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N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N,2-dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
ethyl({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl){[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}amine
4-({methyl[1-(1,2-oxazol-3-yl)ethyl]amino}methyl)-1H-pyrazole-3-carboxylic acid
2-(2H-1,3-benzodioxol-5-yl)-N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
2-(2H-1,3-benzodioxol-5-yl)-1-[(3R,4R)-4-cyclopropyl-4-hydroxy-3-methylpiperidin-1-yl]ethan-1-one
4-(propan-2-yl)-1-{5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carbonyl}piperidine
3-cyclopentyl-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]propanamide
3-(2-methoxyphenyl)-N-{2-[2-(1-methyl-1H-pyrrol-3-yl)acetyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}propanamide
8-chloro-2-[3-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]quinoline
methyl 6-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-2-[(2-methylpropyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-(1-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-N-(furan-2-ylmethyl)piperidine-4-carboxamide
2-methoxy-5-{[(2-methoxyethyl)[(3-methylthiophen-2-yl)methyl]amino]methyl}phenol
2-({3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}methyl)benzonitrile
3-[3-(aminomethyl)phenyl]-1-(oxan-4-yl)urea
N-[(3S,4R)-4-(propan-2-yl)-1-(thiophene-3-sulfonyl)pyrrolidin-3-yl]acetamide
2-[1-(2-methylpropyl)-4-[(3-methylquinoxalin-2-yl)methyl]piperazin-2-yl]ethan-1-ol
(2S)-2-({5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-4-methylpentan-1-ol
2-chloro-4-(5,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)benzamide
3-(1-benzothiophen-7-yl)-6-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-1-(cyclopropylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2-[4-(2-methylquinolin-4-yl)-2-(morpholin-4-ylmethyl)phenoxy]acetamide
N-[2-(1H-indol-3-yl)ethyl]-6-(methoxymethyl)pyrimidin-4-amine
propyl 1-methyl-4-[3-(methylsulfanyl)butyl]-1,4,9-triazaspiro[5.5]undecane-9-carboxylate
1-(1H-imidazole-5-carbonyl)-4-{[4-(4-methylphenyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
3-{[1-cyclohexyl-3-(cyclopropylmethyl)-1H-1,2,4-triazol-5-yl]methyl}pyridine
2-{1-[(5-methylfuran-2-yl)methyl]piperidin-2-yl}pyridine
7-[4-(1H-pyrazol-3-yl)benzoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(3S,4S)-4-methyl-1-[4-(trifluoromethyl)pyridin-2-yl]piperidine-3,4-diol
1-[(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-methoxypropan-1-one
3-{2-[3-(hydroxymethyl)-3-(2-phenylethyl)piperidin-1-yl]-2-oxoethyl}-1,3-thiazolidine-2,4-dione
3-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-[4-(methylsulfanyl)phenyl]urea
N-methyl-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-[(2-fluorophenyl)methyl]-N-[(6-methyl-2H-1,3-benzodioxol-5-yl)methyl]piperidin-3-amine
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-3-(methylsulfanyl)propanamide
2-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine-1-carbonyl}pyridin-3-ol
5-{2-[(3aR,5R,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-2-oxoethyl}-2-ethyl-6-methyl-3,4-dihydropyrimidin-4-one
2-chloro-N-(2-{[1-(2-fluorophenyl)cyclopropyl]formamido}ethyl)benzamide
(3R,4S)-1-(3-chloropyridin-2-yl)-4-cyclopropyl-N,N-dimethylpyrrolidin-3-amine
7-[(2,3-difluorophenyl)methyl]-6-oxo-N-propyl-2,7-diazaspiro[4.5]decane-2-carboxamide
(3R,9aR)-8-(cyclopropylmethyl)-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
7-(5-phenylpentanoyl)-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4-(4-chlorophenoxy)-1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperidine
1-{2-[5-(1H-imidazol-4-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-4-methylpiperazine
N3-benzyl-N5-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-1-cyclopropyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]benzonitrile
N,1-diethyl-N-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-1H-pyrazole-3-carboxamide
4-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
(2-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridin-4-yl)methanol
1-[(2-phenylethyl)carbamoyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
1-[(4-ethoxyphenyl)methyl]-4-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperazine