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2-{4-[(4-chlorophenyl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
1,5-dimethyl-N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)-1H-pyrazole-3-carboxamide
4-cyclopentyl-N-(dimethyl-1H-1,2,4-triazol-3-yl)-3-oxopiperazine-1-carboxamide
6-(cyclopropylmethoxy)-1-[(3-methoxyphenyl)methyl]-4-(pyrazine-2-carbonyl)-1,4-diazepan-2-one
N-[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]-3-(furan-2-yl)propanamide
ethyl({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})[(1-methylpyrrolidin-3-yl)methyl]amine
N-({3,5-dimethoxy-4-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-2,6-difluoro-N-[(3S)-2-oxoazepan-3-yl]benzene-1-sulfonamide
3-{1-[3-(acetamidomethyl)phenyl]-1H-imidazol-2-yl}benzoic acid
1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-4-(3-methylpyridin-2-yl)piperazine
5-[4-(pyridin-2-ylmethyl)-1,4-diazepane-1-carbonyl]-1,2-oxazol-3-ol
5-cyclopropanecarbonyl-1'-[(2-fluoro-5-methoxyphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-[4-(1H-imidazol-2-yl)piperidin-1-yl]-6-methyl-2-(methylsulfanyl)pyrimidine
5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-(2-methoxyethyl)-N-methylpyridin-2-amine
N-({4-hydroxy-1-[(1-phenyl-1H-pyrazol-5-yl)methyl]azepan-4-yl}methyl)methanesulfonamide
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-methyl-N-[2-(piperidin-1-yl)ethyl]-1H-pyrazole-3-carboxamide
3-{[2-chloro-5-(1H-pyrazol-1-yl)phenyl]formamido}-N-cyclohexylpropanamide
N-[1-(4-cyclopentyl-4H-1,2,4-triazol-3-yl)ethyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
methyl 2-(5-{1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidin-4-yl}-1H-pyrazol-3-yl)acetate
1-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}-3-(1,2-oxazinan-2-yl)propan-1-one
1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-4-{[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
3-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-5-fluoropyridine
5-[(3aR,6aS)-5-methyl-octahydropyrrolo[3,4-c]pyrrole-2-carbonyl]-1-(2-ethoxyethyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-(2-ethoxy-1-hydroxyethyl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[3-(2-chlorophenoxy)propyl]-N-methyl-2-[(1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonan-3-yl]acetamide
(1R,5S,6R,7S)-3-methyl-6-{3-[(1-propylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
N-cyclopentyl-N'-[(8-methoxyquinolin-5-yl)methyl]-N'-methylbutanediamide
3-({[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]amino}methyl)pyrrolidin-3-ol
3-(2,1,3-benzothiadiazol-5-ylmethyl)-3H,4H-pyrido[3,4-d]pyrimidin-4-one
N-[2-(2-fluorophenyl)-1-{1-[(4-methoxyphenyl)methyl]piperidin-4-yl}ethyl]-N,2-dimethylfuran-3-carboxamide
1-(3-benzoylpiperidin-1-yl)-2-(3-methoxyphenoxy)ethan-1-one
2-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}-1,2,3,4-tetrahydroisoquinolin-4-ol
1-[(2,5-dimethoxyphenyl)methyl]-4-[2-(thiomorpholine-4-carbonyl)-1-benzofuran-5-yl]piperidin-4-ol
6-chloro-2-{1-[5-(2,6-dimethoxyphenyl)-1,2,4-triazin-3-yl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
N-[2-(4-methoxyphenyl)phenyl]-1-(pentan-3-yl)piperidine-3-carboxamide
N-{1-[1-(3-phenylpropyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-methyl-2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}acetamide
1-[3-(methylsulfanyl)propyl]-3-[3-(trifluoromethyl)benzoyl]piperidine
N-(1,3-benzoxazol-2-ylmethyl)-N-methyl-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
2-{3-[1-(oxan-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}-1,3-thiazole
2-{2-[3-(2-chlorophenoxy)azetidin-1-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
methyl 8-[(1,3-diphenyl-1H-pyrazol-4-yl)methyl]-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
N-({3-methyl-7-[2-(methylsulfanyl)benzoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-2-carboxamide
[3-(2-methoxyethyl)-1-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]piperidin-3-yl]methanol
(3R,4R)-4-ethyl-1-(5-ethyl-2,6-dimethylpyrimidin-4-yl)piperidine-3,4-diol
N-[2-(2-fluorophenyl)-1-{1-[2-(1-methyl-1H-pyrrol-3-yl)acetyl]piperidin-4-yl}ethyl]-N-methyl-3-(methylsulfanyl)propanamide
N-[2-(pyrrolidine-1-sulfonyl)ethyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl)[(4-methylphenyl)methyl]amine
N-{[2-(3-chlorophenyl)-7-methylquinolin-3-yl]methyl}-N-(3-methoxypropyl)-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
N-(2,6-dimethoxypyridin-3-yl)-2-(pyridin-3-yl)piperidine-1-carboxamide
N-[(4-fluorophenyl)methyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide