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N5-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-N6-(3-methoxypropyl)-N5-methyl-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
2-(pyridin-3-yl)-5-[3-(pyridine-3-carbonyl)piperidine-1-carbonyl]pyrimidin-4-ol
3-{2-[2-(furan-2-yl)pyrrolidin-1-yl]-2-oxoethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-cyclopropyl-9-[2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
N-{[(2S,4S)-4-fluoro-1-[(3R)-1,2,3,4-tetrahydroisoquinoline-3-carbonyl]pyrrolidin-2-yl]methyl}ethane-1-sulfonamide
1-(4-fluorophenyl)-4-(furan-3-carbonyl)-1,4-diazepane
N-({1-[(5-chloro-3-methyl-1H-indol-2-yl)methyl]pyrrolidin-3-yl}methyl)acetamide
(1R,6S)-9-methyl-N-(2-methyl-1,3-benzothiazol-5-yl)-3,9-diazabicyclo[4.2.1]nonane-3-carboxamide
4-(2-phenylpyrrolidine-1-carbonyl)-1,2-dihydroquinolin-2-one
(1S,5R)-6-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonane
N2-[2-(1-benzylpiperidin-4-yl)ethyl]-5-fluoro-N4,N4-dimethylpyrimidine-2,4-diamine
1-cyclobutanecarbonyl-3-[2-(2,6-difluorophenyl)ethyl]piperidine
2-({1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}oxy)-4-methoxy-N-(2-methoxyethyl)benzamide
1-(2-benzylmorpholin-4-yl)-4-(1H-1,2,4-triazol-1-yl)butan-1-one
(4aR,8aS)-1-[2-(3-chlorophenoxy)propanoyl]-N,N-dimethyl-decahydro-1,6-naphthyridine-6-sulfonamide
(1-{1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]piperidin-3-yl}piperidin-4-yl)methanol
1-(furan-3-carbonyl)-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-(cyclopentylmethyl)-6-methyl-4-oxo-1-(pyridin-3-ylmethyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,4-dihydropyridine-3-carboxamide
1-[6-(quinolin-8-yl)pyridin-2-yl]ethan-1-ol
N-benzyl-4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidine-1-sulfonamide
{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[(3-methoxyphenyl)methyl]methylamine
(1R,5R)-N-[(4-chlorophenyl)methyl]-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
2-({4-[2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)acetyl]piperazin-1-yl}methyl)benzonitrile
(3R)-1-(4-methoxypyrimidin-2-yl)-3,4,4-trimethylpyrrolidin-3-ol
3-(pentan-2-yl)-8-(pyridazine-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[1-(hydroxymethyl)cyclopentyl]-5-(2-methoxy-4-methylphenoxymethyl)-1,2-oxazole-3-carboxamide
2-methyl-6-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
N-(2,2-dimethyloxan-4-yl)-1-[4-(1H-pyrazol-1-yl)phenyl]piperidin-4-amine
2-{[3-(aminomethyl)pyrrolidin-1-yl]methyl}-6-methoxyphenol
N-[(3S,4R)-4-(propan-2-yl)-1-{[2-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-3-yl]acetamide
N-[1-(dimethyl-1,3-thiazol-2-yl)propyl]-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide
(2S,4R)-1-[(3-chlorophenyl)methyl]-4-{[(4-methoxy-2,3-dimethylphenyl)methyl]amino}-N-methylpyrrolidine-2-carboxamide
3-(4-{[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}piperazin-1-yl)propan-1-ol
(3aR,6aR)-2-(oxan-4-yl)-5-(5-propylpyrimidin-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(2-{3-[(4-methoxyphenyl)amino]piperidine-1-carbonyl}thiophen-3-yl)acetamide
1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-2-(2-hydroxyphenyl)ethan-1-one
3-(azepane-1-carbonyl)-1-ethyl-N-[2-(propan-2-yloxy)ethyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
7-(5-propyl-1,2-oxazole-3-carbonyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
4-(1,7-dimethyl-1H-indole-2-carbonyl)-N,N-dimethylpiperazine-1-sulfonamide
2-[(3R,4S)-3-amino-4-(propan-2-yl)pyrrolidin-1-yl]-N-cyclopropylacetamide
4-[(2-methyl-1,3-thiazol-4-yl)methyl]-1,3λ6,4-oxathiazinane-3,3-dione
(3S,4R)-1-[(2-aminopyridin-3-yl)methyl]-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
(4aS,7aR)-1-(pyridazine-3-carbonyl)-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{4-[(oxolan-3-yl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
6-[1-(4-chloro-1-methyl-1H-indole-2-carbonyl)piperidin-3-yl]pyrimidin-4-ol
5-(3-methoxyphenyl)-N-[3-(methylsulfanyl)propyl]-1,2,4-triazin-3-amine
4-(6-methoxypyridin-2-yl)-1H-indole
ethyl 3,5-dimethyl-4-{4-[3-oxo-3-(pyrrolidin-1-yl)propyl]piperidine-1-carbonyl}-1H-pyrrole-2-carboxylate
1-{2-[4-(2-ethoxyphenyl)piperazin-1-yl]pyrimidin-4-yl}pyrrolidin-3-ol