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3-{5-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-N-cyclopropylpropanamide
4-[3-cyclopropyl-1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]-1-methyl-1,2-dihydropyridin-2-one
2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]-N-[3-(1H-pyrazol-1-yl)propyl]acetamide
1-(3-chloro-4-ethoxyphenyl)-3-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]urea
N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
methyl 6-(2-methoxy-2-phenylacetyl)-2-[(prop-2-en-1-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(2S,4R)-4-amino-N-methyl-1-(5-phenyl-1,3,4-thiadiazol-2-yl)pyrrolidine-2-carboxamide
(2S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-N-methyl-4-[(naphthalen-2-ylmethyl)amino]pyrrolidine-2-carboxamide
N-methyl-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-1H-pyrazole-3-carboxamide
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}piperidine
8-fluoro-2-({4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}methyl)quinolin-4-ol
4-(2-ethoxyphenyl)-3-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl 4-[2-amino-3-cyano-6-(3-hydroxyphenyl)pyridin-4-yl]-1H-pyrazole-3-carboxylate
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[2-(4-hydroxypiperidin-1-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-4-methoxybenzamide
1-[1-(benzenesulfonyl)piperidin-3-yl]-4-(4-methoxyphenyl)piperazine
ethyl 2-[2-(morpholine-4-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]pyridine-3-carboxylate
1-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-3-ethylurea
1-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-4-methanesulfonylpiperazine
2-[1-(1-benzofuran-2-sulfonyl)pyrrolidin-2-yl]pyridine
2-(2,5-dimethylphenyl)-1-[(1R,5R)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
1,9-dimethyl-4-[2-(2H-1,2,3,4-tetrazol-2-yl)acetyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
4-(1H-pyrazol-4-yl)-1-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}butan-1-one
3-[(3R,4S)-4-(morpholin-4-yl)-1-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-3-yl]propanoic acid
N-(1,5-dimethyl-1H-pyrazol-4-yl)-2-methyl-4-[(4-methylphenyl)methyl]-3-oxopiperazine-1-carboxamide
{5-[3-(3-ethylphenoxy)azetidine-1-carbonyl]furan-2-yl}methanol
2-phenyl-7-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(3S,4S)-N-(4-ethenylphenyl)-3-hydroxy-4-(pyrrolidin-1-yl)pyrrolidine-1-carboxamide
1-(2-phenylethyl)-3-(4H-1,2,4-triazol-4-ylmethyl)piperidine
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-2-(pyridin-3-yl)acetamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[2-(2-oxopyrrolidin-1-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{[5-methyl-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclobutanecarboxamide
2-(1H-imidazol-2-yl)-N-methyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]benzamide
5-[1-(methoxymethyl)cyclopropanecarbonyl]-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-(2-phenoxyethyl)piperazine
8-[3-(benzyloxy)propyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-(2,3-dihydro-1H-inden-2-yl)-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
(1S,5R)-3-(pyridin-3-ylmethyl)-6-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
(2-{[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl][(3-methylthiophen-2-yl)methyl]amino}ethyl)dimethylamine
[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-(3-phenylpropyl)piperidin-4-yl]methanol
5-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]pyridin-2-amine
methyl (2S,4R)-1-(1,3-benzothiazole-6-carbonyl)-4-(dimethylamino)pyrrolidine-2-carboxylate
1-butyl-4-{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
methyl 2-{3-oxo-4-[3-(pyridin-3-yl)propyl]-3,4-dihydro-2H-1,4-benzoxazin-2-yl}acetate
1-{3-[4-({[2-(2-fluorophenyl)ethyl]amino}methyl)-2-methoxyphenoxy]-2-hydroxypropyl}piperidin-4-ol
N-[3-({[3-(4-chloro-1H-pyrazol-1-yl)propyl]carbamoyl}amino)-4-methoxyphenyl]acetamide
4-[(2-methylprop-2-en-1-yl)oxy]-N-(oxan-2-ylmethyl)benzamide
(3S,4S)-1-{[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}-4-(morpholin-4-yl)pyrrolidin-3-ol
1-ethyl-5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-(1-{1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-4-yl}-2-phenylethyl)-N-methylthiophene-3-carboxamide
2-[(1r,4r)-4-hydroxycyclohexyl]-9-(1,3-thiazol-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one