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N-[(2-ethoxy-3-methoxyphenyl)methyl]-1,2,3,4-tetrahydronaphthalen-2-amine
4-(dimethylamino)-N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]benzamide
3-{1-[(4-methyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(cyclopropylmethyl)-5-methyl-N-propyl-4-[(pyridin-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
1-(3-{6-[(2-methoxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)ethan-1-ol
1-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-amine
N-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-3-methylfuran-2-carboxamide
2-{[4-(quinolin-3-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}ethan-1-ol
2-(dimethyl-1,3-thiazol-5-yl)-N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}acetamide
4-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidine-1-carbonyl]benzonitrile
N-[(3R,4S)-1-cyclobutanecarbonyl-4-cyclopropylpyrrolidin-3-yl]-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)-2-(1H-pyrazol-1-yl)acetamide
3-{[6-hydroxy-4-(pyridin-4-yl)-1,4-diazepan-1-yl]methyl}benzonitrile
3-{1-[2-(2,3-dimethoxyphenyl)-1H-imidazol-1-yl]-2,2,2-trifluoroethyl}pyridine
1-[(2,3-difluoro-4-methylphenyl)methyl]-2-(oxolan-3-yl)-1H-imidazole
1-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-3-(2-methoxyphenoxy)azetidine
1-(2H-1,3-benzodioxol-5-ylmethyl)-5-(1-methoxyethyl)-3-(oxan-4-yl)-1H-1,2,4-triazole
(2R,3R,6R)-3-phenyl-5-[2-(pyrrolidin-1-yl)benzoyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
(2S,4S)-N-ethyl-1-(2-hydroxyethyl)-4-[2-(naphthalen-1-yl)acetamido]pyrrolidine-2-carboxamide
6-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-1,3-benzothiazole
5-ethyl-N-[3-(1H-imidazol-1-yl)propyl]-2-methylpyrimidin-4-amine
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N-methyl-3-[(2-methylprop-2-en-1-yl)oxy]benzamide
5-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-1-methyl-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(2-fluoro-4-methoxyphenyl)-5-methyl-4-(1H-pyrazol-1-ylmethyl)-1,3-oxazole
N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-2-(1H-pyrazol-1-yl)butanamide
1-(2-methylpropyl)-4-(pyrrolidin-3-yl)piperidine
2-(1-ethylpiperidin-4-yl)-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]acetamide
3-cyclohexyl-N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
2-[4-(5-ethyl-2-methylpyrimidin-4-yl)piperazin-1-yl]-N-phenylacetamide
[5-({3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}methyl)furan-2-yl]methanol
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-[3-(1H-pyrazol-1-yl)propyl]piperazin-2-yl}ethan-1-ol
3-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]phenol
4-(2-methyl-4-phenylpyrimidine-5-carbonyl)-4-azatricyclo[4.3.1.13,8]undecane
N3-[2-(3,5-dimethoxyphenyl)ethyl]piperidine-1,3-dicarboxamide
3-(1,2-dihydroacenaphthylene-5-carbonyl)-N,N-dimethylpiperidine-1-sulfonamide
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-(thiophen-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(3-{[1-(1,3-thiazole-4-carbonyl)piperidin-4-yl]oxy}benzoyl)morpholine
2-amino-4-(3,4-dihydroxyphenyl)-6-[4-fluoro-2-(trifluoromethyl)phenyl]pyridine-3-carbonitrile
(1S,5R)-N-(3-methylphenyl)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
(3S,9aR)-3-[(benzyloxy)methyl]-8-(quinolin-8-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-methyl-2-phenyl-N-(pyrazin-2-ylmethyl)benzamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-{[5,8-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}propanamide
4-{[6-(3-tert-butyl-5-methylphenyl)pyridin-3-yl]methyl}morpholine
(4aR,7aS)-1-(2-methylpropyl)-4-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[4-(4-fluorophenyl)-2-[(4-methylpiperazin-1-yl)methyl]phenoxy]-N-{[4-(trifluoromethyl)phenyl]methyl}acetamide
3-{3-[5-(ethanesulfonyl)thiophen-2-yl]phenyl}-1H-pyrazole
2-{4-[2-(pyridin-2-yl)pyrrolidin-1-yl]quinazolin-2-yl}ethan-1-amine
5-methyl-1-(2-oxo-2-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione