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2-{1-[(4-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-(1H-imidazol-2-ylmethyl)acetamide
1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
3-[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-1-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)urea
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-(2,2-difluoroethyl)acetamide
1-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-[2-(thiophen-2-yl)ethyl]piperidine
(3R,5S)-5-[(2,3-dihydro-1H-inden-5-yloxy)methyl]-N-[3-(morpholin-4-yl)propyl]-1-(pyridin-4-ylmethyl)piperidine-3-carboxamide
2-(4-{[4-(difluoromethoxy)phenyl]methyl}morpholin-3-yl)acetic acid
(1S,5R)-6-benzyl-3-(6-methylpyridazin-3-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[(2-methylpyridin-4-yl)methyl]piperidin-2-one
9-hydroxy-4-oxo-N-{2-[(trifluoromethyl)sulfanyl]ethyl}-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
1-[4-(dimethylamino)-5-methylpyrimidin-2-yl]piperidin-4-ol
2-(1-ethyl-1H-pyrazol-4-yl)-6,8-dimethyl-4-(2-methylpiperidine-1-carbonyl)quinoline
N-[3-(4-{[4-(2-chlorophenyl)piperazin-1-yl]methyl}phenoxy)propyl]pyridine-4-carboxamide
2-[2-({[(4-fluorophenyl)methyl](oxolan-2-ylmethyl)amino}methyl)phenoxy]acetamide
N-[2-(dimethylamino)-2-(5-methylfuran-2-yl)ethyl]-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
1-methyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-1H-pyrazole-4-carboxamide
1-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]-3-(methoxymethyl)piperidine
2-(ethanesulfonyl)-N-[2-(2-methylphenyl)-1,3-benzoxazol-6-yl]acetamide
9-(4-hydroxybenzoyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
4-oxo-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-4H-chromene-2-carboxamide
N-{[4-(3-methoxyphenyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}-5-methylthiophene-2-carboxamide
6-(2-aminoethyl)-2-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-3,4-dihydropyrimidin-4-one
N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
2-(4-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl)ethan-1-ol
1-ethyl-4-[(4-hydroxy-1,2,3,4-tetrahydroisoquinolin-2-yl)methyl]-1H-pyrrole-2-carbonitrile
4-(2,2-diphenylethyl)-3-[2-oxo-2-(pyrrolidin-1-yl)ethyl]piperazin-2-one
(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-3-ol
2-methyl-6-[2-(2-methylphenyl)-2-(4-methylpiperidin-1-yl)ethyl]-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
5-[2-(piperidin-1-yl)acetyl]-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
(3R,4R)-4-cyclopropyl-1-[(5-ethylfuran-2-yl)methyl]-3-methylpiperidin-4-ol
N-(3-chloro-2-fluorophenyl)-4-[(1-methylpiperidin-3-yl)methyl]piperazine-1-carboxamide
(1-methyl-1H-imidazol-2-yl)({1-[4-(pyridin-2-yl)pyrimidin-2-yl]piperidin-4-yl})methanol
(4aS,8aR)-1-(4-hydroxybutyl)-6-(1H-indol-2-ylmethyl)-decahydro-1,6-naphthyridin-2-one
(3S,4R)-1-(4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
N-[(3-methoxyphenyl)methyl]-N-[(4-methyl-1H-imidazol-5-yl)methyl]cyclopropanamine
3-[(1-methyl-1H-imidazol-2-yl)methyl]-1-[4-(oxan-2-ylmethoxy)phenyl]-3-(propan-2-yl)urea
1-(4-{[(furan-2-ylmethyl)(3-methylbutan-2-yl)amino]methyl}thiophen-2-yl)ethan-1-one
1-(2-methoxyethyl)-8-{[3-(2-methylphenyl)phenyl]methyl}-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
8-[(5-chlorothiophen-2-yl)sulfonyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}-2-(pyrrolidin-1-yl)acetamide
1-{[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}-4-(pyridin-4-yl)piperazine
N-methyl-4-{6-methyl-5-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine-2-carbonyl}pyridin-2-amine
4-{methyl[2-(methylcarbamoyl)ethyl]sulfamoyl}-N-(oxolan-3-yl)benzamide
2-[4-(propan-2-yloxy)phenyl]-2-(thiomorpholin-4-yl)acetic acid
N-(1H-1,3-benzodiazol-2-yl)-2-[4-hydroxy-4-(pyridin-2-yl)piperidin-1-yl]acetamide
3-[1-(6-methoxypyridin-2-yl)-3,5-dimethyl-1H-pyrazol-4-yl]propanoic acid
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-2-(pyrazin-2-yl)ethan-1-one
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-N,4-dimethyl-2-(piperidin-1-yl)pyrimidine-5-carboxamide
N,2-dimethyl-N-[(3-methylpyridin-4-yl)methyl]-1H-1,3-benzodiazole-4-carboxamide