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2-cyclopropyl-4-hydroxy-N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)pyrimidine-5-carboxamide
N,2-dimethyl-N-[(4-phenoxyphenyl)methyl]-1,3-thiazole-5-carboxamide
N-methyl-2-(2-phenyl-1H-imidazol-1-yl)-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}acetamide
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(2-phenylethyl)acetamide
1-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}-2-(methylamino)ethan-1-one
5-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidine-1-carbonyl}-2-methyl-1,3-benzothiazole
1-ethyl-5-(2,4,5-trimethoxyphenyl)-1H,4H-pyrazolo[3,4-d]imidazole
5-{3-[4-(2-chlorophenyl)-3-oxopiperazin-1-yl]-3-oxopropyl}imidazolidine-2,4-dione
{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl){[5-(methylsulfanyl)-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl}amine
7-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-2-methyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N-[2-(azepan-1-yl)ethyl]-2,6-dihydroxy-N-methylbenzamide
7-[3-(1H-1,2,3-benzotriazol-1-yl)propanoyl]-2-(dimethylamino)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4,5,6-trimethyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[2-ethyl-1-(pyridin-3-ylmethyl)-7-(2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-1H-1,3-benzodiazol-5-yl]acetamide
3-{[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]sulfamoyl}-N-(2,2,2-trifluoroethyl)benzamide
2-methyl-6-[1-(1-methyl-1H-indole-3-carbonyl)piperidin-3-yl]pyrimidin-4-ol
7-fluoro-4-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]-1,2-dihydroquinolin-2-one
2-[5-(2H-1,2,3-benzotriazol-2-ylmethyl)-3-methyl-1H-1,2,4-triazol-1-yl]ethan-1-ol
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-2-(1H-1,2,4-triazol-3-yl)benzamide
N4-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-5,6-dimethylpyrimidine-2,4-diamine
1,3-dimethyl-6-(pyridin-3-yl)-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
[(4-methoxyphenyl)methyl][(2-phenoxypyridin-3-yl)methyl]amine
4-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridin-6-yl]-6-(propan-2-yl)pyrimidine
methyl (2S,4R)-4-{2-[2-(dimethylamino)pyrimidin-5-yl]-1H-imidazol-1-yl}-1-methylpyrrolidine-2-carboxylate
8-[(2R)-2-aminopropanoyl]-3-(2-ethylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-(3-hydroxyazetidine-1-carbonyl)-2-(3-methylphenyl)pyrimidin-4-ol
8-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-{4-[4-(4-acetyl-1,4-diazepan-1-yl)piperidin-1-yl]phenyl}-3-phenylpropanamide
(2S,4R)-4-amino-N-(propan-2-yl)-1-(2,3,4,9-tetrahydro-1H-carbazole-8-carbonyl)pyrrolidine-2-carboxamide
ethyl 1-benzoyl-3-[(4-fluorophenyl)methyl]piperidine-3-carboxylate
(3R,4R)-1-(furan-2-ylmethyl)-4-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-3-ol
3-cyclopentyl-1-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
N-[3-(furan-2-yl)phenyl]-1-(thiophen-3-ylmethyl)piperidine-4-carboxamide
N-[3-(oxolan-3-yl)propyl]quinoxaline-6-carboxamide
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)cyclobutanamine
2-[3-(4-chlorophenyl)-5-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}-1H-1,2,4-triazol-1-yl]ethan-1-ol
[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl](methyl){4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}amine
3-{[2-(1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidin-3-yl)-1H-imidazol-1-yl]methyl}pyridine
6-(3,5-dimethyl-1H-pyrazol-4-yl)-1,2,3,4-tetrahydroquinazoline-2,4-dione
2-amino-7-hydroxy-4-[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-5H-indeno[1,2-b]pyridine-3-carbonitrile
N-methyl-1-(4-methyl-1H-pyrrole-2-carbonyl)-N-[2-(pyridin-2-yl)ethyl]piperidin-3-amine
N-{2-[(4aS,8aR)-1-(3-methylbutyl)-2-oxo-decahydro-1,6-naphthyridin-6-yl]-2-oxoethyl}methanesulfonamide
6-methyl-2-({4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}methyl)quinolin-4-ol
(1R,5R)-6-[2-(4-fluorophenoxy)ethyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
N-(1-cyclopentyl-4-methyl-1H-pyrazol-5-yl)-2-(2-methyl-1H-1,3-benzodiazol-1-yl)acetamide
2-(2,4-dichlorophenoxy)-N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]acetamide
N-(1-phenylcyclopropyl)-3-(2-phenylpropyl)-1,2-oxazole-5-carboxamide
5-{2-[5-(3-fluoro-4-methylphenyl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1H-1,2,3,4-tetrazole
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(2-hydroxyphenoxy)acetamide
3-methoxy-N-{2-[2-(phenylsulfanyl)acetyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}propanamide