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methyl 2-[butyl(methyl)sulfamoyl]-6-[(2-fluoro-4-methoxyphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-{4-[(3-fluorophenyl)methyl]-1-[(4-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-6-(2-methylpropyl)-2-oxo-1,2-dihydropyrimidine-4-carboxamide
[1-(2-{[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethyl)piperidin-2-yl]methanol
3-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-1-{3-[(trifluoromethyl)sulfanyl]phenyl}urea
(3S,5R)-1-(2-phenylacetyl)-5-[(pyridin-2-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
(1R,5S,6R)-3-(1H-1,3-benzodiazole-2-carbonyl)-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
3-(1-methyl-1H-pyrrol-2-yl)-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-1H-pyrazole-5-carboxamide
7-methyl-N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-[1,2,4]triazolo[4,3-a]pyrimidine-3-carboxamide
5-[(4-benzylpiperidin-1-yl)methyl]-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-1,2-oxazole-3-carboxamide
1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-5-phenylpentan-1-one
6-(1-{8-thiatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}piperidin-4-yl)-3,4-dihydropyrimidin-4-one
7-methoxy-3-{[4-(4-methylpyridin-2-yl)piperazin-1-yl]methyl}-1,2-dihydroquinolin-2-one
N-[(3R,4R)-3-hydroxy-1-{[2-(2-hydroxyethoxy)phenyl]methyl}piperidin-4-yl]pyridine-4-carboxamide
(3R,5S)-N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
N-[2-(benzylsulfanyl)ethyl]-3-ethyl-5-methyl-1,2-oxazole-4-carboxamide
{4-ethyl-1-[5-(2-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]piperidin-4-yl}methanol
1-{2-[3-(4-methoxyphenoxymethyl)piperidin-1-yl]-2-oxoethyl}piperidin-2-one
2-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-{4-[1-(1H-imidazol-2-ylmethyl)-4-phenyl-1H-imidazol-5-yl]phenyl}acetamide
3-butanamido-N-ethyl-4-methyl-N-(pyridin-4-ylmethyl)benzamide
(1R,4S)-N-cyclopropyl-N-[(2-methoxyphenyl)methyl]-1,7,7-trimethyl-3-oxo-2-oxabicyclo[2.2.1]heptane-4-carboxamide
1-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-2-(2-methoxyethoxy)ethan-1-one
5-[3-(pyrrolidine-1-carbonyl)pyridin-2-yl]-1H-indole
2-methoxy-3-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrazine
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-[(4-hydroxy-3-methoxyphenyl)methyl]-5-methylpiperidin-2-one
3-{2-[4-benzyl-2-(hydroxymethyl)piperazin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
2-methyl-5-{4-[(3-methylphenyl)sulfanyl]piperidine-1-carbonyl}pyrazine
1-[4-(2-fluorophenyl)piperazin-1-yl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
(1S,2S)-2-[4-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)piperazin-1-yl]cyclohexan-1-ol
4-{1-[(4-methoxyphenyl)methyl]-1H-imidazol-2-yl}-2-(propan-2-yl)pyrimidine
N-(oxolan-2-ylmethyl)-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-4-carboxamide
3-methyl-N-{[4-(methylsulfanyl)phenyl]methyl}-N-propyl-1H-pyrazole-5-carboxamide
1-[4-(dimethylamino)azepan-1-yl]-2-[3-(trifluoromethyl)phenoxy]ethan-1-one
N-{[4-({[3-(trifluoromethyl)phenyl]methyl}amino)quinazolin-2-yl]methyl}ethane-1-sulfonamide
2-methyl-3-(3-{1-[(3-methylpyridin-4-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyrazine
(2S,4R)-1-[(2-chlorophenyl)methyl]-4-{[(4-fluorophenyl)methyl]amino}-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-6-[(dimethylamino)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
[(2S,6S)-11-methoxy-4-(1,3-thiazol-2-yl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
1-[(4aR,8aS)-1-[3-(thiophen-2-yl)propanoyl]-decahydro-1,6-naphthyridin-6-yl]-3-phenoxypropan-1-one
1-[2-(dimethylamino)ethyl]-4-[3-(3-ethylphenoxy)azetidine-1-carbonyl]pyrrolidin-2-one
2-{[methyl({[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}phenol
1-(4-{6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl}phenyl)imidazolidine-2,4-dione
4-(1-methyl-1H-imidazole-5-carbonyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(2H-1,3-benzodioxol-5-ylmethyl)-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
N,6-dimethyl-N-[1-(1,3-thiazol-2-yl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylpent-4-enamide
4-(propan-2-yl)-3-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-2-one
N-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)propyl]-1-(propan-2-yl)piperidine-3-carboxamide
4-[3-(1H-imidazol-2-yl)-2,5-dimethyl-1H-pyrrol-1-yl]-4H-1,2,4-triazole