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2-[3-oxo-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-9-yl]-N-phenylacetamide
2-ethyl-9-(3-methyl-1,2-oxazole-5-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecane
1-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-3-(1-methyl-1H-imidazol-2-yl)piperidine
methyl 3-(oxolane-3-amido)-5-[(pentan-3-yl)amino]-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-{1-[2-(2-chloro-4-fluorophenyl)acetyl]piperidin-3-yl}-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
2-[3-(2-chlorophenyl)-1-(3-methoxypropyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-(quinoxalin-6-ylmethyl)acetamide
2-(4-{[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]methyl}-3-methyl-1H-pyrazol-1-yl)ethan-1-ol
methyl (2S)-2-{3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamido}-2-phenylacetate
4-methoxy-1-{[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl}piperidine
(3aR,6aR)-2-{[3-(2-hydroxyethoxy)phenyl]methyl}-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-fluoro-2-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine
1,5-dimethyl-4-({2-[2-(morpholin-4-yl)ethyl]piperidin-1-yl}methyl)-1H-pyrrole-2-carbonitrile
2-{[(3-tert-butyl-1H-pyrazol-5-yl)methyl](methyl)amino}-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-6-methoxy-1,3-benzothiazol-2-amine
(3S,4S)-1-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-4-(propan-2-yloxy)pyrrolidin-3-ol
1-ethyl-3-(pyrrolidine-1-carbonyl)-N-[2-(thiophen-2-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
methyl 2-(1-{[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl}-3-oxopiperazin-2-yl)acetate
9-(1-methylpyrrolidine-3-carbonyl)-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(2,2-dimethyl-4-phenyloxan-4-yl)ethyl]-3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propanamide
1-(3-{[(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-3-hydroxypiperidin-1-yl]methyl}phenyl)ethan-1-one
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-1-(2-methylpropyl)-N5-(2-phenylethyl)piperidine-3,5-dicarboxamide
1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-3-(pyrazin-2-yl)propan-1-one
N-(cyclopropylmethyl)-2-[(2R)-2-hydroxypropanoyl]-N-propyl-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
1-ethyl-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-5-oxopyrrolidine-3-carboxamide
N-{3-[ethyl(methyl)amino]butyl}-1-(2-methoxyphenyl)-1H-pyrazole-4-carboxamide
1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-2-methyl-4-(4-methylphenyl)piperazine
2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-N-[2-(5-methylfuran-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
ethyl 4-{[3-(2-{[(2-chlorophenyl)methyl]carbamoyl}ethyl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylate
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(thiophen-2-yl)ethan-1-one
5-{[3-(3-methylthiophene-2-carbonyl)piperidin-1-yl]methyl}isoquinoline
1-[3-(1-methyl-5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]butane-1,2-dione
5-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidine-1-carbonyl]-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
5-[1-(3-phenoxypropyl)-1H-1,2,3-triazol-4-yl]pyrimidine
methyl 4-(3,5-dimethyl-1-benzofuran-2-yl)-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxylate
(3S,5R)-N-(cyclohexylmethyl)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidine-1-carboxamide
[1-(1-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidin-4-yl)piperidin-3-yl]methanol
5-[1-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-3-yl]-4-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1,3-thiazol-2-amine
9-(3-hydroxypyridine-2-carbonyl)-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
3-{imidazo[1,2-a]pyridin-2-yl}-N-[2-(1H-indol-1-yl)ethyl]-N-methylpropanamide
1-(3-{[ethyl(2-methylprop-2-en-1-yl)amino]methyl}phenoxy)-3-(4-ethylpiperazin-1-yl)propan-2-ol
2-{4-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]methanesulfonamide
4-(4-fluorophenyl)-1-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}butan-1-one
(4aS,8aR)-6-(1-aminocyclopropanecarbonyl)-1-[3-(methylsulfanyl)propyl]-decahydro-1,6-naphthyridin-2-one
2-chloro-4-{2-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}benzamide
4-{4-[(2,6-difluorophenyl)methyl]piperazin-1-yl}-2-[2-(2-fluorophenyl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
5-methyl-1-{3-[2-(oxolan-3-yl)-1H-imidazol-1-yl]phenyl}-1H-1,2,3,4-tetrazole
1-(4-{[(cyclohexylmethyl)amino]methyl}-2-methoxyphenoxy)-3-(diethylamino)propan-2-ol
2-{2-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-oxoethyl}-3-phenylcyclopent-2-en-1-one
1-methyl-4-({5-[3-(1H-pyrazol-1-ylmethyl)phenyl]-1,2,4-oxadiazol-3-yl}methyl)piperidine