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methyl 2-({[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)acetate
1-cyclohexyl-3-[(1-ethylpyrrolidin-3-yl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
4-hydroxy-N-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}-2-(4-methylphenyl)pyrimidine-5-carboxamide
methyl N-{2-[(4aS,8aR)-2-oxo-1-(2-phenylethyl)-decahydro-1,6-naphthyridin-6-yl]-2-oxoethyl}carbamate
(cyclopropylmethyl)({[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl})(oxolan-2-ylmethyl)amine
3-[3-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]-1-[(5-methylpyrazin-2-yl)methyl]urea
2-methoxy-N-({5-[(4-methyl-1H-imidazol-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
N-[2-(dimethylamino)ethyl]-2-(pyridin-4-yl)-N-(thiophen-3-ylmethyl)acetamide
6-({[1-(2-hydroxyethyl)piperidin-4-yl]methyl}amino)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
N-(1,5-dimethyl-1H-pyrazol-4-yl)-2-[2-(2-methylpropyl)-3-oxo-2,8-diazaspiro[4.5]decan-8-yl]acetamide
1-ethyl-5-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-(2-methoxyethyl)-N-[(2-methoxyphenyl)methyl]-3,5-dimethyl-1H-indole-2-carboxamide
9-{3-[(dimethylamino)methyl]benzoyl}-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N3-(pentan-3-yl)-N3-(2-phenylethyl)piperidine-1,3-dicarboxamide
3-{[5-(1-cycloheptyl-1H-imidazol-2-yl)furan-2-yl]sulfanyl}-4-methyl-4H-1,2,4-triazole
N-[4-(oxolan-2-yl)butyl]-4-pentanamidobenzamide
2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]-4-[1-(propan-2-yl)piperidine-4-carbonyl]morpholine
1-(cyclopropylmethyl)-6-(1-methylpiperidin-4-yl)-3-(2-methylquinolin-5-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
2-{3-[4-(pyridin-4-yl)piperidine-1-carbonyl]piperidin-1-yl}pyridine
N,2-dimethyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]oxane-2-carboxamide
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
(2S,4R)-N-ethyl-1-(furan-2-ylmethyl)-4-[2-(pyridin-3-yl)acetamido]pyrrolidine-2-carboxamide
3-(1H-pyrazol-1-yl)-N-[2-(4-sulfamoylphenyl)ethyl]benzamide
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
4-[(2-ethylpyrimidin-4-yl)methyl]-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
4-[5-(1H-pyrazol-3-yl)furan-2-carbonyl]morpholine
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
N-methyl-5-({1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}methyl)-1,2,4-oxadiazole-3-carboxamide
N,1,3,5-tetramethyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1H-pyrazole-4-carboxamide
4-{4-[5-(azepan-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-4-oxobutanamide
N-methyl-2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
2,3-dimethyl-6-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}quinoxaline
3-[(3R,4S)-4-(dimethylamino)-1-[(8-fluoroquinolin-2-yl)methyl]piperidin-3-yl]propanoic acid
(5S,9aS,9bS)-5-[(E)-2-(2-methoxyphenyl)ethenyl]-2-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-amino-4-ethyl-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)-1,3-thiazole-5-carboxamide
1-methyl-3-(2-phenylethyl)-8-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{1-[(4-tert-butyl-1,3-thiazol-2-yl)methyl]-1H-1,2,3-triazol-4-yl}piperidine
N-{1-[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}-N-methylfuran-2-carboxamide
1-[6-(methoxymethyl)pyridine-2-carbonyl]-4-(thiophen-2-ylmethyl)piperazine
6-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carbonyl]-5-methyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
1-[(2,2-diphenylcyclopropyl)methyl]-4,4-difluoropiperidine
N-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-(1-{2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetyl}piperidin-4-yl)-1,4-diazepan-5-one
5-{1-[5-(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1H-1,2,3,4-tetrazole
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-[(5-methylthiophen-2-yl)sulfonyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
(3S,4R)-3-methoxy-1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperidin-4-amine
7-(cyclohexylmethyl)-2-(5-methyl-1,3-oxazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
(3R)-1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]pyrrolidin-3-ol
6-({methyl[(2-methylpyridin-4-yl)methyl]amino}methyl)pyrazolo[1,5-a]pyrimidine-3-carboxylic acid
N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-2-(2,3,6-trimethylphenoxy)acetamide