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N-(furan-2-ylmethyl)-2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-(2-methylpropyl)acetamide
(oxolan-2-ylmethyl)({[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl})(thiophen-3-ylmethyl)amine
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[4-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]propan-1-one
4-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-2,6-dimethylpyrimidine
2-phenyl-1-{1-[2-(1H-pyrazol-1-yl)benzoyl]piperidin-3-yl}ethan-1-one
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-2-(1H-imidazol-2-yl)benzamide
3-fluoro-2-methoxy-N-[1-(pyridin-2-yl)propyl]benzamide
3-(2-methylphenyl)-5-[(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)methyl]-1,2,4-oxadiazole
1-{3-[ethyl(methyl)amino]propyl}-4-(6-hydroxypyrimidin-4-yl)-1,4-diazepan-6-ol
6-fluoro-4-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1,2,3,4-tetrahydroquinolin-2-one
2-methyl-N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
2-[2-fluoro-6-(propan-2-yloxy)phenyl]-N-methylpyrimidin-4-amine
(3R,4R)-4-(azepan-1-yl)-1-[(6-chloro-2H-chromen-3-yl)methyl]piperidin-3-ol
(4aS,8aR)-1-(3-aminopropyl)-6-[2-(1-methyl-1H-pyrrol-3-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
1-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-2-(piperidin-1-yl)ethan-1-one
3-[2-(2-oxopyrrolidin-1-yl)ethyl]-5-(2-phenylethyl)-5-(piperidin-4-yl)imidazolidine-2,4-dione
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzamide
4-{[3-(2-methylpiperidin-1-yl)azetidin-1-yl]methyl}quinoline
6-{[ethyl(oxan-4-yl)amino]methyl}naphthalen-2-ol
N-(furan-2-ylmethyl)-2,5-dimethyl-N-(pyridin-2-ylmethyl)-1,3-thiazole-4-carboxamide
1-[(4-methoxyphenyl)methyl]-4-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]piperazin-2-one
N-[(1-benzylpiperidin-3-yl)methyl]thian-4-amine
ethyl 2-{4-[3-(piperidine-1-carbonyl)pyridin-2-yl]piperazin-1-yl}acetate
3-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-1-(thiophen-2-yl)urea
3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methoxyethyl)-8-[3-(5-methylfuran-2-yl)butyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
1-[4-(2-methylphenyl)-3-oxopiperazin-1-yl]-4-phenylbutane-1,4-dione
1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-2-(phenylsulfanyl)ethan-1-one
4,6-dihydroxy-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}pyridine-3-carboxamide
3-[2-fluoro-4-(pyrrolidin-1-ylmethyl)phenoxy]-6-methylpyridazine
2-[4-(2,6-dimethylphenyl)phenoxy]-N-methylacetamide
2-(4-methoxyphenyl)-1-[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-6-oxopiperazine-2-carboxamide
3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazine-1-carbonyl]-1λ6-thiolane-1,1-dione
1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-(4-{[(3R,4S)-3-amino-4-phenylpyrrolidin-1-yl]sulfonyl}phenyl)-3-methylurea
(2R,3S,6R)-5-[(3,5-dimethoxyphenyl)methyl]-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
2-{8-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl}acetamide
2-(5-methyl-1,2-oxazol-3-yl)-N-(1-oxo-2,3-dihydro-1H-inden-5-yl)piperidine-1-carboxamide
N-[2-(pyridin-4-yl)ethyl]-4-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
7-(oxan-4-yl)-2-[2-(phenylsulfanyl)ethyl]-2,7-diazaspiro[4.5]decan-6-one
N-cyclopropyl-5-(1H-indole-2-carbonyl)-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-{6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
2-{5-[(1,1-dioxo-1λ6-thiomorpholin-4-yl)methyl]-2-methoxyphenoxy}acetic acid
[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl][(2E)-3-(furan-2-yl)prop-2-en-1-yl]methylamine
4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-[(4-methoxyphenyl)methyl]piperidine
1-[4-(3,4-dichlorophenyl)piperazin-1-yl]-4-(1H-imidazol-1-yl)butan-1-one
3-{4-[(4-fluorophenyl)methyl]-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl}-N-methylpropanamide
1-(2,3-dimethoxyphenyl)-2-(furan-3-ylmethyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-4-(1H-1,2,4-triazol-3-yl)benzamide