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2,6-diamino-4-{3-methoxy-2-[(2-methylprop-2-en-1-yl)oxy]phenyl}-5,6,7,8-tetrahydroquinoline-3-carbonitrile
3-fluoro-4-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine
4-chloro-N-{1-[(3-chlorophenyl)methyl]-1H-pyrazol-5-yl}-1-methyl-1H-pyrazole-5-carboxamide
5-{3-[2-(2-phenyl-1,3-oxazol-4-yl)-1H-imidazol-1-yl]propyl}-1H-1,2,3,4-tetrazole
5-[4-hydroxy-1-(4-methylphenyl)-6-oxo-1,6-dihydropyridazine-3-carbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
5-(2-chlorophenyl)-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]furan-2-carboxamide
2-(2,5-dioxo-1-propylimidazolidin-4-yl)-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]acetamide
N-methyl-N-[2-(pyridin-2-yl)ethyl]-1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
1-(2-{5-[2-(methylsulfanyl)propyl]-4-phenyl-1H-imidazol-1-yl}ethyl)piperidine
1-[(4aR,8aR)-7-[(2-chloro-3,4-dimethoxyphenyl)methyl]-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]ethan-1-one
3-[2-(piperidin-2-yl)ethyl]-5-[3-(pyrrolidine-1-carbonyl)pyridin-2-yl]phenol
1-(5-ethyl-1,3-oxazole-4-carbonyl)-4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine
(1R,5S,8R)-3-(5,6-dimethylpyrimidin-4-yl)-N,N-dimethyl-3-azabicyclo[3.2.1]octan-8-amine
(1R,5R)-6-(1H-indazole-3-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
3-{1-[2-(phenoxymethyl)-1,3-oxazole-4-carbonyl]piperidin-2-yl}pyridine
1-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidin-4-amine
1-(2-methanesulfonylethyl)-5,5-diphenylpiperidin-2-one
N-ethyl-5-methyl-N-{[3-(prop-2-en-1-yloxy)phenyl]methyl}pyridine-3-carboxamide
(3S,4R)-1-(4-fluorobenzoyl)-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
N-benzyl-4-(3-methoxypropyl)piperazine-1-sulfonamide
4-({2-[1-(3-chloro-5-fluorobenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}(2-methoxyethyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-oxo-2-(propan-2-yl)-1,6-dihydropyrimidine-5-carboxamide
N-cyclopropyl-1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}piperidine-3-carboxamide
1-benzyl-8-[(2-butyl-1H-imidazol-4-yl)methyl]-3-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2-benzamido-5-methylphenyl)-5-[(dimethylamino)methyl]furan-2-carboxamide
9-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3,9-diazaspiro[5.6]dodecane
N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)acetamide
1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-(2-phenylindolizin-3-yl)ethane-1,2-dione
9-(6-chloroquinolin-4-yl)-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
8-[1-(hydroxymethyl)cyclopropanecarbonyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
4-{[1-benzyl-5-(4-methyl-1,3-thiazol-5-yl)-1H-1,2,4-triazol-3-yl]methyl}-1-methylpiperidine
(1S,6R)-9-[2-amino-6-(2-methylpropyl)pyrimidine-4-carbonyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
N-cyclohexyl-1-(2-ethoxyethyl)-N-methyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
4-(3-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}phenyl)-4H-1,2,4-triazole
5-{[(1R,5S,8S)-8-methoxy-3-azabicyclo[3.2.1]octan-3-yl]methyl}-N,N-dimethylpyridin-2-amine
1-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-2-(4-fluorophenyl)pyrrolidine
2-({8-cyclopropyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}sulfonyl)benzonitrile
(2R)-2-hydroxy-2-phenyl-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
1-(2-chloro-4-fluorophenyl)-3-[2-(ethylsulfanyl)ethyl]urea
[3-(3-methylbut-2-en-1-yl)-1-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}piperidin-3-yl]methanol
(2S,4S)-1-[(2-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-({[4-(methylsulfanyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
7-(3-methoxypropyl)-2-[4-(1H-pyrazol-4-yl)butanoyl]-2,7-diazaspiro[4.5]decan-6-one
4-[3-(3-fluorophenoxymethyl)-1-(1-methylpiperidin-4-yl)-1H-1,2,4-triazol-5-yl]pyridine
4-(4-methyl-1,3-thiazole-5-carbonyl)-1-[(4-methylphenyl)methyl]piperazin-2-one
({2,5-dimethyl-3-[(3-methylpiperidin-1-yl)methyl]phenyl}methyl)(methyl)[2-(2-methyl-1H-imidazol-1-yl)ethyl]amine
methyl({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)(1,2-oxazol-5-ylmethyl)amine
N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}quinolin-7-ol
4-benzyl-3-ethyl-1-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-1,4-diazepan-5-one