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11-{[(2-methylphenyl)methyl]amino}-4-(pyridin-2-ylmethyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-(2-aminoethyl)-4-(2-ethoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{4-[2-(1,2-benzoxazol-3-yl)acetyl]morpholin-3-yl}-N-(pyridin-3-yl)acetamide
2-{methyl[(4-methyl-5-{1-[(2-methylpyrimidin-5-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]amino}ethan-1-ol
[(1,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl){[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}amine
3-[(3S,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[3-(trifluoromethyl)phenyl]urea
4-[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]-6-(2-methylpropyl)pyrimidin-2-amine
N-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-N-[(1-methyl-1H-imidazol-2-yl)methyl]cyclopropanamine
(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-{[5-(2-methylpropyl)thiophen-2-yl]methyl}piperidin-3-ol
2-(1-ethylpiperidin-4-yl)-N-[1-(6-methylpyridin-3-yl)ethyl]acetamide
2-(4-{imidazo[1,2-b]pyridazine-3-carbonyl}morpholin-3-yl)-N-(2-methylpropyl)acetamide
1-(4-methoxyphenyl)-N-{[5-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclopentane-1-carboxamide
2-[3-(2-chlorophenyl)-1-methyl-2,5-dioxopyrrolidin-3-yl]-N-[(4-ethylphenyl)methyl]-N-methylacetamide
1-[2-(4-chlorophenyl)ethyl]-N-[3-(2-methoxyphenyl)propyl]-6-oxopiperidine-3-carboxamide
1-(4-ethylpiperazin-1-yl)-3-[1-(pyridin-4-ylmethyl)piperidin-4-yl]propan-1-one
2-(5-acetylthiophen-3-yl)-N-(2-oxoazepan-3-yl)acetamide
N-(2-{4-[1-(3-methylpyridin-2-yl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}ethyl)acetamide
N-(3-hydroxypropyl)-1-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidine-3-carboxamide
(4aS,8aR)-1-(3-methoxypropyl)-6-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
6-methyl-5-(2-oxo-2-{4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}ethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-[methyl(2-phenylethyl)amino]-2-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}-2,3-dihydropyridazin-3-one
6-(2-chlorophenyl)-7-(cyclopropylmethyl)-2-(piperidine-1-carbonyl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
2-(3-chlorophenyl)-N-[4-(4-{[1-(thiophen-2-yl)propan-2-yl]amino}piperidin-1-yl)phenyl]acetamide
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-methyl-5-oxo-1-[4-(propan-2-yl)phenyl]pyrrolidine-3-carboxamide
5-(6-fluoro-2-oxo-1,2-dihydroquinoline-4-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
N-[2-(1H-imidazol-4-yl)ethyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-[4-(azocane-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethan-1-amine
2-(2-{[1-(pyridin-4-yl)propyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[5-(azepan-1-ylmethyl)-2-methoxyphenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
7-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-methoxy-3-[5-(piperidine-1-carbonyl)-1H-pyrrol-3-yl]quinoline
N-(4-{3-[1-(1,4-dioxan-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}phenyl)-N-methylacetamide
1-(6-hydroxy-1,4-oxazepan-4-yl)-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-1-[(4-methylphenyl)amino]cyclopentane-1-carboxamide
2-{4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
3-(4-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl}-4-oxobutyl)-3,4-dihydroquinazolin-4-one
N-(2-{1-[(4-methylphenyl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}ethyl)morpholine-4-carboxamide
4-{2-ethyl-3-methyl-6-oxo-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}-2,6-dimethylphenyl acetate
14-(3-ethyl-1,2-oxazol-5-yl)-5-methyl-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
2-(3-{[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}phenyl)ethan-1-amine
N5-[(3,5-difluorophenyl)methyl]-N3-methyl-N3-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
2-[4-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-1-yl]propanamide
7-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
N-{2-[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-oxoethyl}acetamide
5-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidine-1-carbonyl]-N,N,4-trimethylpyrimidin-2-amine
2-{2-[6-(methylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]phenoxy}propanamide
2-hydroxy-1-[4-(3-methylpyridin-2-yl)piperazin-1-yl]-4-(methylsulfanyl)butan-1-one
{1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}diphenylmethanol
3-({[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)propan-1-ol