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methyl 4-[(6-methoxy-4-oxo-3,4-dihydroquinazolin-3-yl)methyl]benzoate
4-methoxy-N-(2-methoxyethyl)-2-{[1-(oxolan-3-ylmethyl)piperidin-4-yl]oxy}benzamide
N-[(2S)-oxolan-2-ylmethyl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
1-(5-chloro-6-oxo-1,6-dihydropyridine-3-carbonyl)-2-methylpiperidine-2-carboxylic acid
1-(2-methoxyethyl)-4-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazine
3-(azocan-1-yl)-N-[2-(3-hydroxy-4-methoxyphenyl)ethyl]propanamide
1-methyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-1H-indole-2-carboxamide
1-tert-butyl-3-(4-ethoxyphenoxymethyl)-5-(oxan-3-ylmethyl)-1H-1,2,4-triazole
2-(2,4-dimethoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-{1-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]piperidin-4-yl}-3-methylbutan-1-ol
5-chloro-2-{3-oxa-9-azaspiro[5.5]undecane-9-carbonyl}phenol
4-{[3-(2-oxopyrrolidin-1-yl)piperidin-1-yl]sulfonyl}benzonitrile
methyl 5-{[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}-3-(2-methoxyacetamido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-cyclopropyl-2-{4-[1-(morpholin-4-yl)ethyl]phenyl}pyridine-4-carboxamide
4-{4-[4-(azepan-1-yl)piperidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
2-[(4-ethyl-3,3-dimethylpiperazin-1-yl)methyl]-3,5-dimethoxybenzoic acid
[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl](methyl){[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
2-(2-aminoethyl)-N-{[3-methyl-4-(pyrrolidin-1-yl)phenyl]methyl}quinazolin-4-amine
3-{[ethyl(oxan-4-yl)amino]methyl}-6,7-dimethoxy-1,2-dihydroquinolin-2-one
1-(3,5-dichloro-4-methylbenzoyl)-N-[2-(dimethylamino)ethyl]-N-methylpiperidin-3-amine
2-(3-aminopropanoyl)-N-methyl-N-(1,3-thiazol-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
2-methoxyethyl 4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
(4aR,7aS)-1-(2-methoxyacetyl)-4-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-(1H-indol-1-ylmethyl)-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1H-pyrazole-3-carboxamide
1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-4-(pyridin-3-yl)piperidin-4-ol
3-{1-[(3,5-dimethoxyphenyl)methyl]piperidin-3-yl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-amino-6-(4-hydroxyphenyl)-4-[2-(propan-2-yl)pyrimidin-5-yl]pyridine-3-carbonitrile
2-(cyclopropylmethyl)-9-[4-(1H-imidazol-1-yl)butanoyl]-2,9-diazaspiro[5.5]undecan-3-one
3-(3-hydroxy-3-methylbutyl)-N-[1-(methoxymethyl)cyclopentyl]benzamide
2-(3-methyl-1,2-oxazol-5-yl)-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]ethan-1-one
[(3R,4S)-4-[(4-ethylpiperazin-1-yl)methyl]-1-[(4-methoxy-2,3-dimethylphenyl)methyl]pyrrolidin-3-yl]methanol
1-{imidazo[1,2-a]pyridine-6-carbonyl}-4-(pyridin-4-ylmethyl)-1,4-diazepane
2-(3-hydroxypiperidin-1-yl)-1-[4-(4-methoxybenzoyl)piperazin-1-yl]ethan-1-one
2-amino-N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-methylpropanamide
benzyl (7S,9aR)-7-[(4-methoxyphenyl)methyl]-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
4-{1-[1-(3-phenylbutyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carbonyl}morpholine
1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}pyrrolidin-3-ol
1-(carbamoylmethyl)-N-[3-(4-chlorophenyl)propyl]piperidine-4-carboxamide
4-{[3-(methanesulfonylmethyl)piperidin-1-yl]methyl}quinoline
(4aR,8aR)-4a-hydroxy-N,N-dimethyl-7-[(6-methyl-2H-1,3-benzodioxol-5-yl)methyl]-decahydro-2,7-naphthyridine-2-carboxamide
N-[(1-cyclohexylpiperidin-3-yl)methyl]-2-(diethylamino)-N-(pyridin-3-ylmethyl)acetamide
5-(4-{4-cyclopropyl-5-[(dimethylamino)methyl]-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)-1,2-dihydropyridin-2-one
3-oxo-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
8-(4-ethyl-5-methylthiophene-3-carbonyl)-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(3S,4R)-1-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
4-[3-(2-chlorophenyl)-1H-pyrazol-5-yl]-1-(5-methyl-1,2-oxazole-3-carbonyl)piperidine
3-[(2R,3R,6R)-5-(5-methylthiophene-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
N-[3-(azepan-1-yl)-2-hydroxypropyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
7-(3-chlorophenyl)-4-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-9-(furan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(5-{[methyl({[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl})amino]methyl}furan-2-yl)benzonitrile