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3-{5-[(2,2,3,3-tetrafluoropropoxy)methyl]-1,2,4-oxadiazol-3-yl}pyridazine
[(4-methoxy-2,5-dimethylphenyl)methyl](methyl){2-[4-(4-methylpiperazine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}amine
6-methyl-2-(5-methyl-1H-indol-3-yl)pyridine-3-carboxamide
N-({5-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methoxyacetamide
N-[4-(3-methoxyphenyl)phenyl]-1-[2-(1H-1,2,4-triazol-1-yl)acetyl]piperidine-3-carboxamide
5-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]isoquinoline
(4aS,8aR)-1-(2-aminoethyl)-6-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-decahydro-1,6-naphthyridin-2-one
1-[8-methyl-3-(pyrrolidin-1-ylmethyl)imidazo[1,2-a]pyridine-2-carbonyl]piperidine
N-[(2-methoxyphenyl)methyl]-2-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}acetamide
(3R,4R)-4-ethyl-1-[2-(1,1,2,2-tetrafluoroethoxy)benzoyl]piperidine-3,4-diol
2-[3-(oxan-4-yl)-5-[2-(1H-pyrazol-4-yl)ethyl]-1H-1,2,4-triazol-1-yl]acetic acid
8-{2-[(cyclopropylmethyl)sulfanyl]acetyl}-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[(2-chlorophenyl)methyl]-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-methyl-N-[2-methyl-1-(pyridin-3-yl)propyl]-6-(propan-2-yl)pyrimidin-4-amine
{3-[({[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)methyl]-2,4,6-trimethylphenyl}methanol
1-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]-3-(1-propyl-1H-1,2,3-triazol-4-yl)urea
5-methyl-1-propyl-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-1H-pyrazole-4-carboxamide
5-{4-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]phenyl}-2-methyl-2H-1,2,3,4-tetrazole
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-4-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperazin-2-yl}ethan-1-ol
[(5-{[(3-fluorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl](methyl)[(5-methylfuran-2-yl)methyl]amine
6-(2,5-dimethylfuran-3-yl)-N-(5-hydroxypentyl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
8-(cyclopropanesulfonyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-(3-chloro-4-hydroxyphenyl)-N-methyl-N-(quinoxalin-2-ylmethyl)acetamide
(3S,4S)-4-cyclopropyl-1-(2,3-difluoro-6-methoxybenzoyl)pyrrolidine-3-carboxylic acid
5-amino-4-chloro-N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]-1H-pyrazole-3-carboxamide
[(1-{[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]dimethylamine
1'-(4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
1-(4-{[3-(morpholin-4-yl)azetidin-1-yl]methyl}phenoxy)-3-(piperidin-1-yl)propan-2-ol
N-cyclohexyl-2-(2,6-dioxo-1,3-diazinan-1-yl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
2-cyclopentyl-N-cyclopropyl-N-({3-[(1-methylpiperidin-3-yl)methoxy]phenyl}methyl)acetamide
4-amino-1-[2-(4-chlorophenyl)morpholin-4-yl]butan-1-one
(1S,5R)-6-[2-methyl-2-(morpholin-4-yl)propyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-cyclopropyl-9-(3,4,5-trifluorobenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[1-methyl-4-(propan-2-yloxy)-1H-indazol-3-yl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
[(2S,6S)-4-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
2-[5-(4-methoxypyrimidin-2-yl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
(3S,4R)-1-(2-methoxy-5-methylbenzoyl)-4-(3-methylthiophen-2-yl)piperidin-3-ol
1-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidine
3-(5-methylthiophen-2-yl)-5-(morpholine-4-sulfonyl)-N-(propan-2-yl)benzamide
1-(furan-2-ylmethyl)-N-[1-(5,6,7,8-tetrahydronaphthalen-2-yl)ethyl]piperidine-4-carboxamide
N-(2-hydroxyethyl)-3-(5-methylfuran-2-yl)-N-(thiophen-2-ylmethyl)benzamide
N-methyl-5-{[(6-methylpyridin-3-yl)oxy]methyl}-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,2-oxazole-3-carboxamide
N-(oxolan-2-ylmethyl)-3-[1-(1-phenylpiperidin-4-yl)piperidin-4-yl]propanamide
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-1H-pyrazole-3-carboxamide
2-[3-benzyl-1-(2-methoxyphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(1-hydroxypropan-2-yl)acetamide
1-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]-4-(4-methylphenoxy)piperidine
3-[9-oxo-8-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-2-yl]-N-(propan-2-yl)propanamide
(1S,5R)-3-(4-amino-6,7-dimethoxyquinazolin-2-yl)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one