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4-[(2,3-dimethoxyphenyl)methyl]-1λ6-thiomorpholine-1,1-dione
(4aS,8aR)-1-(2-aminoethyl)-6-(2-methoxy-4-methylbenzoyl)-decahydro-1,6-naphthyridin-2-one
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2,2-dimethylpropanamide
N-[3-(4-fluorophenyl)phenyl]-1-(5-methyl-1,2-oxazole-3-carbonyl)piperidine-3-carboxamide
1-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidin-1-yl]-2-[methyl(phenyl)amino]ethan-1-one
2-{2-[2-(pyrrolidin-1-yl)ethyl]piperidine-1-carbonyl}thiophen-3-amine
N-[3-(1H-imidazol-1-yl)propyl]-3-(pyrrolidine-1-sulfonyl)-5-[(thiophen-3-ylmethyl)amino]benzamide
9-({5-[(4-methylphenyl)sulfanyl]furan-2-yl}methyl)-1,4,9-triazaspiro[5.5]undecan-5-one
3-{[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl}-N-[(1-methyl-1H-imidazol-2-yl)methyl]benzamide
5-(2-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-oxoethyl)pyrrolidin-2-one
{1-[5-(3-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]azepan-2-yl}methanol
1-[3-(furan-2-yl)propanoyl]-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
N-(5-acetyl-2-methoxyphenyl)-4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carboxamide
methyl 2-(cyclopentylsulfamoyl)-6-[(3,4,5-trifluorophenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
9-(5-ethyl-1,2,4-oxadiazol-3-yl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-cyclopropyl-1-{2-[1-(3,4-dimethoxybenzoyl)piperidin-2-yl]ethyl}-1H-1,2,3-triazole-4-carboxamide
1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-4-[3-(trifluoromethyl)phenoxy]piperidine
1-(3-chloro-2-methylphenyl)-3-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}urea
1-{[4-(diethylamino)phenyl]methyl}-5-oxopyrrolidine-3-carboxylic acid
3-methyl-N-[1-(3-methylpyridin-2-yl)propan-2-yl]-5-propyl-1-benzofuran-2-carboxamide
2-[1-(cyclopropylmethyl)-4-(2,2-dimethylpropyl)piperazin-2-yl]ethan-1-ol
3-[1-(1,2,4-oxadiazol-3-ylmethyl)piperidin-3-yl]-N-[4-(trifluoromethyl)phenyl]propanamide
2-(5-{1-[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-4-yl}-1H-pyrazol-3-yl)acetic acid
5-(1-cyclohexanecarbonylpiperidin-4-yl)-5-(pyridin-3-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
N-[(1-cyclopentylpiperidin-4-yl)methyl]-3-(1-methyl-1H-pyrazol-5-yl)-N-(oxolan-2-ylmethyl)propanamide
7-chloro-3-{[3-(3-hydroxypropyl)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
2-(1-methyl-1H-1,3-benzodiazol-2-yl)benzoic acid
2-[5-(1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-2-yl)-1,2,4-oxadiazol-3-yl]pyridine
N-(4-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-3-methylphenyl)acetamide
1-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-1-yl]-2-(dimethyl-1,3-thiazol-5-yl)ethan-1-one
1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
N-{[5,8-dimethoxy-2-(2-methoxyphenyl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)furan-2-carboxamide
3-[5-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl]pyridine
N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-3-(4H-1,2,4-triazol-4-yl)benzamide
6-chloro-5-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-sulfonyl}imidazo[2,1-b][1,3]thiazole
5-acetyl-N-({3-methyl-7-[3-(piperidin-1-yl)propanoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-3-carboxamide
[4-(2-phenylethyl)-1-(pyridin-4-ylmethyl)piperidin-4-yl]methanol
4-{4-[3-(methoxymethyl)piperidine-1-carbonyl]phenoxy}-1-(2-phenylethyl)piperidine
(3R,4R)-1-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]-4-(morpholin-4-yl)piperidin-3-ol
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(2-amino-4,6-dimethylpyrimidin-5-yl)acetamide
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-methyl-N-(2-phenylethyl)-1H-pyrazole-3-carboxamide
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-3-(1H-pyrazol-4-yl)benzamide
4-methyl-2-(1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidin-4-yl)-1H-1,3-benzodiazole
1-{5-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-2-methylphenyl}imidazolidin-2-one
1-(azepan-1-yl)-3-[3-({[2-(pyrazin-2-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
(2S,4S)-4-amino-N-ethyl-1-[2-(pyrrolidin-1-yl)-6-(trifluoromethyl)pyrimidin-4-yl]pyrrolidine-2-carboxamide
N-tert-butyl-1-[(3-methoxyphenyl)methyl]-6-oxopiperidine-3-carboxamide
methyl 3-(2-methoxyacetamido)-5-[(1-methoxypropan-2-yl)amino]-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-(furan-2-yl)-1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-3-phenylpropan-1-one
N-(1H-1,3-benzodiazol-2-ylmethyl)-5-(2-chloro-4-methoxyphenoxymethyl)-N-methyl-1,2-oxazole-3-carboxamide