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(4aR,7aS)-1-cyclobutanecarbonyl-4-(pyridine-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(4-chlorophenyl)methyl]-N-[(4-hydroxy-1-methylpiperidin-4-yl)methyl]-6-oxopiperidine-3-carboxamide
N-[(5-methyl-1H-imidazol-4-yl)methyl]-1-[6-methyl-2-(piperidin-1-yl)pyrimidin-4-yl]piperidin-4-amine
4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-N,5-dimethyl-N-[2-(pyridin-2-yl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
3-(dimethyl-1H-1,2,4-triazol-3-yl)-1-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}urea
(4aS,8aR)-6-[(3-ethoxyphenyl)methyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
N-(3,4-dimethylphenyl)-1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-amine
1-(3,4-dichlorophenyl)-4-(2-methyl-1,3-thiazole-4-carbonyl)piperazine
6-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridin-3-amine
2-{1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-4-yl}-5-methyl-1H-1,3-benzodiazole
1-(oxolane-2-carbonyl)-4-(2-propyl-1,3-thiazole-4-carbonyl)piperazine
4-({[(1S)-1-carbamoyl-2-methylpropyl]carbamoyl}amino)-N-(2-methoxyethyl)-3-methylbenzamide
N-[3-(4-fluorophenyl)-3-(furan-2-yl)propyl]-3-{5-[(3-methylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
3-({1-[(5-ethylfuran-2-yl)methyl]piperidin-4-yl}oxy)-N-(2-methoxyethyl)benzamide
(3R,4R)-3-methyl-4-(oxan-4-yl)-1-[4-(1H-pyrazol-3-yl)benzoyl]piperidin-4-ol
4-(2-fluoro-5-methoxyphenyl)-2-methyl-1H-imidazole
N-(5-{[3-(4-methyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}thiophen-2-yl)acetamide
(2S)-3-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propane-1,2-diol
N-(3-methoxypropyl)-4-(3-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-amine
1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine
2-(cyclopropylmethyl)-8-[1-(2-hydroxyethyl)piperidine-4-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
3-[(4aR,7aS)-4-[2-(tert-butylcarbamoyl)ethyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
2-(2H-1,3-benzodioxol-4-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)-1H-1,3-benzodiazole
N,6-dimethyl-2-[2-(propan-2-yloxy)phenyl]pyrimidin-4-amine
3-[1-(4-methylpyridine-3-carbonyl)piperidin-3-yl]benzoic acid
3-{1-[(1-cycloheptanecarbonylpiperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}pyridine
7-(2-methoxyphenyl)-2-(1-methyl-1H-pyrazol-4-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
(2S,4S)-4-amino-1-(4-ethyl-5-methylthiophene-3-carbonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-{[(3-{3-[cyclohexyl(methyl)amino]-2-hydroxypropoxy}phenyl)methyl]amino}propane-1,3-diol
2-(5-chloropyridin-2-yl)-7-(3-methoxypropyl)-2,7-diazaspiro[4.5]decan-6-one
5-acetyl-3-{2-[2-(4-hydroxyphenyl)ethyl]piperidine-1-carbonyl}-6-methyl-1,2-dihydropyridin-2-one
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
4-[(2-fluorophenyl)methyl]-1-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
4-[3-(2-ethylphenoxy)azetidin-1-yl]-N,N-dimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-amine
6-methoxy-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
3-(2-{1-cyclohexyl-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-5-yl}ethyl)pyridine
1-{2-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
{[2-(butan-2-ylsulfanyl)pyrimidin-5-yl]methyl}({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl})methylamine
1-[2-(3-methoxyphenyl)ethyl]-2-(propan-2-yl)-1H-imidazole
7-({methyl[1-(1,2-oxazol-3-yl)ethyl]amino}methyl)-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
2-{4-methyl-1-[3-(4H-1,2,4-triazol-4-yl)phenyl]-1H-1,3-benzodiazol-2-yl}ethan-1-ol
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-methylpropanamide
1-{7-methyl-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline-4-carbonyl}piperidine-4-carbonitrile
N-{2-[(2S)-2-amino-3-(1,3-thiazol-4-yl)propanamido]-4-methylphenyl}pentanamide
(4aS,7aR)-1-(3-hydroxypyridine-2-carbonyl)-4-[(5-methylfuran-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(3-methyl-1,2,4-thiadiazol-5-yl)-1-{[3-(1H-1,2,4-triazol-1-yl)phenyl]methyl}urea
(2S,4S)-4-amino-1-(3-chloro-4-fluoro-1-benzothiophene-2-carbonyl)-N-ethylpyrrolidine-2-carboxamide
2-(4-{[3-(dimethylamino)pyrrolidin-1-yl]methyl}phenyl)-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
4-{2-methyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1-(pyridin-3-ylmethyl)pyrrolidin-2-one