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3-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-3,9-diazaspiro[5.6]dodecan-10-one
(3S,4R)-1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-methyl-3-(2-methylpropyl)piperidin-4-ol
2-(2H-1,2,3-benzotriazol-2-yl)-1-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
2-(1H-indol-3-yl)-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]acetamide
N-{2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}-1-oxo-1,2-dihydroisoquinoline-4-carboxamide
1-{[(2R,5S)-5-(1-benzothiophen-3-ylmethyl)oxolan-2-yl]methyl}piperidine-4-carboxylic acid
[3-(2-methoxyethyl)-1-(oxan-4-yl)piperidin-3-yl]methanol
3-{4-[1-(2-phenylethyl)pyrrolidin-3-yl]piperidine-1-carbonyl}pyridin-2-ol
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-{1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}propanamide
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-(4-hydroxypiperidin-1-yl)pyridine-3-carboxamide
2-(cyclopropylmethyl)-9-(6-methyl-2-propylpyrimidin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(2R,3R)-1'-(2H-1,3-benzodioxol-4-ylmethyl)-2-(benzyloxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
3-[({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)carbamoyl]pyridin-1-ium-1-olate
8-(4-methylpyridine-3-carbonyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-4,4,4-trifluorobutanamide
4-[(2,2-difluoroethyl)sulfamoyl]-N-[2-(2-hydroxyethoxy)ethyl]benzamide
3-{[(1S)-1-carbamoyl-2-hydroxyethyl]sulfamoyl}-N-(2-fluorophenyl)benzamide
5-(2,6-dimethylphenoxymethyl)-N-[(4-hydroxy-1-methylpiperidin-4-yl)methyl]-1,2-oxazole-3-carboxamide
4-[(2-ethyl-2-methyl-3-oxopiperazin-1-yl)methyl]-1H-pyrazole-3-carboxylic acid
3-(3-chloro-2,6-dimethylphenyl)-1-(oxan-4-yl)urea
8-{[4-(furan-2-yl)phenyl]methyl}-1-(2-methoxyethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]propan-1-one
1-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
2-(3,4-dimethoxyphenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
(2R,3R)-1'-(4-methyl-1H-imidazole-2-carbonyl)-3-(pyrrolidin-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-[(3R,4S)-3-(3-hydroxypropyl)-4-(morpholin-4-yl)piperidin-1-yl]-2-(3-methylphenoxy)ethan-1-one
3-(1-{3-chloro-6-methylpyrazolo[1,5-a]pyrimidine-2-carbonyl}piperidin-4-yl)phenol
1-[2-(4-chlorophenyl)morpholin-4-yl]-2-(morpholin-4-yl)ethan-1-one
3-butyl-4-(3-{imidazo[1,2-a]pyridin-2-yl}propanoyl)-1-methylpiperazin-2-one
1-[(2,6-difluorophenyl)methyl]-4-(1-ethyl-1H-imidazol-2-yl)piperidine
1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-4-(thian-4-yl)piperazine
1-cyclohexyl-4-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
3-{[methyl(quinoxalin-6-ylmethyl)amino]methyl}pyrrolidin-3-ol
(1S,3R)-N-(5-fluoro-2-methylphenyl)-3-[(morpholine-4-sulfonyl)amino]cyclopentane-1-carboxamide
2-chloro-N-(1-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
1-[1-(4,6-dimethylpyrimidin-2-yl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
1-[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidin-1-yl]-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propan-1-one
3-(1,2-oxazinan-2-yl)-1-{2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidin-1-yl}propan-1-one
3-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidine-1-carbonyl}-4H-pyrido[1,2-a]pyrimidin-4-one
5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-[2-(pyridin-3-yl)ethyl]-1,2-oxazole-3-carboxamide
3-[3-(ethoxycarbonyl)pyridin-2-yl]benzoic acid
(1R,5S)-6-{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}-6-azabicyclo[3.2.1]octane
(1S,5R)-3-[(2-ethoxyphenyl)methyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{[4-(2-methoxyphenoxy)piperidin-1-yl]methyl}benzonitrile
2-{3-[4-(1,3-thiazol-2-yl)-1H-1,2,3-triazol-1-yl]propyl}-1,3-benzothiazole
5-methoxy-2-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]-1H-indole
4-[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-methylpyrimidine
1-{[(3R,4R)-4-(hydroxymethyl)-1-(quinoline-3-carbonyl)pyrrolidin-3-yl]methyl}piperidin-4-ol
3-[2-(azocan-1-yl)-2-oxoethyl]-4-(naphthalen-1-ylmethyl)piperazin-2-one
N-(4-fluoro-3-methoxyphenyl)-4-(3-methoxypropyl)piperazine-1-carboxamide