(butan-2-yl)(pyridin-4-ylmethyl)amino]methyl}-N-methylpyridin-2-amine
N-{3-methyl-1-[7-(2-methylpropyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]butyl}pyridine-3-carboxamide
1-ethyl-4-{[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}piperazine
1-{1-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-4-phenylpiperidin-4-yl}ethan-1-one
4-(2,3-dihydro-1-benzofuran-5-carbonyl)-N-(3-methylphenyl)morpholine-2-carboxamide
N-methyl-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}acetamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methyl-6-propylpyrimidin-4-amine
(1R,5S,8S)-N-[4-ethoxy-3-(trifluoromethyl)phenyl]-8-methoxy-3-azabicyclo[3.2.1]octane-3-carboxamide
2-hydroxy-N-[(3R,4S)-1-(1-phenylpiperidin-4-yl)-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
5-(2-chloro-4-fluorophenyl)-1-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole
N-(pyridin-2-ylmethyl)-2-[2-(trifluoromethyl)morpholin-4-yl]acetamide
1-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-3-phenylpiperazine
2-[3-benzyl-1-(4-methoxyphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-ethyl-N-methylacetamide
1-(cyclopropylmethyl)-4-(6-methylpyridine-2-carbonyl)-2-(propan-2-yl)-1,4-diazepane
ethyl 3-[(3-methoxyphenyl)methyl]-1-(oxane-4-carbonyl)piperidine-3-carboxylate
4-(4-methoxyphenyl)-1-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}butan-1-one
4-(1H-pyrazol-3-yl)-N-[1-(thian-4-yl)piperidin-4-yl]benzamide
1,6-dimethyl-2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1H-indole
5-[(3R,4R)-3-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
6-[(oxolan-3-ylmethyl)amino]-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
3-(5-{[1-(propan-2-yl)piperidin-4-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)benzonitrile
N-cyclohexyl-2-{[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]amino}butanamide
2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-N-[2-(pyridin-4-yl)ethyl]-1,3-oxazole-4-carboxamide
3-[({5-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]pyridin-2-yl}amino)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(5-methylfuran-2-yl)-N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-1H-pyrazole-5-carboxamide
3-ethyl-1-{[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperidin-3-ol
3-cyclopropyl-1-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]propan-1-one
methyl 2-(azocane-1-sulfonyl)-6-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-{4-[5-(azepan-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-cyclopropylethan-1-one
3-cyclopropyl-3-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)urea
1-(3-carboxybenzoyl)-4-(pyrimidin-2-yl)piperazine-2-carboxylic acid
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
1-{1-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]piperidin-4-yl}-2-phenylethan-1-ol
3-[5-(2-cyclohexylethyl)-1,3,4-oxadiazol-2-yl]-N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}propanamide
1'-(8-methoxy-4-methylquinolin-2-yl)-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(2S,4S,5R)-4-[(carboxymethyl)carbamoyl]-5-(4-chlorophenyl)-1,2-dimethylpyrrolidine-2-carboxylic acid
1-{5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidin-3-ol
3-methyl-7-(2,4,5-trimethoxybenzoyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
(5-{1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-phenyl-1H-imidazol-5-yl}furan-2-yl)methanol
5-(2-{[(2-chloro-4-fluorophenyl)methyl]amino}pyrimidin-4-yl)-2-ethoxybenzoic acid
14-(5-chloro-2,3-dimethoxyphenyl)-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
4-{7-[(2S)-2-hydroxypropanoyl]-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl}benzamide
1-[(2-ethyl-1,3-thiazol-4-yl)methyl]-4-(2-methylpropyl)pyrrolidin-2-one
1-{8-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)ethan-1-one
3-{5-[4-(2-methyl-1H-imidazol-1-yl)butanoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
1-{1-[(5-methylthiophen-2-yl)methyl]azetidin-3-yl}piperidine
2-(3-chloro-4-hydroxyphenyl)-1-{4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]piperidin-1-yl}ethan-1-one
6-ethyl-2-oxo-N-{[1-(phenoxymethyl)cyclopropyl]methyl}-1,2-dihydropyridine-4-carboxamide
{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}(2-methoxyethyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
4-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyridin-2-amine