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[4-(1-butyl-3-ethyl-1H-1,2,4-triazol-5-yl)phenyl]methanol
8-(morpholine-4-sulfonyl)-2-(oxolane-3-carbonyl)-1,2,3,4-tetrahydroisoquinoline
1-[3,5-dimethyl-4-(3-{[4-(propan-2-yl)phenyl]amino}piperidine-1-carbonyl)-1H-pyrrol-2-yl]ethan-1-one
(3S,4S)-1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
({4-cyclopropyl-5-[1-(2-fluorobenzoyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
(3aR,6aR)-2-methanesulfonyl-5-[(2-methylpyridin-3-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-benzyl-3-ethyl-1-(3-methyl-1H-pyrazole-5-carbonyl)-1,4-diazepan-5-one
(3R,4R)-1-[(2,3-difluoro-6-methoxyphenyl)methyl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
12-(1H-pyrazol-4-yl)-8-thia-5-azatricyclo[7.4.0.02,7]trideca-1(13),2(7),9,11-tetraen-6-one
3-(pentan-2-yl)-8-(quinoline-8-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-benzyl-3-[1-(2-methanesulfonylacetyl)piperidin-4-yl]-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-methyl-5-{4-[3-(5-methylfuran-2-yl)butyl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
N-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-5-(2-methoxyethyl)-1,3,4-thiadiazol-2-amine
3-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-1-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}urea
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]-1,3-thiazole-4-carboxamide
N-[(3R,4R)-3-hydroxy-1-[3-(4-hydroxyphenyl)propanoyl]piperidin-4-yl]pyridine-3-carboxamide
1-methyl-N-{2-[methyl(2-phenylethyl)amino]ethyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
(1S,5R)-6-[(2-ethoxyphenyl)methyl]-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
5-(hydroxymethyl)-2-methyl-4-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}pyridin-3-ol
[1-(5-cyclopropyl-1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-1H-pyrazole-4-carbonyl)piperidin-4-yl]methanol
2-methoxy-5-methyl-N-{[1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]methyl}benzamide
3-{[1-(6-oxo-1,6-dihydropyridine-3-carbonyl)piperidin-4-yl]methyl}benzoic acid
1-[2-(2-methoxyphenyl)ethyl]-N,2,6-trimethyl-4-oxo-N-(thiophen-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
3-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-3-methyl-1-[3-(1,3-oxazol-5-yl)phenyl]urea
(1S,5R)-6-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
(2S,4S)-4-{[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]amino}-1-{[4-(diethylamino)phenyl]methyl}-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
4-[(2,4-dimethoxy-3-methylphenyl)methyl]-1-(4-methoxyphenyl)piperazin-2-one
(4aS,8aR)-6-[2-(propylsulfanyl)acetyl]-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
{3-[(1-{[4-(difluoromethoxy)phenyl]methyl}pyrrolidin-3-yl)methyl]phenyl}methanol
[(2-methoxy-5-{[(1S,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}phenyl)methyl]dimethylamine
4-{[2-(benzylamino)pyrimidin-5-yl]methyl}piperazin-2-one
2-(1H-indol-3-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)-1H-1,3-benzodiazole
3-fluoro-N-[3-(1H-indol-1-yl)propyl]pyridine-4-carboxamide
N-cyclopentyl-4-[4-hydroxy-4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-4-oxobutanamide
2-(1,2,3,4-tetrahydroisoquinolin-2-yl)-2-(trimethyl-1H-pyrazol-4-yl)acetic acid
[(3R,5R)-1-(5-ethoxyfuran-2-carbonyl)-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
2-(2,6-dimethoxyphenyl)-N-ethylpyrimidin-4-amine
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-(3-fluoro-4-methoxyphenyl)-1,2,4-triazin-3-amine
N-[2-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)ethyl]acetamide
2,2-dimethyl-N-(1-{1-[2-(pyridin-3-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)propanamide
1-(3-{[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl}benzoyl)piperidine-4-carbonitrile
3-[4-(1,3-benzoxazol-2-yl)piperazine-1-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
4-{4-[({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}amino)methyl]phenyl}but-3-yn-1-ol
(2S)-2,6-diamino-N-ethyl-N-[(2E)-3-phenylprop-2-en-1-yl]hexanamide
5-methyl-1-[4-(4-{[3-(methylsulfanyl)propyl]amino}piperidin-1-yl)phenyl]pyrrolidin-2-one
2-cyclopropyl-8-(4-methylpyridin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
N,N-dimethyl-2-{methyl[2-(quinoxalin-2-yloxy)hex-5-en-1-yl]amino}acetamide
{[(3S,4R)-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
2-({6-[4-benzyl-3-(2-hydroxyethyl)piperazin-1-yl]pyrimidin-4-yl}amino)ethan-1-ol
1-ethyl-4-[2-(3-methoxypiperidine-1-carbonyl)-2,3-dihydro-1H-inden-2-yl]piperazine