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N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-ethyl-5-methylthiophene-3-carboxamide
1,3-dimethyl-2,6-dioxo-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-1,2,3,6-tetrahydropyrimidine-4-carboxamide
4-{[4-(pyrazin-2-yl)piperazin-1-yl]methyl}-2,1,3-benzoxadiazole
7-[(2S)-2-methoxy-2-phenylacetyl]-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(4aR,7aS)-1-acetyl-4-{[3-(2-methylpropoxy)phenyl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-methyl-2-[5-(trifluoromethyl)pyridin-2-yl]-2,7-diazaspiro[4.5]decan-6-one
N-(2,1,3-benzothiadiazol-5-ylmethyl)-5-ethylpyrazolo[1,5-a]pyrimidin-7-amine
1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-4,4-difluoropiperidine
2-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
4-({5-[3-(4-fluorophenyl)-1H-pyrazol-4-yl]-1H,4H-pyrazolo[3,4-d]imidazol-1-yl}methyl)pyridine
4-(pyridin-3-ylmethyl)-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-1-methylpiperidine-3-carboxamide
3-[5-(3,4-dihydro-2H-1-benzopyran-2-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
N-[(1r,4r)-4-hydroxycyclohexyl]-6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
[(5-{1-[(2-chlorophenyl)methyl]piperidin-3-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1H-imidazol-2-ylmethyl)piperidine
3-{[(2-amino-6-ethyl-5-methylpyrimidin-4-yl)amino]methyl}-1,2,4-oxadiazole-5-carboxamide
N-(2-methoxyethyl)-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-3-carboxamide
3-(hydroxymethyl)-1-{2-[2-(3-methoxyphenyl)ethyl]benzoyl}piperidin-3-ol
N-cyclohexyl-N-(pyridin-4-ylmethyl)-4-(4H-1,2,4-triazol-4-yl)benzamide
N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-2-(2-phenylethyl)-1,3-benzoxazole-5-carboxamide
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-(3-methoxypyrazin-2-yl)piperidine-4-carboxylic acid
ethyl 3-{[2-(2-chloro-6-fluorobenzamido)-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazol-5-yl]formamido}propanoate
1-{3-[4-(1H-pyrazol-1-ylmethyl)piperidin-1-yl]propyl}-1H-1,3-benzodiazole
3-({[(4-chlorophenyl)(phenyl)methyl]amino}methyl)-7-methoxy-1-(prop-2-yn-1-yl)-1,2-dihydroquinolin-2-one
N-[(1R,3R)-3-aminocyclopentyl]-4-phenyl-1H-imidazole-5-carboxamide
3-methoxy-N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-4-[(1-methylpiperidin-4-yl)oxy]benzamide
N-(1-hydroxy-2-methylpropan-2-yl)-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
N2-(2-methoxyethyl)-N4-[1-(1-methyl-1H-pyrazol-4-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
2-methyl-3-[3-(pyridin-4-yl)propanamido]-N-(1,3-thiazol-2-yl)benzamide
methyl (2S)-1-(3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}propanoyl)pyrrolidine-2-carboxylate
N-(3-ethoxy-2-hydroxypropyl)-4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(4-propyl-1,2,3-thiadiazole-5-carbonyl)piperidine
4-({[(2-amino-1,3-thiazol-4-yl)methyl]amino}methyl)-2,6-dimethylphenyl acetate
2-(3-methoxyphenyl)-1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidine
3-(1H-indol-3-yl)-N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]propanamide
1-[(4aR,8aS)-6-(1-benzothiophen-2-ylmethyl)-decahydro-1,6-naphthyridin-1-yl]-2,2-dimethylpropan-1-one
1-[(5-ethylpyridin-2-yl)methyl]-4-(4-methoxyphenyl)-2-methylpiperazine
4-({3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}methyl)-2,1,3-benzoxadiazole
N-(butan-2-yl)-5-methyl-N-(pyridin-3-ylmethyl)pyridine-3-carboxamide
2-{4-[1-(oxane-4-carbonyl)pyrrolidin-3-yl]piperidin-1-yl}pyrimidine
ethyl 4-[(4-{[1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]piperazine-1-carboxylate
1-[3-(1H-pyrazol-1-yl)propyl]-N-[4-(1,3-thiazol-4-yl)phenyl]pyrrolidine-2-carboxamide
2-[3-(5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]pyridine-4-carbonitrile
ethyl 1-[2-(2-methoxyphenoxy)acetyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine
1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-4-(1H-imidazol-2-yl)piperidine
4-benzyl-3-ethyl-1-[2-(2H-1,2,3,4-tetrazol-2-yl)acetyl]-1,4-diazepan-5-one
2-amino-4-(3-ethyl-1H-pyrazol-5-yl)-6-(4-hydroxyphenyl)-5-methylpyridine-3-carbonitrile