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(4aR,7aS)-1-{2-[4-(methoxymethyl)piperidin-1-yl]pyrimidin-4-yl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]-3-(pyridin-4-yl)propan-1-one
1-(4-{1-phenyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenyl)-1H-1,2,4-triazole
1-[2-amino-6-(pyrrolidin-1-yl)pyrimidin-4-yl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
1-[(4-methoxyphenyl)methyl]-5-(2-methylpentanoyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-butyl-N-(furan-2-ylmethyl)-3-(piperidine-1-carbonyl)pyrazine-2-carboxamide
N-[(1-phenylcyclopentyl)methyl]-3-(pyridin-3-yl)propanamide
(1S,5R)-6-(5-methylthiophene-3-carbonyl)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-[(3aR,5S,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-3-(1H-1,3-benzodiazol-1-yl)propan-1-one
4-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
(3aS,6aS)-N,N-dimethyl-5-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]-octahydropyrrolo[2,3-c]pyrrole-1-carboxamide
N-[(3R,4S)-1-(cyclobutylmethyl)-4-(propan-2-yl)pyrrolidin-3-yl]cyclopropanecarboxamide
4-[(2S)-2-(methylamino)propanoyl]-1-(2-phenylphenyl)piperazin-2-one
5-{[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]methyl}-N,N-dimethylfuran-2-carboxamide
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetamide
1-acetyl-N-[2-(1H-pyrrol-1-yl)ethyl]piperidine-3-carboxamide
(1R,5R)-N,N-dimethyl-6-(thiophene-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
2-(4-{[methyl(oxan-4-ylmethyl)amino]methyl}phenyl)-3H,4H,5H,6H,7H,8H,9H-cyclohepta[d]pyrimidin-4-one
2-[({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amino]-N-(1,3-thiazol-2-yl)acetamide
3-(diphenylmethyl)-5-ethyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amine
2-{1-[(1-{spiro[2.5]octane-1-carbonyl}piperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}pyridine
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
N-[(3-methoxyphenyl)methyl]-3-[1-(2-methyl-1H-pyrrole-3-carbonyl)piperidin-3-yl]propanamide
4-(2-hydroxyethyl)-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-amino-4-chloro-N-[1-(2-hydroxyethyl)piperidin-4-yl]-1H-pyrazole-3-carboxamide
2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)-N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N-methylacetamide
5-[(4-benzylpiperidin-1-yl)methyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,2-oxazole-3-carboxamide
ethyl 3-[(2-methylphenyl)methyl]-1-(propane-1-sulfonyl)piperidine-3-carboxylate
3-(2-methoxyethyl)-1-(2-phenylethyl)-8-(pyridin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{1-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]piperidin-3-yl}benzoic acid
3-methyl-7-(6-phenylpyridazin-3-yl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
8-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-3,7-dimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-dione
(1R,7S)-3-tert-butyl-6-(5,6,7,8-tetrahydro-1,6-naphthyridine-6-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
1-[3-(diethylamino)pyrrolidin-1-yl]-2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethan-1-one
5-{[4-hydroxy-4-(hydroxymethyl)piperidin-1-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-[2-(4-methoxyphenoxy)ethyl]-4,5-dimethyl-2,3-dihydro-1,3-oxazol-2-one
N-[(4-ethoxyphenyl)methyl]-N-(2-methoxyethyl)azepane-4-carboxamide
4-{[3-(2-hydroxyethyl)-4-[(5-methylfuran-2-yl)methyl]piperazin-1-yl]methyl}phenol
1-(carboxymethyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylic acid
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]propan-1-one
1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-N-(3-phenylpropyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[3-(4-{[2-(azepan-1-yl)-2-phenylethyl]amino}piperidin-1-yl)phenyl]ethane-1-sulfonamide
2-chloro-5-{5-[(4-propylpiperazin-1-yl)methyl]furan-2-yl}benzoic acid
2-(2,3-difluorophenoxymethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,3-oxazole-4-carboxamide
1-cyclohexyl-N-cyclopropyl-5-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-4-oxo-1,4-dihydropyridine-3-carboxamide
4-amino-2-(8-methoxy-2-methylquinolin-5-yl)pyrimidine-5-carbonitrile
(3aS,6aS)-2-[(dimethyl-1,3-thiazol-4-yl)methyl]-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-ol
1-{[1-(cyclohexylmethyl)-3-methyl-1H-1,2,4-triazol-5-yl]methyl}-1,2-dihydropyridin-2-one