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2-(1-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperidin-3-yl)-4-methyl-1H-1,3-benzodiazole
1-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
4-[4-({4-[(3,3-dimethylpyrrolidin-1-yl)methyl]-1H-1,2,3-triazol-1-yl}methyl)piperidine-1-carbonyl]pyrrolidin-2-one
5-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonane-7-carbonyl]-2,3-dimethylbenzene-1-sulfonamide
4-{1-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]piperidin-3-yl}benzoic acid
N-{[5-methyl-2-(trifluoromethyl)furan-3-yl]methyl}-5-phenyl-1,2-oxazole-3-carboxamide
3-(1-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-1H-1,2,3-triazol-4-yl)piperidine
5-methyl-N-[2-methyl-2-(morpholin-4-yl)propyl]-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
5-[1-(2,3-dihydro-1H-inden-2-yl)-1H-pyrazol-3-yl]-N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-methyl-1,3-thiazol-2-amine
4-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-ylmethyl]-N-(1-ethyl-5-methyl-1H-pyrazol-3-yl)benzamide
1-(4-fluorophenyl)-4-{3-[5-(hydroxymethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}butane-1,4-dione
4-cyclopentyl-11-{[(1-hydroxycyclohexyl)methyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
[1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)pyrrolidin-3-yl]methanamine
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[2-(1H-imidazol-1-yl)phenyl]methyl}benzamide
2-cyclopropyl-5-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-3,4-dihydropyrimidin-4-one
2-cyclopentyl-1-[9-methoxy-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
1-(2,3-difluoro-6-methoxybenzoyl)-2-(4-fluorophenyl)piperidine
N-(3,5-dimethoxyphenyl)-3-{1-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]piperidin-3-yl}propanamide
4-{[(4aS,8aR)-1-[3-(methylsulfanyl)propyl]-2-oxo-decahydro-1,6-naphthyridin-6-yl]methyl}-1,5-dimethyl-1H-pyrrole-2-carbonitrile
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
3-[6-(4-methylpiperazin-1-yl)pyridazin-3-yl]-5-[2-(piperidin-2-yl)ethyl]phenol
N-(2-fluorophenyl)-3-(1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidin-3-yl)propanamide
3,3-dimethyl-1-[(3S,4R)-4-(propan-2-yl)-1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}pyrrolidin-3-yl]urea
1-(4-methylphenyl)-4-[3-(morpholin-4-yl)benzoyl]piperazin-2-one
3-{[ethyl(propyl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
4-{2-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)formamido]ethyl}benzoic acid
1-[7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]-3-(2-ethyl-1H-imidazol-1-yl)propan-1-one
N-cyclohexyl-3-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
2-{[4-(pyrrolidin-3-yl)piperazin-1-yl]methyl}benzoic acid
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-(1-phenylcyclopropyl)piperidine-4-carboxamide
6-methyl-2-[1-(1-methyl-1H-indole-4-carbonyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
ethyl 2-(1-{2-[methyl(phenyl)amino]acetyl}piperidin-2-yl)acetate
3-{1-[3-(3-hydroxy-3-methylbutyl)benzoyl]pyrrolidin-2-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(4-methoxyphenyl)methyl]-5,6-dimethyl-2-oxo-N-(oxolan-2-ylmethyl)-1,2-dihydropyridine-3-carboxamide
3-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1-[2-(propan-2-ylsulfanyl)phenyl]urea
3-[1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]-N-(4-methoxy-2-methylphenyl)propanamide
N,N,5,7-tetramethyl-2-[1-(2,2,2-trifluoroethyl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
(2S,4R)-4-amino-N-ethyl-1-[2-(methylamino)pyridine-3-carbonyl]pyrrolidine-2-carboxamide
3-(3-fluorophenyl)-1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]propan-1-one
2-{[3-(2,4-dimethoxybenzoyl)piperidin-1-yl]methyl}-1-methyl-1H-1,3-benzodiazole
(5R)-5-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}pyrrolidin-2-one
1-[4-(4-hydroxypiperidin-1-yl)pyrimidin-2-yl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
5-chloro-N-[1-(3,5-difluorophenyl)ethyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
8-(1,3-benzothiazol-2-ylmethyl)-3-[3-(dimethylamino)propyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-[4-(2-methoxyphenoxy)piperidine-1-carbonyl]quinoxaline
9-[(2S)-2-(dimethylamino)-3-phenylpropanoyl]-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
(2R,6R)-4-(1H-pyrazole-3-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-{6-[(propan-2-yl)amino]pyrimidin-4-yl}piperidin-3-yl]propanoic acid
1-(2-chlorophenyl)-4-{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
(3R)-1-({1-[(1-{thieno[3,2-d]pyrimidin-4-yl}piperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}methyl)pyrrolidin-3-ol