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N-[2-(diethylamino)ethyl]-N,2-diethyl-6-methyl-1-[(5-methylfuran-2-yl)methyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-cyclopropyl-5-(1H-imidazol-2-ylmethyl)-1-[2-(4-methoxyphenyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(butane-1-sulfonyl)-4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine
2-[2-methyl-4-(4-methylphenyl)-5-oxopiperazin-1-yl]-N-[(2-methylphenyl)methyl]acetamide
1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-[(2-methoxyethyl)(methyl)amino]ethan-1-one
2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]-N-[2-(morpholin-4-yl)ethyl]acetamide
3-butyl-4-(3-chloro-4-hydroxybenzoyl)-1-methylpiperazin-2-one
1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)azocane
3-[(3S,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2-chlorophenyl)urea
N-(1-{1-[(4-phenylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)acetamide
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-4-carboxamide
N-(1-methyl-2-oxopyrrolidin-3-yl)-3-[(piperidin-4-yl)sulfamoyl]benzamide
dimethyl({4-[1-(1-methyl-1H-pyrazole-4-carbonyl)piperidin-2-yl]phenyl}methyl)amine
3-[3-({[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]amino}methyl)-1H-indol-1-yl]propanamide
{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)(pyridin-2-ylmethyl)amine
N-[(2S,4R,6S)-2-benzyl-6-(2,3-dihydro-1,4-benzodioxin-6-yl)oxan-4-yl]acetamide
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-4-methyl-1H-imidazole-5-carboxamide
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-{[(2-methylprop-2-en-1-yl)amino]methyl}piperidin-2-one
{[2-methyl-1-(2-methylpropyl)-1H-indol-3-yl]methyl}[(3-methyl-1H-pyrazol-5-yl)methyl]amine
3-[3-chloro-4-(1H-imidazol-1-yl)phenyl]-1-[2-(morpholin-4-yl)ethyl]urea
5-(3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamido)-1H-indole-3-carboxamide
2-(5-cyclopropyl-4-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-1H-pyrazol-1-yl)-4-(furan-2-yl)pyrimidine
5-(methoxymethyl)-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-N-{[1-(piperidin-1-yl)cyclopentyl]methyl}-1H-pyrazole-4-carboxamide
1-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]-3-[5-(4-methylphenyl)furan-2-yl]propan-1-one
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
3-({2-[1-(pyrrolidine-1-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
N-ethyl-N-[3-(morpholin-4-yl)propyl]-2-(pyrrolidin-3-yl)benzamide
5-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-4-methyl-2-(propan-2-yl)pyrimidine
5-({3-[3-oxo-3-(pyrrolidin-1-yl)propyl]piperidin-1-yl}sulfonyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-(2H-1,3-benzodioxol-5-yl)-N-[2-(2-oxopiperidin-1-yl)ethyl]-3-phenylpropanamide
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(1-methyl-1H-indol-3-yl)acetamide
3-(isoquinolin-5-yl)benzonitrile
1,3-dimethyl-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-1-(pyrrolidin-1-yl)propan-1-one
5-(propan-2-yl)-3-[2-(4H-1,2,4-triazol-4-yl)ethyl]-1,2,4-oxadiazole
2,3,5-trimethyl-N-[2-(pyridin-2-ylsulfanyl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-{3-[2-(3-methoxyphenyl)ethyl]piperidin-1-yl}pent-4-en-1-one
2-(ethoxymethyl)-N-[2-(propane-2-sulfonyl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-{[(2-methoxyethyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amino]methyl}-N-methylpyridin-2-amine
7-(propan-2-yl)-2-(3-propyl-1H-pyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
4-(5-ethylpyrimidin-2-yl)-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane
4-(2,4-dimethoxypyrimidin-5-yl)-2-phenylquinazoline
1-phenyl-4-(5-propyl-1,2-oxazole-3-carbonyl)piperazin-2-one
3-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl}-5-methoxybenzoic acid
4-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-3-propyl-1H-pyrazole
[(1,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl){[5-(methylsulfanyl)-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl}amine
3-butyl-1-methyl-4-[2-(methylsulfanyl)pyrimidine-5-carbonyl]piperazin-2-one
({5-[1-(cyclohexylmethyl)piperidin-4-yl]-4-cyclopropyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
N-{[2-(2,3-difluoro-4-methylphenoxy)pyridin-3-yl]methyl}-2-(1,4-dimethylpiperazin-2-yl)acetamide